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(1)
By Target- Cannabinoid Receptor
- GABA Receptor(1)
- cAMP(1)
- Others(3)
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Search Result
Results for "
negative allosteric modulator (nams)
" in TargetMol Product Catalog- Inhibitors & Agonists5
CB1R Allosteric modulator 1
T620162513102-41-3
CB1R Allosteric Modulator 1 (compound 11) is a potent allosteric modulator of CB1Rs, negatively affecting the functional activity of orthosteric ligands [NAM] at CB1Rs.
- $1,520
Size
QTY
CB1R Allosteric modulator 4
T613712633686-53-8
CB1R Allosteric modulator 4 is an effective and positive modulator of cannabinoid type-1 (CB1R), exhibiting significant biological activity. This compound inhibits the production of cAMP and demonstrates strong β-arrestin-2 recruitment [1].
- $1,520
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QTY
CB1R Allosteric modulator 3
T615622633686-36-7
CB1R Allosteric modulator 3 is a potent CB1R modulator that inhibits cAMP and β-Arrestin and can be used for the study of obesity and nicotine addiction.
- $35
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QTY
CB1R Allosteric modulator 2
T612762513102-64-0
CB1R Allosteric Modulator 2 (compound 18) is a potent negative allosteric modulator (NAM) of CB1R receptor activity, as demonstrated in previous studies [1].
- $1,520
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QTY
Basmisanil
T71651159600-41-5
Basmisanil (RG1662) is a negative allosteric modulator inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the treatment of cognitive impairments associated with Down syndrome.
- $32
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