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Compounds

Cat No. Product Name
T12253 Nrf2-IN-1 Others , Nrf2
Nrf2-IN-1 是 Nrf2抑制剂,可用于研究急性髓性白血病药物。
T39719 Nrf2 activator-1 Nrf2 activator-1
Nrf2 activator-1, a highly potent activator of NF-E2 related factor 2 (Nrf2), shows promising therapeutic potential for ...
T24546 Nrf2-Activator-12G Nrf2 Activator-IV,Nrf2 Activator IV
Nrf2-Activator-12G is a potent Nrf-2 activator.
T39514 Keap1-Nrf2-IN-3 Keap1-Nrf2-IN-3
Keap1-Nrf2-IN-3 is a KEAP1:NRF2 protein protein interaction inhibitor, and with a K d value of 2.5 nM for KEAP1 protein.
T11752 Keap1-Nrf2-IN-1 Keap1–Nrf2-IN-1 Src
Keap1–Nrf2 IN-1 activates Nrf2-regulated cytoprotective response and antagonizes acetaminophen-induced liver injury both...
T72697 Nrf2 activator-6
Nrf2 activator-6 是一种四氢异喹啉化合物,是一种 Nrf2激活剂。Nrf2 activator-6 抑制 Kelch 结构域-Nrf2 相互作用的 IC50为 5 nM (WO2021214470A1 ; Example ...
T63016 Nrf2 activator-4
Nrf2 activator-4 (Compound 20a) 是一种高效的、口服具有活力的 Nrf2 激活剂 (EC50: 0.63 μM)。Nrf2 activator-4 对小神经胶质细胞中活性氧的产生具有抑制作用。在 scopola...
T72417 AChE/Nrf2 modulator 1
AChE/Nrf2 modulator 1 是乙酰胆碱酯酶 (AChE) /核因子红系 2 相关因子 2 (Nrf2) 调节剂,具有口服活性。AChE/Nrf2 modulator 1 具有 Nrf2 诱导活性和AChE 抑制活性,对 ee...
T74600 Keap1-Nrf2-IN-9
Keap1-Nrf2-IN-9(compound 11)是一种有效的Keap1-Nrf2PPI (Keap1-Nrf2 蛋白质-蛋白质相互作用)抑制剂,IC50值为 0.575 µM。Keap1-Nrf2-IN-9 增加 Nrf2 靶基因的...
T72706 Keap1-Nrf2-IN-13
Keap1-Nrf2-IN-13 是一种 Keap1-Nrf2蛋白质-蛋白质相互作用 (Keap1-Nrf2PPI) 抑制剂,IC50值为 0.15 μM。 Keap1-Nrf2-IN-13 可与 Keap1 蛋白的关键极性残基 (Asn4...
T61688 Nrf2 activator-2
Nrf2 activator-2 (referred to as compound O15), an Osthole derivative, is a highly potent Nrf2 agonist exhibiting an EC ...
T63364 Nrf2 activator-5
Nrf2 activator-5 是 Nrf2 的有效激活剂,能够减轻 BV-2 小胶质细胞中 H2O2诱导的氧化应激和 LPS 刺激的炎症,表现出抗氧化和抗炎活作用。
T72760 Keap1-Nrf2-IN-6
Keap1-Nrf2-IN-6 是一种有效且选择性的Keap1-Nrf2PPI (Keap1-Nrf2 protein-protein interaction)抑制剂,IC50为 41 nM,Kd 为 68 nM。
T61522 Nrf2/HO-1 activator 2
Nrf2/HO-1 activator 2 (compound 13m), a difluoro-substituted derivative, is a highly potent activator of Nrf2/HO-1. It e...
T72687 Keap1-Nrf2-IN-11
Keap1-Nrf2-IN-11 是一种Keap1-Nrf2抑制剂,其KD2值为 0.21 nM。Keap1-Nrf2-IN-11 抑制 ROS 和 NO 的产生以及 TNF-α 的表达。Keap1-Nrf2-IN-11 通过增加 Nrf2...
T63987 Keap1-Nrf2-IN-14
Keap1-Nrf2-IN-14 是一种 KEAP1-NRF2 抑制剂,可有效破坏 KEAP1-NRF2 相互作用 (IC50: 75 nM),其对 KEAP1的 Kd=24 nM。Keap1-Nrf2-IN-14 可诱导 NRF2 靶基因...
T63294 Keap1-Nrf2-IN-5
Keap1-Nrf2-IN-5 是 Keap1-Nrf2 PPI (Keap1-Nrf2 protein-protein interaction) 的有效抑制剂 (IC50: 4.1 μM, Kd: 3.7 μM)。
T64190 Keap1-Nrf2-IN-12
eap1-Nrf2-IN-12 是一种 Keap1-Nrf2 的有效抑制剂 (IC50: 2.30 μM)。Keap1-Nrf2-IN-12 在人肝微粒体中具有代谢稳定性。
T61773 Keap1-Nrf2-IN-4
Keap1-Nrf2-IN-4, a powerful neddylation inhibitor, demonstrates significant anti-proliferation activity against MGC-803 ...
T64218 Keap1-Nrf2-IN-1 TFA
Keap1-Nrf2-IN-1 TFA (compound35) 是一种 Keap1-Nrf2 蛋白-蛋白相互作用抑制剂 (IC50: 43 nM),可以激活 Nrf2 调节的细胞保护反应。在细胞和体内模型中。Keap1-Nrf2-IN-1...
Nrf2-IN-1
T12253
synonym:
Target:
Nrf2 activator-1
T39719
synonym: Nrf2 activator-1
Target:
Nrf2-Activator-12G
T24546
synonym: Nrf2 Activator-IV,Nrf2 Activator IV
Target:
Keap1-Nrf2-IN-3
T39514
synonym: Keap1-Nrf2-IN-3
Target:
Keap1-Nrf2-IN-1
T11752
synonym: Keap1–Nrf2-IN-1
Target:
Nrf2 activator-6
T72697
synonym:
Target:
Nrf2 activator-4
T63016
synonym:
Target:
AChE/Nrf2 modulator 1
T72417
synonym:
Target:
Keap1-Nrf2-IN-9
T74600
synonym:
Target:
Keap1-Nrf2-IN-13
T72706
synonym:
Target:
Nrf2 activator-2
T61688
synonym:
Target:
Nrf2 activator-5
T63364
synonym:
Target:
Keap1-Nrf2-IN-6
T72760
synonym:
Target:
Nrf2/HO-1 activator 2
T61522
synonym:
Target:
Keap1-Nrf2-IN-11
T72687
synonym:
Target:
Keap1-Nrf2-IN-14
T63987
synonym:
Target:
Keap1-Nrf2-IN-5
T63294
synonym:
Target:
Keap1-Nrf2-IN-12
T64190
synonym:
Target:
Keap1-Nrf2-IN-4
T61773
synonym:
Target:
Keap1-Nrf2-IN-1 TFA
T64218
synonym:
Target:
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