T21915 |
TBCA
|
Casein Kinase II Inhibitor III, TBCA |
Casein Kinase
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|
TBCA is a highly selective CK2 (casein kinase II) inhibitor, IC50 = 110 nM, Ki = 77 nM. TBCA shows selectivity for CK2 o... |
T60005 |
WAY-296817
|
|
Casein Kinase
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WAY-296817 is casein kinase 1 (CK1) inhibitor and can be used for research on the treatment or prevention of diseases as... |
T2008 |
LY294002
|
NSC 697286 , SF 1101 , LY 294002 |
Casein Kinase
,
DNA-PK
,
Apoptosis
,
PI3K
,
Autophagy
|
|
LY294002 is an inhibitor of PI3K (IC50s: 0.5/0.57/0.97 μM for PI3Kα/δ/β in cell-free assays). It also blocks autophagoso... |
T60295 |
Casein kinase 1δ-IN-1
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Casein kinase 1δ-IN-1 (compound 822) is an inhibitor of casein kinase 1 delta ( CK1δ ), exhibits inhibition of greater t... |
TP1509 |
Casein Kinase Substrates 3
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Casein Kinase Substrates 3 is a substrate of casein kinase. |
T9175 |
Casein Kinase inhibitor A51
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Casein Kinase inhibitor A51 is a potent and orally active casein kinase 1α (CK1α) inhibitor. Casein Kinase inhibitor A51... |
T10687L |
Casein Kinase II Inhibitor IV Hydrochloride
|
Casein Kinase II Inhibitor IV Hydrochloride (863598-09-8 free base) |
Others
|
|
Casein Kinase II Inhibitor IV Hydrochloride is a small-molecule inducer of epidermal keratinocyte differentiation. |
T11524 |
H-89
|
Protein kinase inhibitor H-89 |
Others
|
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H-89 is a selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A; IC50: 48 nM). H-89 has weak inhi... |
T60740 |
TMX-4113
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TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1... |
T21642 |
4,5,6,7-Tetrabromobenzimidazole
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4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1]. |
T60608 |
FPFT-2216
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FPFT-2216 is a “molecular glue” compound that degrades Aiolos (IKZF3), casein kinase 1α (CK1α), phosphodiesterase 6D (PD... |
T61754 |
TMX-4116
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TMX-4116 is a casein kinase 1α ( CK1α ) degrader. TMX-4116 shows the degradation preference for CK1α with DC 50 s less t... |
T8305 |
Ellagic acid (hydrate)
|
Ellagic Acid hydrate |
Antioxidant
,
Casein Kinase
|
|
Ellagic acid hydrate is a natural antioxidant and acts as a potent and ATP-competitive CK2 inhibitor (IC50:40 nM, Ki: 20... |
T39482 |
Casein Kinase inhibitor A86
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Casein Kinase inhibitor A86 is a potent and orally active casein kinase 1α (CK1α) inhibitor. Casein Kinase inhibitor A86... |
T10687 |
Casein Kinase II Inhibitor IV
|
|
Casein Kinase
|
|
Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation. |
T2449 |
D4476
|
D 4476 , Casein Kinase I Inhibitor |
Casein Kinase
,
Apoptosis
,
ALK
,
Autophagy
|
|
D4476 is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay). |
T5056 |
PF-4800567
|
|
Casein Kinase
|
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PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over ... |
T2695 |
TBB
|
4,5,6,7-tetrabromobenzotriazole , NSC 231634 , Casein Kinase II Inhibitor I |
GSK-3
,
Casein Kinase
,
CDK
|
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TBB(NSC 231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2). |
T23138 |
PF 4800567 hydrochloride
|
|
Others
|
|
casein kinase 1ε inhibitor |
T14069 |
A-3 hydrochloride
|
|
PKA
,
CaMK
,
Casein Kinase
,
PKC
|
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A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. ... |