1
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6940 | PHA-767491 hydrochloride | CAY10572 , PHA-767491 , PHA767491 HCl , CAY-10572 hydrochloride | GSK-3 , Apoptosis , CDK |
PHA-767491 hydrochloride (CAY-10572 hydrochloride) is an effective ATP-competitive dual Cdc7/CDK9 inhibitor (IC50: 10/34 nM). It has ~20-fold selectivity against GSK3-β and CDK1/2, 50-fold selectivity against CDK5 and MK... |