Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | 6-8 weeks | $ 297.00 | |
25 mg | 6-8 weeks | $ 916.00 | |
50 mg | 6-8 weeks | $ 1,190.00 | |
100 mg | 6-8 weeks | $ 1,860.00 | |
1 mL * 10 mM (in DMSO) | 6-8 weeks | $ 296.00 |
Description | GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2). |
Targets&IC50 | BD1:83 nM, BD2:78 nM, BRD4:1.3-3.2 nM (kd), BRD2:0.59-2.5 nM (kd), BRD3:0.65-0.66 nM (kd) |
Molecular Weight | 394.47 |
Formula | C25H22N4O |
CAS No. | 1637770-13-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
GS-626510 1637770-13-8 Chromatin/Epigenetic Epigenetic Reader Domain GS 626510 GS626510 inhibitor inhibit