Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist. It has a strong activating effect on rat GPR35 and a certain activating effect on human GPR35. It reduces vascular remodeling through anti-proliferative and pro-apoptotic effects.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 32.00 | |
10 mg | In stock | $ 55.00 | |
25 mg | In stock | $ 97.00 | |
50 mg | In stock | $ 172.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 39.00 |
Description | Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist. It has a strong activating effect on rat GPR35 and a certain activating effect on human GPR35. It reduces vascular remodeling through anti-proliferative and pro-apoptotic effects. |
Molecular Weight | 271.27 |
Formula | C13H13N5O2 |
CAS No. | 37762-06-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 30 mg/ml (110.59 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Zaprinast 37762-06-4 Metabolism PDE inhibit Phosphodiesterase (PDE) Inhibitor M&B 22948 inhibitor