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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T3036 | Dydrogesterone | Progesterone Receptor | |
Dydrogesterone is a potent progestogen which can be used in progesterone deficiency studies. | |||
T13703 | Gestonorone Capronate | Prostaglandin Receptor | |
Gestonorone Capronate is a progesterone used to treat benign prostatic hyperplasia and endometrial cancer. | |||
T1514 | Norethindrone | Norethisterone | Estrogen/progestogen Receptor , Progesterone Receptor |
Norethindrone (Norethisterone) is a synthetic progestational hormone with actions similar to those of PROGESTERONE but functioning as a more potent inhibitor of ovulation. It has weak estrogenic and androgenic properties... | |||
T1596 | Chlormadinone acetate | Gestafortin | Progesterone Receptor , Androgen Receptor |
Chlormadinone acetate (Gestafortin) is an orally active synthetic progestational hormone used often in combinations as an oral contraceptive. | |||
T8395 | Nomegestrol acetate | Others , Progesterone Receptor | |
Nomegestrol acetate is a widely used progestin-like drug,which is characterized as a full agonist at the progesterone receptor | |||
T1541 | Drospirenone | ZK 3059,Dihydrospirorenone | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , COX |
Drospirenone (ZK 3059) is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity. | |||
T7537 | Norgestimate | Progesterone Receptor | |
Norgestimate is an acetylated progestinused in combination with ethinyl estradiol as an oral contraceptive. | |||
T28362 | PF-02413873 | PF02413873 | Progesterone Receptor |
PF-02413873 is a competitive antagonist of nonsteroidal progesterone receptor with a Ki of 2.6 nM. PF-02413873 can be used in studies about the treatment of gynecological conditions such as endometriosis. | |||
T6819 | Desogestrel | Org-2969,Desogen,Desogestrelum,Cerazette | Estrogen/progestogen Receptor , Progesterone Receptor |
Desogestrel (Cerazette) is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents. | |||
T0996 | Ethynodiol diacetate | Ethynodiol acetate,8080 CB | Estrogen/progestogen Receptor , Progesterone Receptor |
Ethynodiol diacetate (Ethynodiol acetate) is a synthetic progestational hormone used alone or in combination with estrogens as an oral contraceptive. | |||
T6713 | Ulipristal | Estrogen/progestogen Receptor , Progesterone Receptor | |
Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure. | |||
T2577 | Dienogest | STS 557 | Apoptosis , Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy |
Dienogest (STS 557) is an orally-active, semisynthetic, fourth generation, nonethinylated progestogen with antiproliferative, antiandrogenic, anti-inflammatory and antiangiogenic activities that is used in hormone therap... | |||
T1490 | Gestodene | SHB 331,WL 70 | Estrogen/progestogen Receptor , Progesterone Receptor |
Gestodene (WL 70) is a progestogen hormonal contraceptive. | |||
T0870 | Altrenogest | R2267,RU2267,Allyltrenbolone,A35957 | Estrogen/progestogen Receptor , Progesterone Receptor |
Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone. | |||
T5174 | Nestoron | ST-1435,Segesterone Acetate,Nestorone,Elcometrine | Estrogen/progestogen Receptor , Progesterone Receptor |
Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM). | |||
T2527 | Ulipristal acetate | Ulipristal,CDB-2914 | Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy |
Ulipristal acetate (CDB-2914) is an orally bioavailable, acetate salt of ulipristal, a selective progesterone receptor modulator with anti-progesterone activity. Ulipristal binds to the progesterone receptor (PR), thereb... | |||
T14975 | CJ-42794 | CJ-042794 | Others |
CJ-42794 (CJ-042794) is a selective antagonist of prostaglandin E receptor subtype 4 (EP4). It inhibits [3H]-PGE2 binding to the human EP4 receptor (a mean pKi: 8.5). CJ-42794 is a binding affinity that was at least 200-... | |||
T5317 | Cridanimod | CMA,XBIO-101,10-carboxymethyl-9-acridanone | Progesterone Receptor , STING , IFNAR |
Cridanimod (10-carboxymethyl-9-acridanone, CMA) is a potent STING agonist that directly binds to STING and triggers a strong antiviral response through the TBK1/IRF3 route. | |||
T2567 | Etonogestrel | 3-Oxodesogestrel,3-keto-Desogestrel,Nexplanon,Implanon | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite |
Etonogestrel (Implanon) is a steroidal progestin used as hormonal contraceptives. | |||
T1102 | Mifepristone | C-1073,RU486,RU 38486 | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , NO Synthase , Autophagy |
Mifepristone (C-1073) is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist. | |||
T2231 | Estradiol dipropionate | 17-Beta-Estradiol-3,17-Dipropionate | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Progesterone Receptor |
Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol. | |||
T20720 | Norethisterone enanthate | NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,NSC-9564 | Estrogen/progestogen Receptor |
Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects. |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0478 | Progesterone | Pregn-4-ene-3,20-dione | Estrogen/progestogen Receptor , Progesterone Receptor , Opioid Receptor , Endogenous Metabolite |
Progesterone (Pregn-4-ene-3,20-dione) is the major progestational steroid that is secreted primarily by the CORPUS LUTEUM and the PLACENTA. Progesterone acts on the UTERUS, the MAMMARY GLANDS and the BRAIN. It is require... | |||
T1263 | Levonorgestrel | D-Norgestrel | Others , Estrogen/progestogen Receptor , Progesterone Receptor |
Levonorgestrel (D-Norgestrel) is a Progestin and Progestin-containing Intrauterine Device. The physiologic effect of levonorgestrel is by means of Inhibit Ovum Fertilization. | |||
T5040 | Medroxyprogesterone | Estrogen/progestogen Receptor , Progesterone Receptor | |
Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator. | |||
T1284 | Megestrol acetate | SC10363,BDH1298 | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , HIV Protease , Autophagy |
Megestrol acetate (BDH1298) is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic properties. It is given by mouth in the palliative treatment ... | |||
T1429 | 17α-Hydroxyprogesterone | Hydroxyprogesterone,17-OHP,17-Hydroxyprogesterone | Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite |
17α-Hydroxyprogesterone (17-OHP) is a physiological progestin that is produced during glucocorticoid and steroid hormone synthesis and is increased during the third trimester of pregnancy. Hydroxyprogesterone binds to th... | |||
T1261 | Medroxyprogesterone Acetate | Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,Farlutin,Medroxyprogesterone (acetate) | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , Endogenous Metabolite |
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally or by intramuscular injection and has also been... |