Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PROTAC BRD4 Degrader-1 is an efficacious degrader of BRD4(BRD4 BD1,IC50 of 41.8 nM).
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Description | PROTAC BRD4 Degrader-1 is an efficacious degrader of BRD4(BRD4 BD1,IC50 of 41.8 nM). |
Targets&IC50 | BRD4 BD1:41.8 nM |
In vitro | PROTAC BRD4 Degrader-1 shows high inhibitory activity against the growth of human monocyte lymphoma cell line THP-1(IC50 value of 0.81 μM), and moderate activity against Raji and HL-60 cell lines[1] |
Molecular Weight | 771.78 |
Formula | C40H37N9O8 |
CAS No. | 2133360-00-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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PROTAC BRD4 Degrader-1 2133360-00-4 Chromatin/Epigenetic Epigenetic Reader Domain PROTAC BRD4 Degrader1 PROTAC BRD-4 Degrader-1 PROTAC BRD4 Degrader 1 inhibitor inhibit