T21874 |
CID 2745687
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GPR
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CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn disodium and zaprinast, two ago... |
T8329 |
AR 231453
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GPR
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AR 231453 is a selective and orally available GPR119 agonist,can stimulate β-cell replication and improve islet graft fu... |
T3433 |
TUG-891
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TUG891,TUG 891 |
GPR
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TUG-891 is a G protein-coupled receptor (GPCR) expressed in intestine, adipocytes, and pro-inflammatory macrophages that... |
T10843 |
CMF019
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Apelin receptor
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CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and ... |
T9146 |
Ms48107
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Benzenemethanol, 2-[4-amino-6-[[(4-phenoxyphenyl)methyl]amino]-1,3,5-triazin-2-yl]-3-fluoro- |
Others
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MS48107 is a potent and selective positive allosteric modulator of G protein-coupled receptor 68 (GPR68). It is selectiv... |
T50088 |
N-phenylthiophene-2-carboximidamide
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Others
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N-phenylthiophene-2-carboximidamide is an organic compound of the thiophene derivative class that has been used in the s... |
T27428 |
GP-1681
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GP1681,GP 1681 |
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GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection. |
T26962 |
CBP-307
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CBP307 |
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CBP-307 is a selective second generation S1P1 (a G-protein coupled receptor -GPCR) modulator. |
T10363 |
Arazine
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N-Acetyl-S-farnesyl-L-cysteine |
Others
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Arazine can be a a substrate for isoprenylcysteine methyltransferase by competing with prenylated G protein or its recep... |
T11044 |
Dihydromunduletone
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DHM |
GPR
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Dihydromunduletone (DHM) is a carotenoid derivative and selective strong adhesion G protein-coupled receptor (aGPCR) (GP... |
T73005 |
PF-07054894
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PF-07054894 is a potent CCR6 antagonist. PF-07054894 targets G protein-coupled receptor (GPCR). PF-07054894 can be used ... |
TN5580 |
Rediocide A
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Rediocide A, an insecticide, can inhibit calcium mobilization in Drosophila G-protein- coupled receptors (GPCR)s other t... |
T63340 |
CCG-273220
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CCG-273220 is a covalent inhibitor of G protein-coupled receptor (GPCR) kinase 5 (GRK5) (IC50: 220 nM).CCG-273220 covale... |
T70468 |
MK-8666
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MK-8666 is a partial GPCR (G-protein-coupled receptor) agonist that is coordinated with the action of GPR40. GPR40, also... |
T69953 |
MK-8666 Tris
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MK-8666 is a partial GPCR (G-protein-coupled receptor) agonist that is coordinated with the action of GPR40. GPR40, also... |
T36578 |
Boc-Lys(Ac)-AMC
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Commendamide (N-acyl-3-hydroxypalmitoyl-glycine) is a newly discovered GPCR G2A/GPR132 agonist (EC50=11.8 μM) that isola... |
T36550 |
CAY10535
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TPα and TPβ are two isoforms of the human TP receptor, the G protein-coupled receptor (GPCR) that mediates the actions o... |
T36013 |
Lysophosphatidylcholines
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Lyso-Lecithins (egg) |
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Lysophosphatidylcholines are produced by hydrolysis of the fatty acid of phosphatidylcholine at either the sn-1 or sn-2 ... |