Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SGC-SMARCA-BRDVIII is a potent and selective inhibitor of SMARCA2, SMARCA4, PB1(2), PB1(3) and PB1(5) with Kds of 35 nM, 36 nM, 3.7 μM, 2.0 μM and 13 nM, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 39.00 | |
2 mg | In stock | $ 54.00 | |
5 mg | In stock | $ 64.00 | |
10 mg | In stock | $ 108.00 | |
25 mg | In stock | $ 247.00 | |
50 mg | In stock | $ 397.00 | |
100 mg | In stock | $ 589.00 | |
500 mg | In stock | $ 1,280.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 105.00 |
Description | SGC-SMARCA-BRDVIII is a potent and selective inhibitor of SMARCA2, SMARCA4, PB1(2), PB1(3) and PB1(5) with Kds of 35 nM, 36 nM, 3.7 μM, 2.0 μM and 13 nM, respectively. |
Targets&IC50 | SMARCA2:35 nM, SMARCA4:36 nM, PB1(5):13 nM, PB1(2):3.7 μM, PB1(3):2.0 μM |
In vitro | SGC-SMARCA-BRDVIII blocks adipogenesis in 3T3-L1 murine fibroblasts[1]. |
Molecular Weight | 371.43 |
Formula | C19H25N5O3 |
CAS No. | 1997319-84-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL(134.61 mM)
Ethanol: 5 mg/mL(13.46 mM)
You can also refer to dose conversion for different animals. More
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SGC-SMARCA-BRDVIII 1997319-84-2 Chromatin/Epigenetic Epigenetic Reader Domain adipogenesis SMARCA2/4 inhibit PB1 SGCSMARCABRDVIII Inhibitor SGC SMARCA BRDVIII inhibitor