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GI 181771

Catalog No. T15382 CAS 305366-98-7

GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.

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GI 181771, CAS 305366-98-7

Pack Size	Availability	Price/USD
1 mg	In stock	$ 195.00
5 mg	In stock	$ 448.00
10 mg	In stock	$ 658.00
25 mg	In stock	$ 987.00
50 mg	In stock	$ 1,380.00

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Purity: 95.63%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.

Molecular Weight	605.64
Formula	C34H31N5O6
CAS No.	305366-98-7

Storage

store at low temperature

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Myer JR, et al. Species- and dose-specific pancreatic responses and progression in single- and repeat-dose studies with GI181771X: a novel cholecystokinin 1 receptor agonist in mice, rats, and monkeys. Toxicol Pathol. 2014 Jan;42(1):260-74. 2. Roses AD, et al. Stimulation of cholecystokinin-A receptors with Gl181771X: a failed clinical trial that did not test the pharmacogenetic hypothesis for reduction of food intake. Clin Pharmacol Ther. 2009 Apr;85(4):362-5.

Related compound libraries

This product is contained In the following compound libraries：

GPCR Compound Library

Related Products

Related compounds with same targets

Cholecystokinin (26-33) free acid Lintitript WAY-620645 Pentagastrin CCK-A receptor inhibitor 1 Ceruletide Ammonium Salt Lorglumide sodium salt XL413 hydrochloride

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

GI 181771 305366-98-7 GPCR/G Protein cholecystokinin GI-181771 GI181771 inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.