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Nitrobenzylthioinosine

Catalog No. T8551   CAS 38048-32-7
Synonyms: NBMPR

Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.

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Nitrobenzylthioinosine Chemical Structure
Nitrobenzylthioinosine, CAS 38048-32-7
Pack Size Availability Price/USD Quantity
2 mg In stock $ 36.00
5 mg In stock $ 57.00
10 mg In stock $ 84.00
25 mg In stock $ 139.00
50 mg In stock $ 198.00
100 mg In stock $ 328.00
500 mg In stock $ 789.00
1 mL * 10 mM (in DMSO) In stock $ 71.00
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Purity: 99.87%
Purity: 98.83%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Synonyms NBMPR
Molecular Weight 419.41
Formula C17H17N5O6S
CAS No. 38048-32-7

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 25 mg/mL (59.61 mM)

TargetMolReferences and Literature

1. P J Marangos, et al. [3H]nitrobenzylthioinosine is a photoaffinity probe for adenosine uptake sites in brain. Eur J Pharmacol. 1982 Dec 3;85(3-4):359-60. 2. C M Anderson, et al. Ability of nitrobenzylthioinosine to cross the blood-brain barrier in rats. Neurosci Lett. 1996 Nov 29;219(3):191-4.

TargetMolCitations

1. Wang H, Shao Z, Xu Z, et al. Antiproliferative and apoptotic activity of gemcitabine-lauric acid conjugate on human bladder cancer cells. Iranian Journal of Basic Medical Sciences. 2022, 25(4): 536 2. Teng H, Wang Y, Sui X, et al.Gut microbiota-mediated nucleotide synthesis attenuates the response to neoadjuvant chemoradiotherapy in rectal cancer.Cancer Cell.2022

Related compound libraries

This product is contained In the following compound libraries:
Anti-Viral Compound Library Neuronal Signaling Compound Library Nucleotide Compound Library Bioactive Compounds Library Max Neurotransmitter Receptor Compound Library GPCR Compound Library Bioactive Compound Library NO PAINS Compound Library Anti-Infection Compound Library Inhibitor Library

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
Using the equation C1V1 = C2V2, where C1=10 mM, C2=50 μM, V2=20 ml and V1 is the unknown:
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Nitrobenzylthioinosine 38048-32-7 GPCR/G Protein Neuroscience AChR Adenosine Receptor Inhibitor adenosine neuroprotective P1 receptor BBB inhibit ENT1 NBMPR probe transporter photoaffinity inhibitor

 

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