T21915 |
TBCA
|
Casein Kinase II Inhibitor III, TBCA |
Casein Kinase
|
|
TBCA is a highly selective CK2 (casein kinase II) inhibitor, IC50 = 110 nM, Ki = 77 nM. TBCA shows selectivity for CK2 o... |
T60005 |
WAY-296817
|
|
Casein Kinase
|
|
WAY-296817 is casein kinase 1 (CK1) inhibitor and can be used for research on the treatment or prevention of diseases as... |
T8987 |
Epiblastin A
|
|
Casein Kinase
|
|
Epiblastin A is an inhibitor of Casein Kinase 1 (CK1). Epiblastin A engages CK1 isoenzymes in cell lysate and induces ef... |
T5393 |
CK1-IN-1
|
PUN51207 |
Casein Kinase
,
p38 MAPK
|
|
CK1-IN-1, compound 1c reported in patent WO2015119579A1, is a casein kinase 1 (CK1) inhibitor. It has IC50s of 15 nM, 16... |
T23224 |
(R)-DRF053 dihydrochloride
|
|
Others
|
|
cdk/CK1 inhibitor,potent and ATP-competitive |
T6745 |
5-Iodotubercidin
|
5-ITu , NSC 113939 |
Adenosine Receptor
|
|
5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, ins... |
T2440 |
IC261
|
SU-5607 |
Casein Kinase
,
Apoptosis
,
CDK
|
|
IC261 is a novel inhibitor of CK1, triggers the mitotic checkpoint control. The IC50 of IC261 for CK1 was 16 μM and for ... |
T2449 |
D4476
|
D 4476 , Casein Kinase I Inhibitor |
Casein Kinase
,
Apoptosis
,
ALK
,
Autophagy
|
|
D4476 is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay). |
T4645 |
TA-01
|
|
Casein Kinase
,
p38 MAPK
,
Autophagy
|
|
TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respecti... |
T16141 |
MRT00033659
|
|
Others
|
|
MRT00033659 is an effective broad-spectrum kinase inhibitor of CK1 (IC50=0.9 µM for CK1δ) and CHK1 (IC50=0.23 µM). MRT00... |
T10829 |
CKI-7 free base
|
CKI-7 |
Casein Kinase
|
|
CKI-7 free base is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selecti... |
T19913 |
CKI-7
|
CKI-7 2HCl , CKI7 2HCl , CKI 7 2HCl , CKI7 dihydrochloride , CKI 7 dihydrochloride , CKI-7 dihydrochloride |
ROCK
,
SGK
,
Casein Kinase
,
S6 Kinase
,
CDK
|
|
CKI-7 2HCl is an inhibitor of casein kinase 1 (CK1). |
T22884 |
JW 67
|
|
Wnt/beta-catenin
|
|
inhibitor of canonical Wnt pathway signaling |