T1889 |
CP-640186
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CP 640186 |
Acetyl-CoA Carboxylase
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CP 640186 是一种有效的乙酰辅酶 A 羧化酶 (ACC)抑制剂,抑制大鼠肝脏 ACC1 和大鼠骨骼肌 ACC2 的 IC50分别为 53 nM 和 61 nM。 |
T3622 |
CP-640186 hydrochloride
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CP 640186 HCl,盐酸CP-640186 |
Acetyl-CoA Carboxylase
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CP-640186 hydrochloride 是膜渗透性的乙酰辅酶A 羧化酶(ACC)抑制剂,抑制大鼠肝脏ACC1和大鼠骨骼肌ACC2的IC50为53 nM 和61 nM。 |
T27753 |
KT-362 fumarate
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KT-362 |
Sodium Channel
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Calcium Channel
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Potassium Channel
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KT-362 fumarate 是一种新型化合物,可作为钙通道、钾通道和钠通道的拮抗剂.KT-362 fumarate 通过影响心房肌肉细胞内钙动员导致血管舒张。KT-362 fumarate 对兔子的股动脉和基底动脉条有放松作用。 |
T37459 |
Lipoxin A5
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Lipoxin A5 (LXA5) is produced by enzymatic transformation of EPA by leukocytes. LXA5 slowly contracts pulmonary parenchy... |
T76430 |
GR 87389
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GR 87389 是一种有效的NK2受体拮抗剂。GR 87389 以竞争性方式拮抗 GA 64349 诱导的人类逼尿肌、前列腺和前列腺尿道平滑肌条收缩。 |
T3074L |
CHIR98014 HCl (252935-94-7 free base)
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CHIR-98014 hydrochloride,CT-98014,CHIR98014,CHIR98014 HCl,CHIR 98014,CHIR-98014 |
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CHIR98014 is a reversible, cell-permeable inhibitor of GSK3α and GSK3β (IC50s: 0.65 and 0.58 nM). Through its effects on... |
T35787 |
Obestatin (human) (trifluoroacetate salt)
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Obestatin is a 23 amino acid peptide hormone with a conserved C-terminal glycine residue and amidation site that is form... |
T37620 |
Leukotriene C4 methyl ester
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Leukotriene C4 (LTC4) is the parent cysteinyl-leukotriene produced by the LTC4 synthase-catalyzed conjugation of glutath... |
T35597 |
Neuromedin U-23 (rat) (trifluoroacetate salt)
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Neuromedin U-23 (NMU-23) is a neuropeptide involved in diverse biological processes, including smooth muscle contraction... |