Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Masupirdine free base (SUVN-502 free base) is a potent, selective, and orally bioavailable 5-HT6 receptor antagonist with a Ki of 2.04 nM for the human 5-HT6 receptor, demonstrating high selectivity over the 5-HT2A receptor and other 100 target sites. It is also brain penetrant and has potential for the treatment of Alzheimer's disease.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | In stock | $ 1,520.00 | |
50 mg | In stock | $ 1,980.00 | |
100 mg | In stock | $ 2,500.00 |
Description | Masupirdine free base (SUVN-502 free base) is a potent, selective, and orally bioavailable 5-HT6 receptor antagonist with a Ki of 2.04 nM for the human 5-HT6 receptor, demonstrating high selectivity over the 5-HT2A receptor and other 100 target sites. It is also brain penetrant and has potential for the treatment of Alzheimer's disease. |
Targets&IC50 | 5-HT6 receptor:2.04 nM (ki) |
Synonyms | SUVN-502 free base |
Molecular Weight | 478.4 |
Formula | C21H24BrN3O3S |
CAS No. | 701205-60-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Masupirdine free base 701205-60-9 GPCR/G Protein Neuroscience 5-HT Receptor SUVN502 SUVN 502 Masupirdine SUVN-502 free base SUVN-502 inhibitor inhibit