T72180 |
Acetyl-CoA Carboxylase-IN-1
|
|
|
|
Acetyl-CoA Carboxylase-IN-1 是一种有效的乙酰辅酶 A 羧化酶 (ACC) 抑制剂,IC50值为 <5 nM。 Acetyl-CoA Carboxylase-IN-1 具有抗菌活性。 |
T7163 |
PF-05175157
|
|
Acetyl-CoA Carboxylase
|
|
PF 05175157 是一种广谱的乙酰辅酶 A 羧化酶 (ACC) 抑制剂,对 ACC1 (human),ACC2 (human), ACC1 (rat) 和 ACC2 (rat) 具有抑制作用,IC50分别为 27.0, 33.0, 2... |
T3988 |
TOFA
|
RMI14514,MDL14514 |
Acetyl-CoA Carboxylase
|
|
TOFA 是有效的乙酰辅酶 A 羧化酶-α (ACCA)的变构抑制剂。 |
T7184 |
Firsocostat
|
NDI-010976,ND-630,GS-0976 |
Acetyl-CoA Carboxylase
|
|
ND-630 是有效的乙酰辅酶A 羧化酶 (ACC) 抑制剂,抑制人类 ACC1 和 ACC2 的IC50分别为2.1和6.1 nM。 |
T1889 |
CP-640186
|
CP 640186 |
Acetyl-CoA Carboxylase
|
|
CP 640186 是一种有效的乙酰辅酶 A 羧化酶 (ACC)抑制剂,抑制大鼠肝脏 ACC1 和大鼠骨骼肌 ACC2 的 IC50分别为 53 nM 和 61 nM。 |
T14991 |
CMS-121
|
CMS121 |
Acetyl-CoA Carboxylase
|
|
CMS-121 是喹诺酮衍生物,对乙酰辅酶 A 羧化酶 1 具有抑制作用,具有口服活性。CMS-121具有保护 HT22 细胞免受缺血和氧化损伤的活性,EC50分别为7 nM 和200 nM。CMS-121具有强大的抗炎,抗氧化,神经保护和... |
T3622 |
CP-640186 hydrochloride
|
CP 640186 HCl,盐酸CP-640186 |
Acetyl-CoA Carboxylase
|
|
CP-640186 hydrochloride 是膜渗透性的乙酰辅酶A 羧化酶(ACC)抑制剂,抑制大鼠肝脏ACC1和大鼠骨骼肌ACC2的IC50为53 nM 和61 nM。 |
T3510 |
Olumacostat Glasaretil
|
|
Acetyl-CoA Carboxylase
|
|
Olumacostat glasaretil 是乙酰辅酶A 羧化酶的有效抑制剂。 |
TQ0243 |
ND-646
|
|
Acetyl-CoA Carboxylase
|
|
ND-646 是乙酰辅酶 A 羧化酶(ACC)抑制剂,对重组 hACC1 和 hACC2的IC50分别为 3.5 nM 和 4.1 nM。 |
T5046 |
Haloxyfop
|
Haloxyfop Acid,(±)-Haloxyfop,吡氟氯禾灵 |
Others
,
Acetyl-CoA Carboxylase
|
|
Haloxyfop 是有效的芳氯氧苯氧丙酸除草剂,广泛应用于阔叶作物的野草。对玉米幼苗叶绿体中乙酰辅酶 A 羧化酶 (EC 6.4.1.2) 具有抑制作用,IC50为 0.5 μM,而对豌豆中该酶无影响。 |
T9209 |
PF-05221304
|
STAT5 Inhibitor III,R 6238,,Clesacostat,NSC 170984 |
Acetyl-CoA Carboxylase
|
|
PF-05221304 是一种具有口服活性的肝脏靶向乙酰辅酶A 羧化酶 (ACC) 抑制剂,ACC 是脂肪酸合成的限速酶。 |
T4309 |
CIL56
|
CA3 |
ROS
,
Ferroptosis
|
|
CIL56 是一种选择性铁死亡诱导剂,可通过产生铁依赖性活性氧来诱导细胞铁死亡。 |
T12062 |
MK-4074
|
|
Others
|
|
MK-4074 is a liver-specific acetyl-CoA carboxylase ACC1 and ACC2 inhibitor(IC50 of 3 nM). |
T70663 |
ND-654
|
|
|
|
ND-654 is an acetyl CoA carboxylase inhibitor. |
T69277 |
(±)-Diclofop
|
|
|
|
(±)-Diclofop is an Acetyl-CoA carboxylase (ACCase) inhibiting herbicide. |
T20135 |
Diphenamid
|
Caswell No. 395,Enide 50W,Fenam,Trefmid,Enide 50,Rideon |
|
|
Diphenamid is a chemical compound from the group of acetamides and a herbicide. The effect is based on the inhibition of... |
T36785 |
Fluazifop-P-butyl
|
|
|
|
Fluazifop-P-butyl is an arylophenoxypropionate group graminicide that functions as an inhibitor of acetyl-CoA carboxylas... |
T61430 |
S-2E
|
|
|
|
S-2E is a compound that functions as an orally active, noncompetitive inhibitor of both HMG-CoA reductase and acetyl-CoA... |
T38473 |
Malonyl Coenzyme A lithium
|
|
|
|
Malonyl Coenzyme A (lithium) is a coenzyme A derivative that is utilized in fatty acid and polyketide synthesis and in t... |
T40675 |
CP-610431
|
|
|
|
CP-610431 is a reversible, ATP-uncompetitive inhibitor of acetyl-CoA carboxylase (ACC), exhibiting isozyme nonselectivit... |