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Cat.No. Product Name Information Area
T4495 dBET1 dBET1 is a hybrid molecule that combines (+)-JQ1 and thalidomide. It induces cereblon... Others
T5130 dBET6 dBET6 is a selective and cell-permeable degrader of BET based on PROTAC (IC50: 14 nM)... Others
T4697 ABBV-744 ABBV-744 is a BDII-selective BET bromodomain inhibitor that inhibits BRD2/3/4. It is ...
T6026 CPI-203 CPI-203 is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4). Cancer
TL0007 Bisdemethoxycurcumin Bisdemethoxycurcumin (BDMC) is a natural demethoxy derivative of curcumin. It is a po...
T4365 FL-411 FL-411 is a potent and selective BRD4 inhibitor with an IC50 of 0.43±0.09 μM for BRD4... Cancer
T6389 Anacardic Acid Anacardic Acid is an effective inhibitor of p300 and p300/CBP-associated factor histo... Cancer
T4345 CeMMEC1 CeMMEC1 is an inhibitor of BRD4, and also has a great affinity for TAF1(IC50=0.9 μM).
T3504 AZD5153 6-Hydroxy-2-naphthoic acid AZD 5153 is an orally available, bivalent inhibitor of the bromodomain and extratermi...
T3712 Mivebresib Mivebresib, also known as ABBV-075, is a potent BET inhibitor (bromodomain (BRD)-cont... Cancer
T3311 GSK6853 GSK6853 is a potent, soluble, cell-active, and highly selective inhibitor of the BRPF... Others
T6939 PFI-3 A small molecule FAK kinase inhibitor, GSK2256098, inhibits growth and survival of pa... Others
T6859 I-BRD9 I-BRD9 is the first selective cellular inhibitor for BRD9 with pIC50 of 7.3. others
T6811 CPI-637 CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibit... Others
T6786 BI-9564 BI-9564, a specific cell-permeable BRD9 BD inhibitor. The Kd for BRD9 is 5.9 nM, and ... others
T6783 BI-7273 BI-7273 is an effective, specific, BRD9 BD Inhibitor, which can infiltrate cell. Others
T6668 SGC-CBP30 SGC-CBP30 is an effective CREBBP/EP300 inhibitor (IC50: 21/38 nM). Cancer
T6255 Bromosporine Bromosporine is a broad spectrum inhibitor for bromodomains for BRD2/4/9 and CECR2 (I... others
T6222 PFI-1 PFI-1, a specific BET (bromodomain-containing protein) inhibitor for BRD4, is with th... Cancer
T6032 Birabresib Birabresib is a synthetic, small molecule inhibitor of the BET (Bromodomain and Extra... Cancer
T6021 GSK1324726A GSK1324726A is a greatly specific inhibitor of BET family proteins for BRD2(IC50=41 n... Cancer
T2480 Apabetalone RVX-208, an effective BET bromodomain inhibitor,has been investigated for the treatme... Cancer
T2436 GSK2801 GSK2801 is an effective, specific and cell active acetyl-lysine competitive inhibitor... Cancer
T2379 UNC1215 UNC1215, an effective and specific MBT (malignant brain tumor) antagonist, binds L3MB... Cancer
T2252 UNC669 UNC669 is an effective and specific MBT (malignant brain tumor) inhibitor with IC50 o... Other
T2110 (+)-JQ-1 (+)-JQ1, a BET bromodomain inhibitor, binds to all bromodomains of the BET family. Other
T2091 CPI-0610 CPI-0610 is an effective, specific, and cell-active BET bromodomain inhibitor CPI-061... Other
T2072 BET bromodomain inhibitor BET bromodomain inhibitor is a potent BET inhibitor. Other
T1906 Molibresib GSK 525762A (I-BET 762) is an inhibitor of BET proteins (IC50: about 35 nM). Immunology