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Lafutidine

Catalog No. T0081   CAS 118288-08-7
Synonyms: FRG-8813

Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.

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Lafutidine Chemical Structure
Lafutidine, CAS 118288-08-7
Pack Size Availability Price/USD Quantity
25 mg In stock $ 41.00
50 mg In stock $ 66.00
100 mg In stock $ 98.00
1 mL * 10 mM (in DMSO) In stock $ 50.00
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Purity: 99.94%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.
Synonyms FRG-8813
Molecular Weight 431.55
Formula C22H29N3O4S
CAS No. 118288-08-7

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: < 1 mg/mL (insoluble or slightly soluble)

DMSO: 80 mg/mL (185.4 mM)

Ethanol: 11 mg/mL (25.5 mM)

TargetMolReferences and Literature

1. Kim EH, et al. Dig Dis Sci. 2014 Dec 23.

Related compound libraries

This product is contained In the following compound libraries:
Anti-Cancer Clinical Compound Library Anti-Neurodegenerative Disease Compound Library Anti-Cancer Drug Library Anti-Cancer Approved Drug Library Bioactive Compound Library Angiogenesis related Compound Library Clinical Compound Library Serotonin Receptor-Targeted Compound Library Inhibitor Library Anti-COVID-19 Compound Library

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Keywords

Lafutidine 118288-08-7 GPCR/G Protein Immunology/Inflammation Neuroscience Histamine Receptor 5-HT Receptor inhibit gastric mucus antiulcer reflux mucosal antisecretory Inhibitor histamine protective disease secretion FRG 8813 colonic FRG8813 receptor gastroesophageal FRG-8813 inhibitor

 

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