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Search Result

Search Results for " nonpeptide "

Targets

Oxytocin Receptor

69

Compounds

1

Natural Products

Cat No. Product Name Synonyms Targets
T11857 LIT-001 Oxytocin Receptor
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin receptor agonist with EC50 of 55 nM and Ki of 226 nM.
T11696 Ivachtin Caspase-3 Inhibitor VII Caspase
Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining caspases.
T16850 SB-265610 GSK-CXCR2 CXCR
SB-265610 (GSK-CXCR2) is a nonpeptide and allosteric CXCR2 antagonist. SB-265610 blocks rat cytokine-induced neutrophil chemoattractant-1 (CINC-1)-induced calcium mobilization and neutrophil chemotaxis (IC50s: 3.7 nM and...
T6288 Mozavaptan OPC31260l,OPC-31260 Vasopressin Receptor
Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
T12870 SCH79797 dihydrochloride Apoptosis , Others , Protease-activated Receptor
SCH79797 dihydrochloride is an effective and selective antagonist of protease activated receptor 1 (PAR1) with an IC50 of 70 nM and a Ki of 35 nM. SCH79797 dihydrochloride has antiproliferative and pro-apoptotic effects.
T3178 BIBS 39 RAAS
BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.
T21790 BMS 182874 hydrochloride Endothelin Receptor
BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.
T27762 L-162,313 L-162313,L 162,313,L162,313 RAAS
L-162,313 is an ANG II receptor agonist, a nonpeptide that mimics the biological actions of angiotensin II and induces an increase in MAP.
T1520 Aliskiren hemifumarate CGP 60536,SPP 100,CGP60536B RAAS , Autophagy
Aliskiren hemifumarate (CGP60536B) is an orally active nonpeptide renin inhibitor with antihypertensive activity.
T3347 PF3274167 PF 3274167,Cligosiban,PF-3274167 OX Receptor
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.
T39229 YNT-185 OX Receptor
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R, respectively. Furthermore, YNT-185 effectively alleviates symptoms of ...
T6281 TW-37 TW 37 BCL
TW-37 is an nonpeptide inhibitor to recombinant Bcl-2, Bcl-xL and Mcl-1 (Ki: 0.29/1.11/0.26 μM).
T26594 Allisartan Isoproxil RAAS
Allisartan Isoproxil is a nonpeptide antagonist of angiotensin II receptor and can be used in studies about hypertension and heart diseases.
T25615 Lanepitant LY303870,LY-303870,LY 303870 Others
Lanepitant (LY303870) is a nonpeptide neurokinin-1 (NK-1) antagonist with analgesic activity that inhibits neurogenic dura mater inflammation and is used for the prevention of migraine.
T9692 Paltusotine Somatostatin
Paltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients
TQ0057 AVE 0991 Others
AVE 0991, a nonpeptide analog of angiotensin-(1-7) [Ang-(1-7)], is an orally active Mas agonist with inhibitory effects on [125I]-Ang-(1-7) binding to bovine aortic endothelial cell membranes, and inhibits astrocyte-medi...
T11174 (R)-Elagolix NBI-56418 GNRH Receptor
(R)-Elagolix (NBI-56418) is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a do...
T8691 PD 168368 PD168368 Bombesin Receptor
PD 168368 is a novel, potent, competitive and selective nonpeptide neuromodulin B receptor (NMB-R) antagonist with inhibitory effects on the gastrin-releasing peptide receptor (GRPR).PD 168368 is a potent mixed agonist o...
T6825 Eltrombopag Olamine Promacta Olamine,Revolade,Eltrombopag diethanolamine salt,SB497115,SB-497115GR Thrombin
Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin receptor agonist with megakaryopoiesis-stimulating activity. Eltrom...
T2531L Eprosartan KF-108566J free base,Teveten RAAS
Eprosartan (SKF-108566J free base) is a selective and competitive nonpeptide angiotensin II receptor antagonist with high affinity for AT1 receptor subtypes and can be used as an antihypertensive agent.Eprosartan has an ...
T28813 SM19712 sodium SM 19712,SM19712,SM-19712
SM19712 sodium is an inhibitor of nonpeptide endothelin converting enzyme.
T28814 SM19712 free acid SM 19712,SM-19712,SM19712
SM19712 is an inhibitor of nonpeptide endothelin converting enzyme.
T70136 CAM 4750
CAM 4750 is a nonpeptide tachykinin NK1 receptor antagonist.
T12331 OT-R antagonist 2 Oxytocin receptor antagonist 2 Others
OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .
T28322 PD 123177 PD-123177,PD123177,Exp-655,Exp655,Exp 655
PD 123177 is an inhibitor of Nonpeptide angiotensin AII-2.
T70272 L-162782
L-162782 is a nonpeptide agonist of angiotensin AT1 receptor.
T68486 Fasitibant
Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.
T69097 ARD-353
ARD-353 is a nonpeptide delta receptor agonist with cardioprotective effects.
T29234 ZM 253270 ZM253270,ZM-253270
ZM 253270 is an nonpeptide neurokinin A antagonist.
T27940 LY301875 LY 301875,LY-301875
LY301875 is an antagonist of nonpeptide angiotensin receptor.
T16085 MK-0429 L-000845704 Others
MK-0429 is an orally active, selective, and nonpeptide antagonist of αvβ3 integrin (IC50: 80 nM).
T70137 CAM 4515
CAM 4515 is a nonpeptide tachykinin NK1 receptor antagonist.
T25895 NVP-SAA164 SAA 164,SAA164,SAA-164,NVP SAA164
NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.
T16935 SR 146131 Others
SR 146131 is a potent and selective agonist of the nonpeptide receptor.
T25608 Lamifiban trifluoroacetate Lamifiban trifluoroacetate salt
Lamifiban trifluoroacetate is an antagonist of the nonpeptide platelet fibrinogen receptor (GPIIb/IIIa).
T29177 YM 218 YM218,YM-218
YM 218 is a novel, potent, selective antagonist of nonpeptide vasopressin V1A receptor.
T70295 MDL-105212A HCl
MDL-105212A HCl is a nonpeptide NK-1 and NK-2 receptor antagonist.
T25607 Lamifiban Ro-44-9883/000,Ro 44-9883/000,Ro44-9883/000
Lamifiban is a nonpeptide glycoprotein IIb/IIIa antagonist. It prevents platelet loss during experimental cardiopulmonary bypass.
T70225 L-159884
L-159884 is a radiolabelled, nonpeptide angiotensin II antagonist that is useful for angiotensin II, AT1 receptor imaging
T70658 Ici D8731
Ici D8731 is a nonpeptide angiotensin II antagonist with potential as a treatment for hypertension and heart failure.
T26802 BIBS-222 BIBS 222
BIBS-222, a nonpeptide angiotensin II (Ang II) receptor antagonist, appears to be an effective antihypertensive in the model of the renal hypertensive rat.
T16895 SL910102 Others
SL910102 is a nonpeptide angiotensin antagonist of the AT1 receptor.
T70410 Cam 2445
Cam 2445 is a nonpeptide, alpha-methyltryptophan derivative; an NK1 neurokinin receptor antagonist that is a potentially useful treatment for arthritis, asthma, migraine, anxiety, psychosis, and emesis.
T12331L OT-R antagonist 1 Oxytocin receptor antagonist 1 Others
OT-R antagonist 1 inhibits oxytocin-evoked intracellular Ca2+ mobilization (IC50 = 8 nM). OT-R antagonist 1 is a new effective and selective nonpeptide low molecular weight OT-R antagonist.
T11862 LMD-009 Others
LMD-009 mediates chemotaxis, inositol phosphate accumulation, and calcium release in high potencies with EC50s from 11 to 87 nM. LMD-009 is a selective CCR8 nonpeptide agonist.
T15680 L-159282 MK 996 Others
L-159282 is an orally active and nonpeptide angiotensin II receptor antagonist. It also has anti-hypertensive activity.
T61079 RXFP3 agonist 1
RXFP3 agonist 1 is a nonpeptide RXFP3 agonist ( EC 50 =6937 nM) [1].
T15101 Devazepide L-364,718,MK-329 Others
Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respective...
T36481 BIIE 0246 hydrochloride
Potent, selective and competitive nonpeptide antagonist for the neuropeptide Y Y2 receptor (IC50 = 15 nM). Displays > 650-fold selectivity for NPY Y2 over Y1, Y4 and Y5 receptors. Active in vivo.
T29151 WAY267464 HCl WAY267464,WAY-267464,WAY 267,464 dihydrochloride,WAY-267,464 dihydrochloride,WAY 267464 dihydrochloride,WAY 267464
WAY267464 is a nonpeptide small-molecule OT agonists with anxiolytic activity. WAY267464 may be used for modulation of potency, selectivity over the structurally similar vasopressin receptors, CNS penetration, and oral b...

Compounds

LIT-001
T11857
Synonym:
Target: Oxytocin Receptor
Ivachtin
T11696
Synonym: Caspase-3 Inhibitor VII
Target: Caspase
SB-265610
T16850
Synonym: GSK-CXCR2
Target: CXCR
Mozavaptan
T6288
Synonym: OPC31260l,OPC-31260
Target: Vasopressin Receptor
SCH79797 dihydrochloride
T12870
Synonym:
Target: Apoptosis, Others, Protease-activated Receptor
BIBS 39
T3178
Synonym:
Target: RAAS
BMS 182874 hydrochloride
T21790
Synonym:
Target: Endothelin Receptor
L-162,313
T27762
Synonym: L-162313,L 162,313,L162,313
Target: RAAS
Aliskiren hemifumarate
T1520
Synonym: CGP 60536,SPP 100,CGP60536B
Target: RAAS, Autophagy
PF3274167
T3347
Synonym: PF 3274167,Cligosiban,PF-3274167
Target: OX Receptor
YNT-185
T39229
Synonym:
Target: OX Receptor
TW-37
T6281
Synonym: TW 37
Target: BCL
Allisartan Isoproxil
T26594
Synonym:
Target: RAAS
Lanepitant
T25615
Synonym: LY303870,LY-303870,LY 303870
Target: Others
Paltusotine
T9692
Synonym:
Target: Somatostatin
AVE 0991
TQ0057
Synonym:
Target: Others
(R)-Elagolix
T11174
Synonym: NBI-56418
Target: GNRH Receptor
PD 168368
T8691
Synonym: PD168368
Target: Bombesin Receptor
Eltrombopag Olamine
T6825
Synonym: Promacta Olamine,Revolade,Eltrombopag diethanolamine salt,SB497115,SB-497115GR
Target: Thrombin
Eprosartan
T2531L
Synonym: KF-108566J free base,Teveten
Target: RAAS
SM19712 sodium
T28813
Synonym: SM 19712,SM19712,SM-19712
Target:
SM19712 free acid
T28814
Synonym: SM 19712,SM-19712,SM19712
Target:
CAM 4750
T70136
Synonym:
Target:
OT-R antagonist 2
T12331
Synonym: Oxytocin receptor antagonist 2
Target: Others
PD 123177
T28322
Synonym: PD-123177,PD123177,Exp-655,Exp655,Exp 655
Target:
L-162782
T70272
Synonym:
Target:
Fasitibant
T68486
Synonym:
Target:
ARD-353
T69097
Synonym:
Target:
ZM 253270
T29234
Synonym: ZM253270,ZM-253270
Target:
LY301875
T27940
Synonym: LY 301875,LY-301875
Target:
MK-0429
T16085
Synonym: L-000845704
Target: Others
CAM 4515
T70137
Synonym:
Target:
NVP-SAA164
T25895
Synonym: SAA 164,SAA164,SAA-164,NVP SAA164
Target:
SR 146131
T16935
Synonym:
Target: Others
Lamifiban trifluoroacetate
T25608
Synonym: Lamifiban trifluoroacetate salt
Target:
YM 218
T29177
Synonym: YM218,YM-218
Target:
MDL-105212A HCl
T70295
Synonym:
Target:
Lamifiban
T25607
Synonym: Ro-44-9883/000,Ro 44-9883/000,Ro44-9883/000
Target:
L-159884
T70225
Synonym:
Target:
Ici D8731
T70658
Synonym:
Target:
BIBS-222
T26802
Synonym: BIBS 222
Target:
SL910102
T16895
Synonym:
Target: Others
Cam 2445
T70410
Synonym:
Target:
OT-R antagonist 1
T12331L
Synonym: Oxytocin receptor antagonist 1
Target: Others
LMD-009
T11862
Synonym:
Target: Others
L-159282
T15680
Synonym: MK 996
Target: Others
RXFP3 agonist 1
T61079
Synonym:
Target:
Devazepide
T15101
Synonym: L-364,718,MK-329
Target: Others
BIIE 0246 hydrochloride
T36481
Synonym:
Target:
WAY267464 HCl
T29151
Synonym: WAY267464,WAY-267464,WAY 267,464 dihydrochloride,WAY-267,464 dihydrochloride,WAY 267464 dihydrochloride,WAY 267464
Target:
1 2
Cat No. Product Name Synonyms Targets
T4954L Smilagenin PYM50028,Cogane,AI3-44895,PYM 50028
Smilagenin is an orally active inducer of nonpeptide neurotrophic factor. It also prevents and reverses neuronal damage induced by MPP+ in mesencephalic neurons, and by MPTP in a mouse model of Parkinson's disease.

Natural Products

Smilagenin
T4954L
Synonym: PYM50028,Cogane,AI3-44895,PYM 50028
Target:
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