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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2118 | SC-514 | GK 01140 | CDK , IκB/IKK , p38 MAPK , Serine Protease , Aurora Kinase |
SC-514 (GK 01140) is a selective, orally active, ATP-competitive IKK-2 inhibitor (IC50=11.2±4.7 μM), obstructs NF-κB-dependent gene expression. |