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NVP-BHG712 isomer

Catalog No. T19487 CAS 2245892-85-5

NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.

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NVP-BHG712 isomer, CAS 2245892-85-5

Pack Size	Availability	Price/USD
1 mg	In stock	$ 36.00
2 mg	In stock	$ 51.00
5 mg	In stock	$ 80.00
10 mg	In stock	$ 153.00
25 mg	In stock	$ 273.00
50 mg	In stock	$ 396.00
100 mg	In stock	$ 589.00
1 mL * 10 mM (in DMSO)	In stock	$ 89.00

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Purity: 99.65%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
Targets&IC50	EphA2:163 nM
In vitro	NVP-BHG712 isomer exhibits IC50 of 163 nM and 1660 nM for EPHA2 and EPHA4, respectively[1].

Molecular Weight	503.48
Formula	C26H20F3N7O
CAS No.	2245892-85-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 50 mg/mL (99.31 mM), Sonification is recommended.

H2O: insoluble

References and Literature

1. Tröster A, et al. NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family. ChemMedChem. 2018 Aug 20;13(16):1629-1633.

Related compound libraries

This product is contained In the following compound libraries：

Kinase Inhibitor Library Tyrosine Kinase Inhibitor Library Bioactive Compounds Library Max NO PAINS Compound Library Bioactive Compound Library

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Related compounds with same targets

KYL acetate(676657-00-4 free base) Tesevatinib NVP-BHG712 Sitravatinib 123C4 AZ12672857 Ehp-inhibitor-2 ALW-II-49-7

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

NVP-BHG712 isomer 2245892-85-5 Tyrosine Kinase/Adaptors Ephrin Receptor NVP BHG712 isomer Inhibitor NVPBHG712 isomer inhibit NVP-BHG-712 isomer inhibitor

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