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Search Results for "casein kinase"

Targets

Libraries

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Compounds

Cat No. Product Name
T21915 TBCA Casein Kinase II Inhibitor III, TBCA Casein Kinase
TBCA is a highly selective CK2 (casein kinase II) inhibitor, IC50 = 110 nM, Ki = 77 nM. TBCA shows selectivity for CK2 o...
T60005 WAY-296817 Casein Kinase
WAY-296817 is casein kinase 1 (CK1) inhibitor and can be used for research on the treatment or prevention of diseases as...
T2008 LY294002 NSC 697286 , SF 1101 , LY 294002 Casein Kinase , DNA-PK , Apoptosis , PI3K , Autophagy
LY294002 is an inhibitor of PI3K (IC50s: 0.5/0.57/0.97 μM for PI3Kα/δ/β in cell-free assays). It also blocks autophagoso...
T60295 Casein kinase 1δ-IN-1
Casein kinase 1δ-IN-1 (compound 822) is an inhibitor of casein kinase 1 delta ( CK1δ ), exhibits inhibition of greater t...
TP1509 Casein Kinase Substrates 3
Casein Kinase Substrates 3 is a substrate of casein kinase.
T9175 Casein Kinase inhibitor A51
Casein Kinase inhibitor A51 is a potent and orally active casein kinase 1α (CK1α) inhibitor. Casein Kinase inhibitor A51...
T10687L Casein Kinase II Inhibitor IV Hydrochloride Casein Kinase II Inhibitor IV Hydrochloride (863598-09-8 free base) Others
Casein Kinase II Inhibitor IV Hydrochloride is a small-molecule inducer of epidermal keratinocyte differentiation.
T11524 H-89 Protein kinase inhibitor H-89 Others
H-89 is a selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A; IC50: 48 nM). H-89 has weak inhi...
T60740 TMX-4113
TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1...
T21642 4,5,6,7-Tetrabromobenzimidazole
4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].
T60608 FPFT-2216
FPFT-2216 is a “molecular glue” compound that degrades Aiolos (IKZF3), casein kinase 1α (CK1α), phosphodiesterase 6D (PD...
T61754 TMX-4116
TMX-4116 is a casein kinase 1α ( CK1α ) degrader. TMX-4116 shows the degradation preference for CK1α with DC 50 s less t...
T8305 Ellagic acid (hydrate) Ellagic Acid hydrate Antioxidant , Casein Kinase
Ellagic acid hydrate is a natural antioxidant and acts as a potent and ATP-competitive CK2 inhibitor (IC50:40 nM, Ki: 20...
T39482 Casein Kinase inhibitor A86
Casein Kinase inhibitor A86 is a potent and orally active casein kinase 1α (CK1α) inhibitor. Casein Kinase inhibitor A86...
T10687 Casein Kinase II Inhibitor IV Casein Kinase
Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation.
T2449 D4476 D 4476 , Casein Kinase I Inhibitor Casein Kinase , Apoptosis , ALK , Autophagy
D4476 is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).
T5056 PF-4800567 Casein Kinase
PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over ...
T2695 TBB 4,5,6,7-tetrabromobenzotriazole , NSC 231634 , Casein Kinase II Inhibitor I GSK-3 , Casein Kinase , CDK
TBB(NSC 231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).
T23138 PF 4800567 hydrochloride Others
casein kinase 1ε inhibitor
T14069 A-3 hydrochloride PKA , CaMK , Casein Kinase , PKC
A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. ...
TBCA
T21915
synonym: Casein Kinase II Inhibitor III, TBCA
Target:
WAY-296817
T60005
synonym:
Target:
LY294002
T2008
synonym: NSC 697286 , SF 1101 , LY 294002
Target:
Casein kinase 1δ-IN-1
T60295
synonym:
Target:
Casein Kinase Substrates 3
TP1509
synonym:
Target:
Casein Kinase inhibitor A51
T9175
synonym:
Target:
Casein Kinase II Inhibitor IV Hydrochloride
T10687L
synonym: Casein Kinase II Inhibitor IV Hydrochloride (863598-09-8 free base)
Target:
H-89
T11524
synonym: Protein kinase inhibitor H-89
Target:
TMX-4113
T60740
synonym:
Target:
4,5,6,7-Tetrabromobenzimidazole
T21642
synonym:
Target:
FPFT-2216
T60608
synonym:
Target:
TMX-4116
T61754
synonym:
Target:
Ellagic acid (hydrate)
T8305
synonym: Ellagic Acid hydrate
Target:
Casein Kinase inhibitor A86
T39482
synonym:
Target:
Casein Kinase II Inhibitor IV
T10687
synonym:
Target:
D4476
T2449
synonym: D 4476 , Casein Kinase I Inhibitor
Target:
PF-4800567
T5056
synonym:
Target:
TBB
T2695
synonym: 4,5,6,7-tetrabromobenzotriazole , NSC 231634 , Casein Kinase II Inhibitor I
Target:
PF 4800567 hydrochloride
T23138
synonym:
Target:
A-3 hydrochloride
T14069
synonym:
Target:
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