keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 225.00 | |
5 mg | In stock | $ 488.00 | |
10 mg | In stock | $ 712.00 | |
25 mg | In stock | $ 1,090.00 | |
50 mg | In stock | $ 1,480.00 | |
100 mg | In stock | $ 1,980.00 | |
500 mg | In stock | $ 3,970.00 |
Description | RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM). |
Targets&IC50 | CB2:Ki = 50 nM |
Molecular Weight | 1484.71 |
Formula | C67H109N19O19 |
CAS No. | TP1939L1 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Insoluble
H2O: 10 mM
You can also refer to dose conversion for different animals. More
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RVD-Hpα acetate(1193362-76-3 free base) TP1939L1 GPCR/G Protein Cannabinoid Receptor RVD-Hpalpha acetate(1193362-76-3 free base) RVD Hpα acetate(1193362 76 3 free base) RVD-Hpa acetate(1193362-76-3 free base) RVDHpα acetate(1193362763 free base) inhibitor inhibit