Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Pixantrone dimaleate (Pixantrone Maleate) (BBR 2778 dimaleate) is an experimental antineoplastic drug.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 47.00 | |
10 mg | In stock | $ 72.00 | |
25 mg | In stock | $ 133.00 | |
50 mg | In stock | $ 228.00 | |
100 mg | In stock | $ 347.00 | |
500 mg | In stock | $ 825.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 59.00 |
Description | Pixantrone dimaleate (Pixantrone Maleate) (BBR 2778 dimaleate) is an experimental antineoplastic drug. |
Kinase Assay | Recombinant RT enzymes are expressed, purified, and assessed for inhibition by Efavirenz (L-743726). Ki and Kii values are determined for each enzyme tested. The wild-type RT exhibited exclusively noncompetitive inhibition kinetics (data not shown), and, therefore, the Ki and Kii values are identical. Pure noncompetitive inhibition is not assumed for the mutant enzymes, and, hence, the values of both Ki and Kii are obtained from the linear mixed-type inhibition equation. The two- to threefold differences between the Ki and Kii values probably reflect a small contribution of competitive inhibition with the mutant RTs[1]. |
Synonyms | BBR-2778, Pixantrone Maleate, BBR 2778 dimaleate |
Molecular Weight | 557.21 |
Formula | C25H27N5O10 |
CAS No. | 144675-97-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 91 mg/mL(163.3 mM)
You can also refer to dose conversion for different animals. More
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Pixantrone dimaleate 144675-97-8 DNA Damage/DNA Repair Topoisomerase K562 cell BBR 2778 inhibit Inhibitor intercalator MDCK cell Pixantrone Dimaleate Pixantrone BBR-2778 Pixantrone Maleate BBR2778 Dimaleate BBR-2778 Dimaleate anti-tumor BBR 2778 dimaleate BBR 2778 Dimaleate BBR2778 DNA inhibitor