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Search Results for "ck1 inhibitor"

Libraries

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Reagents



Compounds

Cat No. Product Name
T21915 TBCA Casein Kinase II Inhibitor III, TBCA Casein Kinase
TBCA is a highly selective CK2 (casein kinase II) inhibitor, IC50 = 110 nM, Ki = 77 nM. TBCA shows selectivity for CK2 o...
T60005 WAY-296817 Casein Kinase
WAY-296817 is casein kinase 1 (CK1) inhibitor and can be used for research on the treatment or prevention of diseases as...
T8987 Epiblastin A Casein Kinase
Epiblastin A is an inhibitor of Casein Kinase 1 (CK1). Epiblastin A engages CK1 isoenzymes in cell lysate and induces ef...
T5393 CK1-IN-1 PUN51207 Casein Kinase , p38 MAPK
CK1-IN-1, compound 1c reported in patent WO2015119579A1, is a casein kinase 1 (CK1) inhibitor. It has IC50s of 15 nM, 16...
T23224 (R)-DRF053 dihydrochloride Others
cdk/CK1 inhibitor,potent and ATP-competitive
T6745 5-Iodotubercidin 5-ITu , NSC 113939 Adenosine Receptor
5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, ins...
T2440 IC261 SU-5607 Casein Kinase , Apoptosis , CDK
IC261 is a novel inhibitor of CK1, triggers the mitotic checkpoint control. The IC50 of IC261 for CK1 was 16 μM and for ...
T2449 D4476 D 4476 , Casein Kinase I Inhibitor Casein Kinase , Apoptosis , ALK , Autophagy
D4476 is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).
T4645 TA-01 Casein Kinase , p38 MAPK , Autophagy
TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respecti...
T16141 MRT00033659 Others
MRT00033659 is an effective broad-spectrum kinase inhibitor of CK1 (IC50=0.9 µM for CK1δ) and CHK1 (IC50=0.23 µM). MRT00...
T10829 CKI-7 free base CKI-7 Casein Kinase
CKI-7 free base is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selecti...
T19913 CKI-7 CKI-7 2HCl , CKI7 2HCl , CKI 7 2HCl , CKI7 dihydrochloride , CKI 7 dihydrochloride , CKI-7 dihydrochloride ROCK , SGK , Casein Kinase , S6 Kinase , CDK
CKI-7 2HCl is an inhibitor of casein kinase 1 (CK1).
T22884 JW 67 Wnt/beta-catenin
inhibitor of canonical Wnt pathway signaling
TBCA
T21915
synonym: Casein Kinase II Inhibitor III, TBCA
Target:
WAY-296817
T60005
synonym:
Target:
Epiblastin A
T8987
synonym:
Target:
CK1-IN-1
T5393
synonym: PUN51207
Target:
(R)-DRF053 dihydrochloride
T23224
synonym:
Target:
5-Iodotubercidin
T6745
synonym: 5-ITu , NSC 113939
Target:
IC261
T2440
synonym: SU-5607
Target:
D4476
T2449
synonym: D 4476 , Casein Kinase I Inhibitor
Target:
TA-01
T4645
synonym:
Target:
MRT00033659
T16141
synonym:
Target:
CKI-7 free base
T10829
synonym: CKI-7
Target:
CKI-7
T19913
synonym: CKI-7 2HCl , CKI7 2HCl , CKI 7 2HCl , CKI7 dihydrochloride , CKI 7 dihydrochloride , CKI-7 dihydrochloride
Target:
JW 67
T22884
synonym:
Target: