Powder: -20°C for 3 years | In solvent: -80°C for 1 year
L-798106 is a highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM). It also has micromolar activities at EP4, EP1, and EP2 receptors (Ki: 916 nM, <5000 nM, and <5000 nM at EP4, EP1, and EP2, respectively).
Description | L-798106 is a highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM). It also has micromolar activities at EP4, EP1, and EP2 receptors (Ki: 916 nM, >5000 nM, and >5000 nM at EP4, EP1, and EP2, respectively). |
Targets&IC50 | EP1/2 receptor:> 5000 nM(ki), EP3 receptor: 0.3 nM(ki), EP4 receptor:916 nM(ki) |
Synonyms | CM9, GW671021 |
Molecular Weight | 536.44 |
Formula | C27H22BrNO4S |
CAS No. | 244101-02-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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L-798106 244101-02-8 GPCR/G Protein Immunology/Inflammation Prostaglandin Receptor CM-9 CM9 L798106 GW 671021 CM 9 GW-671021 GW671021 L 798106 inhibitor inhibit