T8883 |
Pizuglanstat
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Others
,
Prostaglandin Receptor
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Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor. |
T15681 |
L-161982
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Prostaglandin Receptor
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L-161982 is a selective antagonist of EP4 receptor. L-161982 could inhibit PGE2-induced ERK phosphorylation and cell pro... |
T5014 |
Prostaglandin E2
|
PGE2,Dinoprostone,Prostaglandin E2 (PGE2) |
Endogenous Metabolite
,
Prostaglandin Receptor
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Prostaglandin E2 is a hormone-like compound involved in various physiological processes, including smooth muscle contrac... |
T6399 |
AZD1981
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Prostaglandin Receptor
,
GPR
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AZD1981 is an effective and specific CRTh2 (DP2) receptor antagonist (IC50: 4 nM), showing >1000-fold selectivity over m... |
TQ0025 |
E7046
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Prostaglandin Receptor
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E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities. |
T14148 |
AH 6809
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Prostaglandin Receptor
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AH 6809 is an antagonist of EP and DP receptor(with Kis of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, ... |
T9153 |
Picotamide
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Others
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Picotamide has anticoagulant and fibrinolytic properties. |
T5505 |
Terutroban
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Prostaglandin Receptor
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Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis. |
T5386 |
Asapiprant
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Prostaglandin Receptor
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Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and se... |
T2664 |
Timapiprant
|
OC000459 |
Prostaglandin Receptor
,
GPR
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|
OC000459 is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM). |
T4635 |
Ralinepag
|
APD811 |
Prostaglandin Receptor
,
Others
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|
Ralinepag is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 5... |
T2428 |
TG6-10-1
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Prostaglandin Receptor
,
5-HT Receptor
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|
TG6-10-1 is an EP2 antagonist. |
T15133 |
Dinoprost
|
Prostaglandin F2a,PGF2α |
Endogenous Metabolite
|
|
Dinoprost is a naturally occurring prostaglandin. It is used in medicine to induce labor and as an abortifacient. |
T15712 |
Laropiprant
|
MK-0524 |
Prostaglandin Receptor
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|
Laropiprant is a potent and selective DP receptor antagonist (Ki: 0.57 nM and 2.95 nM for DP receptor and TP Receptor, r... |
T1978 |
GW627368
|
GW 627368X |
Prostaglandin Receptor
|
|
GW627368X is a novel, potent and selective antagonist of prostanoid EP4 receptor. |
T11211 |
EP4 receptor antagonist 1
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|
Prostaglandin Receptor
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EP4 receptor antagonist 1 inhibits human and mouse EP4 receptor with IC50s of 6.1 nM and 16.2 nM, respectively. IC50s >1... |
T16280 |
Nedocromil
|
FPL 59002 |
Histamine Receptor
,
Prostaglandin Receptor
,
Leukotriene Receptor
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Nedocromil inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and... |
T7652 |
AM211
|
AM211 free acid |
Prostaglandin Receptor
|
|
AM211 is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2) |
T1626 |
Prostaglandin E1
|
PGE1,Alprostadil |
Prostaglandin Receptor
,
Endogenous Metabolite
|
|
Alprostadil is the naturally occurring prostaglandin E1 (PGE1) which displays a variety of pharmacologic actions. Alpros... |
T3276 |
Benorilate
|
Benorylate,Benoral,Benortan,Salipran |
Prostaglandin Receptor
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Benorylate is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and a... |