Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RORγt Inverse agonist 6 is an agonist of RORγt inverse. RORγt Inverse agonist 6 can be used in research on Th17-driven autoimmune diseases.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 158.00 | |
5 mg | In stock | $ 397.00 | |
10 mg | In stock | $ 589.00 | |
25 mg | In stock | $ 945.00 | |
50 mg | In stock | $ 1,280.00 | |
100 mg | In stock | $ 1,730.00 | |
500 mg | In stock | $ 3,460.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 493.00 |
Description | RORγt Inverse agonist 6 is an agonist of RORγt inverse. RORγt Inverse agonist 6 can be used in research on Th17-driven autoimmune diseases. |
In vivo | RORγt Inverse agonist 6 (30 mg/kg; p.o.) inhibits the expression level of IL-17A by 59% compared to the vehicle after the oral administration at the tested dose. RORγt Inverse agonist 6 suppresses IL-17A gene expression by IL-23 stimulation in a mouse pharmacodynamics model. RORγt Inverse agonist 6 (1 mg/kg; p.o.) exhibits improved drug exposure with AUC of 1289 ng h/mL[1]. |
Molecular Weight | 565.02 |
Formula | C28H29ClN6O5 |
CAS No. | 1887161-80-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (79.64 mM), Sonification is recommended.
You can also refer to dose conversion for different animals. More
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RORγt Inverse agonist 6 1887161-80-9 Metabolism ROR Inhibitor RORγt Inverse agonist-6 inhibit RAR-related orphan receptor RORγt Inverse agonist6 RORrt Inverse agonist 6 RORgammat Inverse agonist 6 inhibitor