Search Result

Search Results for "histone methyltransferase"

Targets

Libraries

Histone Modification Compound Library Methylation Compound Library Chromatin Modification Compound Library Epigenetics Compound Library Stem Cell Differentiation Compound Library Anti-COVID-19 Compound Library

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Compounds

Cat No.	Product Name
T60002	Ethyl 2-amino-4-methyl-5-[(3-nitrophenyl)carbamoyl]thiophene-3-carboxylate	DC-S239	Histone Methyltransferase
	Ethyl 2-amino-4-methyl-5-[(3-nitrophenyl)carbamoyl]thiophene-3-carboxylate is a selective inhibitor of histone methyltra...		Histone Methyltransferase
T13954	UNC6852		DNA Methyltransferase , Histone Methyltransferase
	UNC6852 contains an EED ligand (IC50 = 247 nM) and a von Hippel-Lindau ligand and is a selective polycomb repressive com...		DNA Methyltransferase , Histone Methyltransferase
T40254	MRTX-1719		Histone Methyltransferase
	MRTX-1719 is a potent, first-in-class, selective inhibitor of the PRMT5/MTA complex, with an IC50 of less than 10 nM in ...		Histone Methyltransferase
T6360	3-deazaneplanocin A HCl		Others , Histone Methyltransferase
	3-deazaneplanocin A (DZNeP)HCl, an analog of adenosine, is a competitive inhibitor of S-adenosylhomocysteine hydrolase w...		Others , Histone Methyltransferase
T4583	PFI-2 hydrochloride	(R)-PFI-2 hydrochloride , PFI-2 HCl	Histone Methyltransferase
	PFI-2 hydrochloride is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 ...		Histone Methyltransferase
T40993	Histone H3 (1-21)
	Histone H3 (1-21), derived from Histone H3 1-21 amino acids, is usually used as a substrate for methyltransferase (Histo...
T12887	SGC3027		Others
	SGC3027 is an inhibitor of histone methyltransferase,also is a first potent, selective and cell active chemical probe fo...		Others
T39861	AS-85
	AS-85 is a potent ASH1L histone methyltransferase inhibitor ( IC 50 =0.6 μM) with anti-leukemic activity. AS-85 strongly...
T36975	SETD2-IN-1 TFA
	SETD2-IN-1 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. S...
T28114	MS2177	MS-2177 , MS 2177
	MS2177 is a potent and selective inhibitor of SETD8, the only methyltransferase known to catalyze monomethylation of his...
T36576	Histone H3 (21-44)-GK-biotin (trifluoroacetate salt)
	Histone H3 (21-44)-GK-biotin is a peptide fragment of histone H3 that corresponds to amino acid residues 22-45 of the hu...
T35567	BIX01294 (hydrochloride hydrate)
	The methylation of lysine residues on histones plays a central role in determining euchromatin structure and gene expres...
T36978	AS-99 TFA
	AS-99 TFA is a first-in-class, potent and selective ASH1L histone methyltransferase inhibitor (IC50= 0.79 μM, Kd= 0.89 μ...
T6292	3-Deazaneplanocin A		Histone Methyltransferase
	3-Deazaneplanocin A (DZNep) is an attractive epigenetic anticancer agent through the inhibition of the cellular enhancer...		Histone Methyltransferase
T4314	EPZ020411	EPZ020411 2HCl	Histone Methyltransferase
	EPZ020411 is a specific and effective inhibitor of PRMT6 (IC50=10 nM).		Histone Methyltransferase
T25471	GSK-A	GSK A
	GSK-A is a Histone Lysine Methyltransferase EZH2 inhibitor.
T68613	DC-S238
	DC-S238 is a potent and selective histone methyltransferase SET7 inhibitor.
T1923	BRD4770		Histone Methyltransferase
	BRD4770 is a histone methyltransferase G9a inhibitor and induces cell senescence.		Histone Methyltransferase
T10553	BIX-01338 hydrate		Others
	BIX-01338 hydrate is an inhibitor of histone lysine methyltransferase.		Others
T71918	DC-S100
	DC-S100 is a selective histone methyltransferase SET7 inhibitor.