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Search Results for " monoamine "

Targets

192

Compounds

41

Natural Products

4

Recombinant Proteins

2

Libraries

Cat No. Product Name Synonyms Targets
T75422 Monoamine oxidase
Monoamine oxidase is an enzyme composed of different polypeptides. Monoamine oxidation catalyzes the oxidative deamination of various biological amines in brain and peripheral tissues by producing hydrogen peroxide. Mono...
T60656 Monoamine Oxidase B inhibitor 1
Monoamine Oxidase B inhibitor 1 is a potent, reversible, orally active and selective monoamine oxidase B (MAO-B) inhibitor (IC50 = 0.02 nM) that can across the blood-brain barrier (BBB). Monoamine Oxidase B inhibitor 1 s...
T60806 Monoamine Oxidase B inhibitor 2
Monoamine Oxidase B inhibitor 2 is a potent, reversible, orally active and selective inhibitor of monoamine oxidase B (MAO-B) (IC50 = 1.33 nM) which can across the blood-brain barrier (BBB). Monoamine Oxidase B inhibitor...
T61463 Monoamine oxidase/Aromatase-IN-1
Monoamine oxidase/Aromatase-IN-1 (compound 2q) is a potent dual inhibitor of monoamine oxidase (MAO) and aromatase, with IC50 values of 39 nM and 31 nM for MAO-B and aromatase, respectively. It holds significant potentia...
T4559 Isocarboxazid Monoamine Oxidase
Isocarboxazid has the formula 1-benzyl-2-(5-methyl-3-isoxazolylcarbonyl)hydrazine-isocarboxazid. It is a monoamine oxidase inhibitor.[2] It is used in the treatment of major depression, dysthymic disorder, atypical disor...
T22605 Bifemelane hydrochloride MAO , Monoamine Oxidase
Bifemelane hydrochloride is a MAO inhibitor
T8849 PF-9601N MAO
PF-9601N showed high potency and selectivity as a MAO-BI (monoamine oxidase type B inhibitor) and also demonstrated remarkable neuroprotective properties in several in vivo and cellular models of PD.
T7147 Valbenazine NBI-98854 Monoamine Transporter
Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.
T0235 Modaline sulfate MAO , Monoamine Oxidase
Modaline was a 2-methyl-3-piperidinopyrazine derivative found to inhibit monoamine oxidase (MAO) and showed a curative effect for the anti-depressant. Similar to other MAO inhibitors, it enhanced convulsions induced by t...
T12585 PXS-5153A Others , Monoamine Oxidase
PXS-5153A is an effective, selective, and fast-acting inhibitor of lysyl oxidase like 2/3 enzymes with enzymatic activity almost entirely blocked within 15 minutes. PXS-5153A could reduce crosslinks and ameliorates fibro...
T0084 Moclobemide Ro111163 MAO , Monoamine Oxidase
Moclobemide (Ro111163) is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties.
T6073 OG-L002 Histone Demethylase , Monoamine Oxidase , HSV
OG-L002 is an effective and selective LSD1 inhibitor (IC50: 20 nM), showing 69- and 36-fold selectivity over MAO-A and MAO-B, respectively.
T12584 PXS-5120A Others , Monoamine Oxidase
PXS-5120A is an irreversible fluoroallylamine Lysyl Oxidase-like 2/3 (LOXL2/3) inhibitor with anti-fibrotic activity.
T1993 J-147 J147 Epigenetic Reader Domain , Dopamine Receptor , Monoamine Oxidase
J-147 is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging. It is a curcumin derivative and a potent neurogenic and neuroprotective drug candidate...
T7626 Budipine Others
Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.
T3596 TB5 MAO , Monoamine Oxidase
TB5 is a potent, selective and reversible inhibitor of hMAO-B.
T16803 RS 8359 MAO
RS 8359 is a reversible inhibitor of monoamine oxidase A (MAO-A) with a selectivity ratio of about 2200 for the A:B enzyme types. RS 8359 has antidepressant activity.
T1455 Nialamide Nialamid,Niamidal MAO , Transferase , Monoamine Oxidase
Nialamide (Nialamid) is an MAO inhibitor that is used as an antidepressive agent.
T39986 LOX-IN-3 dihydrochloride Lipoxygenase
LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX). LOX-IN-3 dihydrochloride inhibited bovine LOX (IC50<10 μM) and human LOXL2 (IC50<1 μM)activities.
T8907 Minaprine dihydrochloride MAO , Monoamine Oxidase
Minaprine dihydrochloride is a reversible MAO-A inhibitor; It weakly inhibit acetylcholinesterase. Minaprine dihydrochloride is an antidepressant for treatment of depression.
T7185 (2-Chloropyridin-4-yl)MethanaMine Hydrochloride Monoamine Oxidase
(2-Chloropyridin-4-yl)methanamine hydrochloride is a selective LOXL2 inhibitor(IC50 : 126 nM).
T5053 Eprobemide LIS 630 MAO , Monoamine Oxidase
Eprobemide (LIS 630) is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).
T12441 Phenelzine sulfate Monoamine Oxidase
Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.
T5323 Toloxatone MD 69276 MAO , Monoamine Oxidase
Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.
T18918 Azure B Azure B chloride MAO , Monoamine Oxidase
Azure B (Azure B chloride) is a cationic dye and the major metabolite of Methylene blue. Azure B is a selective, and reversible inhibitor of MAO-A (IC50s: 11 and 968 nM for recombinant human MAO-A and MAO-B).
T0300 Pargyline Pargylamine,Paragyline MAO , Monoamine Oxidase
Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.
T23070 Nisoxetine hydrochloride Sodium Channel , Monoamine Transporter , Norepinephrine
Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor
T22714 Decynium 22 Others
Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor
T1578 Pargyline hydrochloride Pargylamine hydrochloride MAO , Monoamine Oxidase
Pargyline hydrochloride (Pargylamine hydrochloride) is an irreversible monoamine oxidase(MAO) inhibitor with antihypertensive properties.
T0719 Tetrabenazine Xenazine,Ro 1-9569 Others , Dopamine Receptor , Monoamine Transporter
Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high...
T1119 Rasagiline AGN1135,TVP1012 BCL , MAO , Monoamine Oxidase
Rasagiline (AGN1135) is an inhibitor of monamine oxidase used as adjunctive therapy in combination with levodopa and carbidopa in the management of Parkinsons disease.
T1632 Amitraz BTS-27419,NSC 324552 Adrenergic Receptor , Parasite , Monoamine Oxidase
Amitraz (NSC 324552) is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic mange in dogs.
T7048 1,4-Naphthoquinone α-Naphthoquinone,Naphthalene-1,4-Dione,P-Naphthoquinone,para-naphthoquinone Others , MAO , Topoisomerase
1,4-Naphthoquinone (P-Naphthoquinone) was used as a potential inhibitor of monoamine oxidase and DNA topoisomerase activities[2]. It was also used to inhibit the acetyltransferase activity[1].
T7942 Tranylcypromine hemisulfate Tranylcypromine Sulfate,Tranylcypromine (hemisulfate) Histone Demethylase , MAO , Monoamine Oxidase
Tranylcypromine hemisulfate (Tranylcypromine Sulfate) is an inhibitor of monoamine oxidase (MAO) and lysine-specific demethylase 1 (LSD1) with a rapid onset of activity.
T2315 GSK-LSD1 dihydrochloride GSK-LSD1 (hydrochloride),GSK-LSD1 2HCl Histone Demethylase
GSK-LSD1 dihydrochloride (GSK-LSD1 2HCl) is a specificity irreversible LSD1 inhibitor (IC50: 16 nM). The selectivity of GSK-LSD1 for LSD1 is >1000 fold over other closely related FAD utilizing enzymes (i.e. MAO-A, LSD2, ...
T1117 Clorgyline hydrochloride Clorgiline hydrochloride MAO , Monoamine Oxidase
Clorgyline hydrochloride (Clorgiline hydrochloride), a white powder, is served as monoamine oxidase inhibitor.
T26795 PXS-4728A BI-1467335,BI 1467335,BI1467335,BI-1467335 HCl Monoamine Oxidase
BI-1467335 HCl(BI 1467335) is a selective, orally active inhibitor of semicarbazide-sensitive amine oxidase (SSAO) that helps improve chronic obstructive pulmonary disease in mice[2].
T4274 Melitracen hydrochloride Thymeol hydrochloride,Melixeran Dopamine Receptor , 5-HT Receptor
Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.
T6962 Rasagiline Mesylate TVP1012,AGN1135,Azilect Apoptosis , MAO , Autophagy , Monoamine Oxidase
Rasagiline Mesylate (AGN1135) is a novel MAO-B inhibitor, which can treat idiopathic Parkinson's disease.
T3534 Tetrabenazine Racemate Nitoman,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE Monoamine Transporter
Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been ...
T8589 (±)-Amiflamine 4-(dimethylamino)-alpha,Amiflamine,2-dimethylphenethylamine MAO , Monoamine Oxidase
(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.
T5678 Lazabemide hydrochloride N-(2-Aminoethyl)-5-chlor-2-pyridincarbox MAO , Monoamine Oxidase
Lazabemide hydrochloride (N-(2-Aminoethyl)-5-chlor-2-pyridincarbox) is a reversible and selective mao-b inhibitor(Ki:7.9nM).
T6352 (-)-Dizocilpine maleate C13737,(-)-MK 801 (Maleate),(-)-MK 801 Maleate NMDAR , iGluR
(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.
T5887 7-Hydroxy-3,4-dihydro-2(1H)-quinolinone 3,4-Dihydro-7-hydroxy-2(1H)-quinolinone MAO , Monoamine Oxidase
7-Hydroxy-3,4-dihydro-2(1H)-quinolinone is a weak MAO-A inhibitor(with an IC50 of 183 μM) .
T6888 Methylene Blue methylthioninium chloride,CI-52015,Tetramethylthionine chloride,Basic Blue 9 Guanylate cyclase , Microtubule Associated , NO Synthase , Parasite , Monoamine Oxidase
Methylene Blue (Tetramethylthionine chloride) (IC50 of 1.9 μM) inhibits tau filament formation. And it inhibits soluble guanylyl cyclase. It is also used as a dye in chromoendoscopy.
T7563 NBI-98782 (+)-α-Dihydrotetrabenazine,(+)-α-DHTBZ,(+)-DTBZ Monoamine Transporter
NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)
T0821 Iproniazid Phosphate Isoproniazid phosphate MAO , Monoamine Oxidase
Iproniazid Phosphate is a non-selective, irreversible monoamine oxidase inhibitor (MAOI).
T0006 Methylene Blue trihydrate Methylthionine chloride,Basic blue 9,Methylene Blue Guanylate cyclase , Microtubule Associated , NO Synthase , Parasite , Monoamine Oxidase
Methylene Blue trihydrate (Basic blue 9) is a compound consisting of dark green crystals or crystalline powder, having a bronze-like luster. Solutions in water or alcohol have a deep blue color. Methylene Blue trihydrate...
T5470 LAZABEMIDE Ro 19-6327 MAO , Monoamine Oxidase
Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively).
T6651 Safinamide mesylate PNU-151774E,FCE28073,PNU-151774E,NW-1015,EMD 1195686 mesylate MAO , Monoamine Oxidase
Safinamide mesylate (EMD 1195686 mesylate) , a mesylate salt of Safinamide, can reversibly and specifically inhibit MAO-B (IC50: 98 nM), has 5918-fold selectivity against MAO-A.

Compounds

Monoamine oxidase
T75422
Synonym:
Target:
Monoamine Oxidase B inhibitor 1
T60656
Synonym:
Target:
Monoamine Oxidase B inhibitor 2
T60806
Synonym:
Target:
Monoamine oxidase/Aromatase-IN-1
T61463
Synonym:
Target:
Isocarboxazid
T4559
Synonym:
Target: Monoamine Oxidase
Bifemelane hydrochloride
T22605
Synonym:
Target: MAO, Monoamine Oxidase
PF-9601N
T8849
Synonym:
Target: MAO
Valbenazine
T7147
Synonym: NBI-98854
Target: Monoamine Transporter
Modaline sulfate
T0235
Synonym:
Target: MAO, Monoamine Oxidase
PXS-5153A
T12585
Synonym:
Target: Others, Monoamine Oxidase
Moclobemide
T0084
Synonym: Ro111163
Target: MAO, Monoamine Oxidase
OG-L002
T6073
Synonym:
Target: Histone Demethylase, Monoamine Oxidase, HSV
PXS-5120A
T12584
Synonym:
Target: Others, Monoamine Oxidase
J-147
T1993
Synonym: J147
Target: Epigenetic Reader Domain, Dopamine Receptor, Monoamine Oxidase
Budipine
T7626
Synonym:
Target: Others
TB5
T3596
Synonym:
Target: MAO, Monoamine Oxidase
RS 8359
T16803
Synonym:
Target: MAO
Nialamide
T1455
Synonym: Nialamid,Niamidal
Target: MAO, Transferase, Monoamine Oxidase
LOX-IN-3 dihydrochloride
T39986
Synonym:
Target: Lipoxygenase
Minaprine dihydrochloride
T8907
Synonym:
Target: MAO, Monoamine Oxidase
(2-Chloropyridin-4-yl)MethanaMine Hydrochloride
T7185
Synonym:
Target: Monoamine Oxidase
Eprobemide
T5053
Synonym: LIS 630
Target: MAO, Monoamine Oxidase
Phenelzine sulfate
T12441
Synonym:
Target: Monoamine Oxidase
Toloxatone
T5323
Synonym: MD 69276
Target: MAO, Monoamine Oxidase
Azure B
T18918
Synonym: Azure B chloride
Target: MAO, Monoamine Oxidase
Pargyline
T0300
Synonym: Pargylamine,Paragyline
Target: MAO, Monoamine Oxidase
Nisoxetine hydrochloride
T23070
Synonym:
Target: Sodium Channel, Monoamine Transporter, Norepinephrine
Decynium 22
T22714
Synonym:
Target: Others
Pargyline hydrochloride
T1578
Synonym: Pargylamine hydrochloride
Target: MAO, Monoamine Oxidase
Tetrabenazine
T0719
Synonym: Xenazine,Ro 1-9569
Target: Others, Dopamine Receptor, Monoamine Transporter
Rasagiline
T1119
Synonym: AGN1135,TVP1012
Target: BCL, MAO, Monoamine Oxidase
Amitraz
T1632
Synonym: BTS-27419,NSC 324552
Target: Adrenergic Receptor, Parasite, Monoamine Oxidase
1,4-Naphthoquinone
T7048
Synonym: α-Naphthoquinone,Naphthalene-1,4-Dione,P-Naphthoquinone,para-naphthoquinone
Target: Others, MAO, Topoisomerase
Tranylcypromine hemisulfate
T7942
Synonym: Tranylcypromine Sulfate,Tranylcypromine (hemisulfate)
Target: Histone Demethylase, MAO, Monoamine Oxidase
GSK-LSD1 dihydrochloride
T2315
Synonym: GSK-LSD1 (hydrochloride),GSK-LSD1 2HCl
Target: Histone Demethylase
Clorgyline hydrochloride
T1117
Synonym: Clorgiline hydrochloride
Target: MAO, Monoamine Oxidase
PXS-4728A
T26795
Synonym: BI-1467335,BI 1467335,BI1467335,BI-1467335 HCl
Target: Monoamine Oxidase
Melitracen hydrochloride
T4274
Synonym: Thymeol hydrochloride,Melixeran
Target: Dopamine Receptor, 5-HT Receptor
Rasagiline Mesylate
T6962
Synonym: TVP1012,AGN1135,Azilect
Target: Apoptosis, MAO, Autophagy, Monoamine Oxidase
Tetrabenazine Racemate
T3534
Synonym: Nitoman,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE
Target: Monoamine Transporter
(±)-Amiflamine
T8589
Synonym: 4-(dimethylamino)-alpha,Amiflamine,2-dimethylphenethylamine
Target: MAO, Monoamine Oxidase
Lazabemide hydrochloride
T5678
Synonym: N-(2-Aminoethyl)-5-chlor-2-pyridincarbox
Target: MAO, Monoamine Oxidase
(-)-Dizocilpine maleate
T6352
Synonym: C13737,(-)-MK 801 (Maleate),(-)-MK 801 Maleate
Target: NMDAR, iGluR
7-Hydroxy-3,4-dihydro-2(1H)-quinolinone
T5887
Synonym: 3,4-Dihydro-7-hydroxy-2(1H)-quinolinone
Target: MAO, Monoamine Oxidase
Methylene Blue
T6888
Synonym: methylthioninium chloride,CI-52015,Tetramethylthionine chloride,Basic Blue 9
Target: Guanylate cyclase, Microtubule Associated, NO Synthase, Parasite, Monoamine Oxidase
NBI-98782
T7563
Synonym: (+)-α-Dihydrotetrabenazine,(+)-α-DHTBZ,(+)-DTBZ
Target: Monoamine Transporter
Iproniazid Phosphate
T0821
Synonym: Isoproniazid phosphate
Target: MAO, Monoamine Oxidase
Methylene Blue trihydrate
T0006
Synonym: Methylthionine chloride,Basic blue 9,Methylene Blue
Target: Guanylate cyclase, Microtubule Associated, NO Synthase, Parasite, Monoamine Oxidase
LAZABEMIDE
T5470
Synonym: Ro 19-6327
Target: MAO, Monoamine Oxidase
Safinamide mesylate
T6651
Synonym: PNU-151774E,FCE28073,PNU-151774E,NW-1015,EMD 1195686 mesylate
Target: MAO, Monoamine Oxidase
1 2 3 4
Cat No. Product Name Synonyms Targets
T2900 Paeonol Peonol MAO , Autophagy , Monoamine Oxidase
Paeonol (Peonol) is an active extraction from Paeonia suffruticosa. Paeonol inhibits MAO-A and MAO-B with IC50 of 54.6 μM and 42.5 μM, respectively.
TN1120 Osthenol MAO , Monoamine Oxidase
Osthenol is a natural product, and is selective, reversible, and competitive human monoamine oxidase-A (hMAO-A) inhibitor (Ki=0.26 µM).It shows antitumor-promoting activity, it also has antifungal and antibacterial activ...
T3152 Harmol Methylpyridoindolol Others
Harmol (Methylpyridoindolol) is a β-carboline isolated from nature.
TN2004 Obtusin MAO , Monoamine Oxidase
Obtusin is a natural product.
T3158 Harmane Loturine,Harman,Aribine Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T0791 Reserpine Serpalan,Serpasil,Serpivite Others , Potassium Channel , MRP , Monoamine Transporter , Autophagy
Reserpine (Serpalan) is an alkaloid found in the roots of Rauwolfia serpentina and R. vomitoria. Reserpine inhibits the uptake of norepinephrine into storage vesicles resulting in depletion of catecholamines and serotoni...
T4024 Norharmane 2-Azacarbazole,2,9-Diazafluorene,β-Carboline DNA , Endogenous Metabolite , Monoamine Oxidase
Norharmane (β-Carboline) is a natural β-carboline first isolated from plants of the Zygophyllaceae family.
T6862 Isatin Pseudoisatin,Indoline-2,3-dione,2,3-Indolinedione Apoptosis , MAO , Monoamine Oxidase
Isatin (2,3-Indolinedione) is an endogenous MAO inhibitor.
T2765 Rosmarinic acid Labiatenic acid,Rosemary acid Apoptosis , IκB/IKK , MAO , Endogenous Metabolite , Transferase , Monoamine Oxidase
Rosmarinic acid (Labiatenic acid) has shown to contain antioxidant, anti-inflammatory and antimicrobial activities. Possesses promising physiological actions related to cognitive performance, Alzheimer′s disease preventi...
T5S0734 Desmethoxyyangonin Desmethoxy yangonin,Demethoxyyangonin,5,6-Dehydrokavain Others , Monoamine Oxidase
1. Desmethoxyyangonin (5,6-Dehydrokavain) protects LPS or LPS/D-GalN-induced damages in cell or liver tissues mainly through de-regulating IKK/NFκB and Jak2/STAT3 signaling pathways. 2. The induction of CYP3A23 by dihydr...
T3885 ROSIRIDIN 6'-O-Deacetylrosiridoside C,(-)-Rosiridin Others , Monoamine Oxidase
Rosiridin (6'-O-Deacetylrosiridoside C) has cardioprotective activity.
T13475 β-Aminopropionitrile 3-Aminopropionitrile,BAPN Others , Endogenous Metabolite
β-Aminopropionitrile (3-Aminopropionitrile) is a selective inhibitor of lysyl oxidase.
T6S0923 Hypericin Hypericine,Cyclosan Apoptosis , Antiviral , Influenza Virus , Tyrosine Kinases , Antibacterial , PKC
1. Hypericin (Cyclosan) has antineoplastic activity. 2. Hypericin has antibiotic and antiviral activities. 3. Hypericin has antidepressive activity through inhibiting monoamine oxidase enzyme. 4. Hypericin inhibits RANKL...
Fr12415 Ethyl 4-hydroxyphenylacetate Others
Ethyl 4-hydroxyphenylacetate is a selective inhibitor of monoamine oxidase A.
TN7211 Tetrahydroharmine Leptaflorine MAO
Tetrahydroharmine (Leptaflorine) is a natural product found in the stems and large branches of Banisteriopsis caapi cultivar Da Vine. Tetrahydroharmine is a Monoamine oxidase A inhibitor.
T0948L Corticosterone 17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,Corticosterone (From plants) Glucocorticoid Receptor , Endogenous Metabolite
Corticosterone (Kendall's compound B) is a sensitive inhibitor of monoamine transport.
TN1705 Glycyrrhisoflavone MAO , Tyrosinase , NO Synthase , Immunology/Inflammation related
Glycyrrhisoflavone is a tyrosinase inhibitor with anti-inflammatory effects. Glycyrrhisoflavone inhibits α-glucosidase and monoamine oxidase.
T2209 Serotonin hydrochloride 5-HT hydrochloride,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride 5-HT Receptor , Endogenous Metabolite , Transferase
Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (COMT) inhibitor(Ki=44 μM).
T13354 Xanthoangelol Apoptosis , Monoamine Transporter , Antibacterial , AMPK
Xanthoangelol, which can be extracted from Angelica keiskei, inhibits obesity-induced inflammatory responses.Xanthoangelol has antimicrobial activity, inhibits monoamine oxidase, and induces apoptosis in neuroblastoma an...
TN1470 Cassiaside B2 Phosphatase , MAO , 5-HT Receptor
Cassiaside B2 is an inhibitor of protein tyrosine phosphatase 1B (PTP1B) and human monoamine oxidase A (hMAO-A).Cassiaside B2 is an agonist of the 5-HT2C receptor with anti-allergic activity.Cassiaside B2 is one of the a...
T3095 Tyramine 4-hydroxyphenethylamine,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine MAO , Endogenous Metabolite
Tyramine (Uteramine) is an indirect sympathomimetic that occurs naturally in cheese and other foods. Tyramine does not directly activate adrenergic receptors, but it can serve as a substrate for adrenergic uptake systems...
T3933 Jatrorrhizine Yatrorizine,neprotin MAO , 5-HT Receptor , Antibacterial , AChE
Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species. It was found to have antimicrobial and antifungal activity. It binds and noncompetitively inhibits mo...
T0647 Tryptamine Dehydrogenase , 5-HT Receptor , Endogenous Metabolite , TRP/TRPV Channel
Tryptamine is a monoamine alkaloid found in animals, plants, and fungi. It contains an indole ring structure and is structurally analogous to the tryptophan. It is found in trace amounts in the brains of mammals and is r...
T0469 Octopamine hydrochloride (±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl Dopamine Receptor , Endogenous Metabolite , Adrenergic Receptor
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) is a biogenic monoamine structurally associated with noradrenaline. It can serve as a neurohormone, a neurotransmitter, and a neuromodulator in invertebrates.
T3822 Bellidifolin Bellidifoline,Bellidifolium Others , HIV Protease
Bellidifolin (Bellidifoline) has anti-oxidation, hepatoprotective, anti-inflammatory and antitumor actions, it may contribute to the protective effects associated with nerve injury initiated by hypoxia by mechanisms rela...
T1311 4-aminobenzoic acid PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid Endogenous Metabolite
4-aminobenzoic acid (para-Aminobenzoic acid) is an organic acid with UV absorption and antifibrotic properties. When exposed to light, 4-aminobenzoic acid absorbs UV light and emits excess energy via a photochemical reac...
T4848 Mandelic acid acidomandelico,DL-Mandelic acid Others , Endogenous Metabolite , Antibacterial
It is an isomer of cresotinic acid (2-hydroxy-3-methylbenzoic acid) and oxymethylbenzoic acid (2-methoxybenzoic acid). Derivatives of mandelic acid are formed as a result of metabolism of adrenaline and noradrenaline by ...
TN3918 Echitovenidine MAO
Echitovenidine shows monoamine oxidase inhibitor activity.
T36950 Rubrofusarin triglucoside
Rubrofusarin triglucoside is a glycoside compound isolated from Cassia obtusifolia Linn seeds. Rubrofusarin triglucoside inhibits human monoamine oxidase A (hMAO-A) with an IC50 of 85.5 μM[1]. [1]. Pradeep Paudel, et al....
TN3693 Confluentic acid Others
Confluentic acid shows selective inhibition of Monoamine oxidase B with IC50 value of 0.22 microM.
T40244 Methyl citrate
Methyl citrate, obtained from Opuntia ficus-indica var. saboten Makino fruits, serves as a potent Monoamine oxidase B (MAO-B) inhibitor with an IC50 value of 0.23 mM.
TN2790 2'-O-Methylperlatolic acid MAO
2'-O-Methylperlatolic acid and confluentic acid are monoamine oxidase B inhibitors in a Brazilian plant, Himatanthus sucuuba.
TN4137 Glicoricone MAO
Glicoricone acts as a partial estrogen antagonist. Glicoricone inhibited the monoamine oxidase with the IC50 values of 6.0 x 10(-5)-1.4 x 10(-4) M.
T32208 Isogentisin BRN 0258402,BRN-0258402,BRN0258402 MAO
Isogentisin (BRN 0258402), a compound isolated from Gentianaceae, is a novel compound for the prevention of smoking-induced endothelial damage.Isogentisin exhibits inhibitory effects on monoamine oxidase.
TN3116 5-Hydroxy-1-methoxyxanthone MAO , Antifection
5-Hydroxy-1-methoxyxanthone, 1,5-dihydroxyxanthone and 6-deoxyjacareubin are all antifungal against Cladosporium cucumerinum, while they show differing degrees of inhibition of monoamine oxidase A and B.
TN3726 Cudraflavone B IκB/IKK , MAO , ROS , Akt , COX , PI3K , Nrf2 , Autophagy
Cudraflavone B has anti-proliferative activity, mouse brain monoamine oxidase (MAO) inhibitory effects, apoptotic actions in human gastric carcinoma cells and mouse melanoma cells, and hepatoprotective activity. It may b...
T40576 (S)-Salsolidine
(S)-Salsolidine, a chemical compound, functions as a weak inhibitor of monoamine oxidase (MAO), exhibiting an inhibition constant (K i ) of 63 μM. R enantiomer demonstrating a greater efficacy than (S)-Salsolidine, boast...
TC0022 Desoxypeganine Deoxypeganine AChE
Desoxypeganine (Deoxypeganine) is an inhibitor of cholinesterase. It acting preferentially on butyrylcholinesterase, and as a selective inhibitor of monoamine oxidase A but not monoamine oxidase B.Desoxypeganine is being...
TN5901 Cudratricusxanthone A
Cudratricusxanthone A has potent anti-proliferative, antioxidative, and monoamine oxidase inhibitory effects, it also possesses anti-cancer activities and provide a basis for developing effective therapeutic agents to in...
T79979 Methyl piperate Monoamine Oxidase
Methylpiperic acid, a piperine alkaloid, exhibits potent inhibitory activity on monoamine oxidase (MAO), with differing efficacy on isoforms: greater inhibition of MAO-A (IC 50 27.1 μM) compared to MAO-B (IC 50 1.6 μM), ...
T37911 Cis-Resveratrol (Z)-Resveratrol
Resveratrol is a potent phenolic antioxidant found in grapes, red wine, and various berries that also has antiproliferative and anti-inflammatory activity. cis-Resveratrol is the double bond isomer of trans-resveratrol, ...

Natural Products

Paeonol
T2900
Synonym: Peonol
Target: MAO, Autophagy, Monoamine Oxidase
Osthenol
TN1120
Synonym:
Target: MAO, Monoamine Oxidase
Harmol
T3152
Synonym: Methylpyridoindolol
Target: Others
Obtusin
TN2004
Synonym:
Target: MAO, Monoamine Oxidase
Harmane
T3158
Synonym: Loturine,Harman,Aribine
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
Reserpine
T0791
Synonym: Serpalan,Serpasil,Serpivite
Target: Others, Potassium Channel, MRP, Monoamine Transporter, Autophagy
Norharmane
T4024
Synonym: 2-Azacarbazole,2,9-Diazafluorene,β-Carboline
Target: DNA, Endogenous Metabolite, Monoamine Oxidase
Isatin
T6862
Synonym: Pseudoisatin,Indoline-2,3-dione,2,3-Indolinedione
Target: Apoptosis, MAO, Monoamine Oxidase
Rosmarinic acid
T2765
Synonym: Labiatenic acid,Rosemary acid
Target: Apoptosis, IκB/IKK, MAO, Endogenous Metabolite, Transferase, Monoamine Oxidase
Desmethoxyyangonin
T5S0734
Synonym: Desmethoxy yangonin,Demethoxyyangonin,5,6-Dehydrokavain
Target: Others, Monoamine Oxidase
ROSIRIDIN
T3885
Synonym: 6'-O-Deacetylrosiridoside C,(-)-Rosiridin
Target: Others, Monoamine Oxidase
β-Aminopropionitrile
T13475
Synonym: 3-Aminopropionitrile,BAPN
Target: Others, Endogenous Metabolite
Hypericin
T6S0923
Synonym: Hypericine,Cyclosan
Target: Apoptosis, Antiviral, Influenza Virus, Tyrosine Kinases, Antibacterial, PKC
Ethyl 4-hydroxyphenylacetate
Fr12415
Synonym:
Target: Others
Tetrahydroharmine
TN7211
Synonym: Leptaflorine
Target: MAO
Corticosterone
T0948L
Synonym: 17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,Corticosterone (From plants)
Target: Glucocorticoid Receptor, Endogenous Metabolite
Glycyrrhisoflavone
TN1705
Synonym:
Target: MAO, Tyrosinase, NO Synthase, Immunology/Inflammation related
Serotonin hydrochloride
T2209
Synonym: 5-HT hydrochloride,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride
Target: 5-HT Receptor, Endogenous Metabolite, Transferase
Xanthoangelol
T13354
Synonym:
Target: Apoptosis, Monoamine Transporter, Antibacterial, AMPK
Cassiaside B2
TN1470
Synonym:
Target: Phosphatase, MAO, 5-HT Receptor
Tyramine
T3095
Synonym: 4-hydroxyphenethylamine,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine
Target: MAO, Endogenous Metabolite
Jatrorrhizine
T3933
Synonym: Yatrorizine,neprotin
Target: MAO, 5-HT Receptor, Antibacterial, AChE
Tryptamine
T0647
Synonym:
Target: Dehydrogenase, 5-HT Receptor, Endogenous Metabolite, TRP/TRPV Channel
Octopamine hydrochloride
T0469
Synonym: (±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl
Target: Dopamine Receptor, Endogenous Metabolite, Adrenergic Receptor
Bellidifolin
T3822
Synonym: Bellidifoline,Bellidifolium
Target: Others, HIV Protease
4-aminobenzoic acid
T1311
Synonym: PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid
Target: Endogenous Metabolite
Mandelic acid
T4848
Synonym: acidomandelico,DL-Mandelic acid
Target: Others, Endogenous Metabolite, Antibacterial
Echitovenidine
TN3918
Synonym:
Target: MAO
Rubrofusarin triglucoside
T36950
Synonym:
Target:
Confluentic acid
TN3693
Synonym:
Target: Others
Methyl citrate
T40244
Synonym:
Target:
2'-O-Methylperlatolic acid
TN2790
Synonym:
Target: MAO
Glicoricone
TN4137
Synonym:
Target: MAO
Isogentisin
T32208
Synonym: BRN 0258402,BRN-0258402,BRN0258402
Target: MAO
5-Hydroxy-1-methoxyxanthone
TN3116
Synonym:
Target: MAO, Antifection
Cudraflavone B
TN3726
Synonym:
Target: IκB/IKK, MAO, ROS, Akt, COX, PI3K, Nrf2, Autophagy
(S)-Salsolidine
T40576
Synonym:
Target:
Desoxypeganine
TC0022
Synonym: Deoxypeganine
Target: AChE
Cudratricusxanthone A
TN5901
Synonym:
Target:
Methyl piperate
T79979
Synonym:
Target: Monoamine Oxidase
cis-Resveratrol
T37911
Synonym: (Z)-Resveratrol
Target:

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPJ-00379 AOC3 Protein, Human, Recombinant (hFc) Human Human Cells
Membrane primary amine oxidase(AOC3), also known as vascular adhesion protein (VAP-1) and HPAO, this protein is a member of the semicarbazide-sensitive amine oxidase (SSAO) family. VAP-1 is a type 1 membrane-bound glycop...
TMPY-02446 GAPDH Protein, Human, Recombinant (His) Human E. coli
Glyceraldehyde 3-phosphate dehydrogenase (GAPDH or G3PDH) is an enzyme of about 37kDa that is consisdered as a cellular enzyme involved in glycolysis. It catelyzes the sixth step of glycolysis. Glyceraldehyde-3-phosphate...
TMPY-00506 GAPDH Protein, Mouse, Recombinant (His) Mouse E. coli
Glyceraldehyde 3-phosphate dehydrogenase (GAPDH or G3PDH) is an enzyme of about 37kDa that is consisdered as a cellular enzyme involved in glycolysis. It catelyzes the sixth step of glycolysis. Glyceraldehyde-3-phosphate...
TMPY-03056 LSD1 Protein, Human, Recombinant (His & GST) Human Baculovirus-Insect Cells
LSD1 belongs to the flavin monoamine oxidase family. It contains 1 SWIRM domain and is a component of an RCOR/GFI/LSD1/HDAC complex. LSD1 interacts directly with GFI1 and GFI1B. LSD1 specifically removes histone H3K4me2 ...
Cat No. Product Name
L2800 Serotonin Receptor-Targeted Compound Library

275 compounds
A unique collection of 275 compounds targeting serotonin receptors for high throughput screening and high content screening;
L9830 Anti-Parkinson's Disease Compound Library

908 compounds
A unique collection of 908 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS.
TargetMol