Powder: -20°C for 3 years | In solvent: -80°C for 1 year
WM-8014 (MOZ-IN-3) is an inhibitor of MOZ(IC50=55 nM), a member of histone acetyltransferases.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 52.00 | |
2 mg | In stock | $ 75.00 | |
5 mg | In stock | $ 117.00 | |
10 mg | In stock | $ 178.00 | |
25 mg | In stock | $ 352.00 | |
50 mg | In stock | $ 523.00 | |
100 mg | In stock | $ 757.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 138.00 |
Description | WM-8014 (MOZ-IN-3) is an inhibitor of MOZ(IC50=55 nM), a member of histone acetyltransferases. |
Targets&IC50 | MOZ:55 nM |
In vitro | MOZ-IN-3is an inhibitor of MOZ(IC50=55 nM). MOZ-IN-3 causes cell senescence(IC50=1.6 μM) and suppresses the proliferation(IC50=551 nM). |
Kinase Assay | Reactions are set up with Acetyl coenzyme A (AcCoA)(0.4 μM), N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin)(50 nM), MOZ enzyme(10 nM), and an acetyl-lysine specific antibody (final dilution 1: 10000). |
Synonyms | MOZ-IN-3 |
Molecular Weight | 384.42 |
Formula | C20H17FN2O3S |
CAS No. | 2055397-18-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL
You can also refer to dose conversion for different animals. More
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WM-8014 2055397-18-5 Chromatin/Epigenetic Histone Acetyltransferase HAT inhibit Inhibitor HATs WM 8014 MOZ-IN-3 WM8014 inhibitor