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Search Results for " pda "

Targets

22

Compounds

Cat No. Product Name Synonyms Targets
T20571 Cis-PDA cis PDA GluR , NMDAR , iGluR
cis-PDA (cis PDA) is a general ionotropic receptor antagonist. cis-PDA acts by blocking NMDA, AMPA, and kainate-mediated responses.
T31792 Filaminast UNII-CDD69JC61J,Way-pda-641,WAY-PDA 641,CDD69JC61J PDE
Filaminast (UNII-CDD69JC61J) is an analog of a phosphodiesterase 4 inhibitor (PDE4 inhibitor) and roliplam, which is used as an anti-asthma drug.
T33808 12-Oxo phytodienoic acid 12-Oxo-Phytodienoic acid,12-OPDA,12-oxo PDA,OPDA Others
12-Oxo phytodienoic acid (12-oxo PDA) is an endogenous signal converter that increases alkaloid biosynthesis in E. californica cell cultures, increases b. dioica tendril curls, And inhibited jasmonic acid-induced program...
T4367 Mycro 3 Mycro-3 c-Myc , Autophagy
Mycro 3 is potent and selective for c-Myc in whole cell assays.
T18997 GPDA Glycylproline p-nitroanilide tosylate,GPN Others
GPDA (Glycylproline p-nitroanilide tosylate) is a substrate of X-Prolyl dipeptidyl-aminopeptidase in the enzyme assay.
T77661 H-NTPDase-IN-4 Phosphatase
h-NTPDase-IN-4 is a pan-inhibitor of NTPDase, which can inhibit h-NTPDase1, 1h-NTPDase2, h-NTPDase3, h-NTPDase8. The IC50 values were 3.58 μM, 10.21 μM, 0.13 μM and 13.57 μM, respectively.
T79622 H-NTPDase-IN-3 Phosphatase
h-NTPDase-IN-3 is an h-NTPDase inhibitor that inhibits h-NTPDase1, h-NTPDase2, h-NTPDase3 and h-NTPDase8.
T10877 CPDA Phosphatase
CPDA is a new potent inhibitor of SH2 domain-containing inositol phosphatase 2 (SHIP2).
T79492 H-NTPDase8-IN-1 Phosphatase
h-NTPDase8-IN-1 is a specific aminosulfonylbenzamide inhibitor of h-NTPDases8 (IC 50 = 0.28 ± 0.07 μM). h-NTPDase8-IN-1 can be used to study diseases brought about by aberrant h -NTPDase expression.
T79607 H-NTPDase-IN-2 hNTPDase-IN-2 Phosphatase
h-NTPDase-IN-2 is a broad-spectrum NTPDase inhibitor that inhibits multiple h-NTPDas isoforms.
T79491 H-NTPDase-IN-1 Phosphatase
h-NTPDase-IN-1 (Compound 3i) is an inhibitor of human NTPDase (h-NTPDase) with IC50 values of 2.88 μM for h-NTPDase1 and 0.72 μM for h-NTPDase3, indicating its potential utility for thrombosis, inflammation, diabetes, an...
T61377 NTPDase-IN-1
NTPDase-IN-1 (compound 5a) is a selective inhibitor of NTPDase enzymes. It shows inhibitory activity against h-NTPDase-1, h-NTPDase-2, and h-NTPDase-8 with IC50 values of 0.05 μM, 0.23 μM, and 0.54 μM, respectively. NTPD...
TQ0114 CMPDA GluR
CMPDA is a positive allosteric modulator of AMPA receptors (EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor).
T73552 BPDA2
BPDA2 is a highly selective and competitive SHP2 inhibitor, exhibiting IC50 values of 92.0 nM for SHP2, and 33.39 μM and 40.71 μM for SHP1 and SHP1B, respectively. This compound effectively downregulates mitogenic and ce...
T62703 NTPDase-IN-2
NTPDase-IN-2 (compound 5g) selectively inhibits NTPDase-2 and NTPDase-8 with IC50 values of 0.04 µM and 2.27 µM, respectively, and exhibits non-competitive inhibition towards h-NTPDase-1 and h-NTPDase-2, with a Km of 74 ...
T24604 PDAT Propyl Dimethyl Amino Tryptamine
PDAT is a noncompetitive Indolethylamine N-methyltransferase inhibitor.
T23179 PPDA Others
Subtype-selective NMDA receptor antagonist
T79623 H-NTPDase-IN-5 Phosphatase
h-NTPDase-IN-5 (compound 3b) serves as a pan-inhibitor of NTPDase, exhibiting inhibitory concentration 50 (IC50) values of 1.10 μM (h-NTPDase1), 44.73 μM (h-NTPDase2), 26.14 μM (h-NTPDase3), and 0.32 μM (h-NTPDase8).
T62633 NTPDase-IN-3
NTPDase-IN-3 (Compound 5e), an inhibitor of NTPDase, exhibits IC50 values of 0.38 μM (NTPDase3), 0.05 μM (NTPDase8), 0.21 μM (NTPDase1), and 1.07 μM (NTPDase2). It is utilized in cancer and thrombosis research [1].
T37396 13-epi-12-oxo Phytodienoic Acid
13-epi-12-oxo Phytodienoic acid (13-epi-12-oxo PDA) is a lipoxygenase metabolite of α-linolenic acid in the leaves of green plants such as corn. ω-3 and ω-6 polyunsaturated fatty acids in plants are substrates for plant ...
T68713 RX-RA 69
RX-RA 69 is a pyrimido-pyrimidine derivative and PDA-inhibitor which inhibits tumor cell induced platelet aggregation in vitro.
TQ0095 Brincidofovir CMX001,HDP-CDV Others , Antiviral , HSV
Brincidofovir (HDP-CDV) is an orally active, lipophilic form of cidofovir. It has enhanced activity compared to CDV against certain adenoviruses, herpesviruses, and orthopoxviruses.
TargetMol