Histone-Methyltransferase

Cat.No.	Product Name	Information	Area
T7089	SGC2085	SGC2085 is an effective and selective coactivator-associated arginine methyltransfera...
T4583	(R)-PFI-2 hydrochloride	PFI-2 hydrochloride is a potent, highly selective, and cell-active inhibitor of the m...
T4393	MS049 2HCl (1502816-23-0(free base))	MS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 4...
T4378	MS049	MS 049 is a potent, selective, and cell-active dual inhibitor of PRMT4 and PRMT6 with...
T4343	A-196	A-196 is a potent and selective inhibitor of SUV420 h1 and SUV420 h2 with IC50 values...
T4334	EPZ020411 2HCl (1700663-41-7(free base))	EPZ020411 is an effective and specific small molecule PRMT6 inhibitor (IC50=10 nM).	Cancer
T4314	EPZ020411	EPZ020411 is a specific and effective inhibitor of PRMT6 (IC50=10 nM).	cancer
T3624	A-366	Potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50?= 3.3 n...
T3084	SGC707	SGC707 is a potent, selective, and cell-active allosteric inhibitor of PRMT3.	Others
T6916	OICR-9429	OICR-9429 is a potent antagonist of the interaction that WDR5 effect with peptide reg...	Others
T6900	MS023	MS023 is a potent, selective, and cell-active Type I PRMT inhibitor with IC50 of 30 n...	Others
T6879	LLY-507	LLY-507 is an effective, cell-active, and specific inhibitor of protein-lysine Methyl...	Others
T6857	HLCL-61 hydrochloride	HLCL-61 hydrochloride is a potent and selective PRMT5 inhibitor for the treatment of ...	Others
T6853	GSK591	GSK591，Alternative Names are EPZ015866, GSK3203591， is a potent selective inhibitor o...	Others
T6810	CPI-360	CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 ...	Others
T6809	CPI-169	CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and ...	Others
T6803	Chaetocin	Chaetocin, a natural product from Chaetomium species, is a histone methyltransferase ...	Others
T3257	UNC0638	UNC0638 is an inhibitor of β-protein lysine methyltransferases G9a(IC50<15 nM) and GL...
T3201	WDR5-0103	WDR5-0103 is an effective and specific WD repeat-containing protein 5 (WDR5) antagoni...	Cancer
T6484	EI1	EI1 is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (W...
T2649	MI-2	MI-2 (Menin-MLL Inhibitor) is a potent menin-MLL interaction inhibitor with IC50 of 4...	Cancer
T2643	MI-3	MI-3 (Menin-MLL Inhibitor) is an effective inhibitor of Menin-MLL interaction (IC50: ...	Cancer
T6076	EPZ015666	EPZ015666 is an orally available inhibitor of PRMT5 enzymatic activity.	Cancer
T6059	GSK343	GSK343，a specific and effective EZH2 inhibitor (IC50=4 nM), exhibits 60 fold specific...	Cancer
T3099	Pinometostat	EPZ5676 has been used in trials studying the treatment of Leukemia, Acute Leukemias, ...	Cancer
T3082	SGC0946	SGC0946 is a highly effective and specific DOT1L methyltransferase inhibitor (IC50: 0...	Cancer
T3081	EPZ004777	EPZ004777 is a potent, selective?DOT1L?inhibitor with?IC50?of 0.4 nM.
T3057	UNC1999	UNC1999 is a orally bioavailable, effective and specific inhibitor of EZH2 (IC50=2 nM...	Cancer
T2435	EPZ011989	EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM ...	Cancer
T2354	UNC0631	UNC0631 is a effectvie histone methyltransferase G9a inhibitor (IC50=4 nM).	Other

Home 1 2 Last