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Search Result

Search Results for "parp"

Compounds

Cat No. Product Name
T70732 APX2014
APX2014 is a novel potent and specific Ref-1 inhibitor, blocking in vitro cell proliferation and activating apoptosis vi...
T41083 PNP-ADPr pNP-ADPr,ADP-ribose-pNP
pNP-ADPr is a colorimetric substrate employed in the first continuous activity assays for Poly(ADP-ribose) glycohydrolas...
T69185 INO-1001 methanesulfonate
INO-1001 methanesulfonate is an isoindolinone derivative and potent inhibitor of the nuclear enzyme poly (ADP-ribose) po...
T39147 Venadaparib hydrochloride IDX-1197 hydrochloride
Venadaparib hydrochloride (IDX-1197) is a potent and selective PARP inhibitor that exhibits significant anticancer prope...
T72017 6(5H)-Phenanthridinone
6(5H)-Phenanthridinone is an inhibitor of poly(ADP-ribose) polymerase 1 (PARP1) and PARP2. It decreases radiation-induce...
T63001 Antitumor agent-72
Antitumor agent-72 是一种有效的抗癌剂。Antitumor agent-72 具有抗癌活性，并通过激活 caspase-3 和裂解PARP 诱导细胞凋亡 (apoptosis)。Antitumor agent-72 可用于...
T68663 GPI-15427
GPI-15427 is a potent PARP-1 inhibitor capable of crossing the blood-brain barrier, which can significantly increased th...
T68878 L-2286
L-2286 is a novel PARP inhibitor. L-2286 exerted significant protective effect against ischemia-reperfusion-induced myoc...
T10896 CSRM617 Others
CSRM617 is a selective small molecule inhibitor of the transcription factor ONECUT2 (OC2, the main regulator of androgen...
T12292 Olaparib-d5 AZD2281 D5,KU0059436 D5,Olaparib D5 Others
Olaparib D5 is a deuterium labeled Olaparib. Olaparib is a potent and oral inhibitor of PARP.
T71757 SC-10914
SC10914 is a highly potent PARP inhibitor (PARP1 IC50 = 7.87 nM) with potent anti-proliferative activity against human B...
T69955 JPI-547 HCl
JPI 547, also known as NOV 1402, is an oral inhibitor of PARP 1/2 and Tankyrase 1/2. JPI-547 demonstrated anti-tumor act...
T62527 INO-1001
INO-1001 是一种有效的、选择性聚 (ADP-核糖) 聚合酶 (PARP) 抑制剂，具有抗肿瘤活性。INO-1001 是一种有效的辐射敏感性增强剂，能够利用干扰 DNA 修复机制，进而提高辐射诱导的细胞杀伤，使坏死细胞死亡。
T75074 6-Methoxypurine-9-β-D-5’(R)-C-methylriboside
6-Methoxypurine-9-β-D-5’(R)-C-methylriboside 是一种次黄嘌呤类似物。次黄嘌呤是一类主要存在于肌肉组织中的嘌呤碱基，由嘌呤氧化酶作用于黄嘌呤而产生的代谢物。次黄嘌呤有典型的抗炎作用，是潜在的内源性 ...
T36571 N-Descyclopropanecarbaldehyde Olaparib
N-Descyclopropanecarbaldehyde Olaparib, an Olaparib analogue, incorporates a DOTA moiety. It acts as a CRBN-based ligand...
T68536 WP-1034
WP-1034 is a novel Jak-Stat inhibitor, which is active against AML blasts. WP-1034 effectively inhibited proliferation o...
T71908 NU1085
NU1085 is a potent poly(ADP-ribose) polymerase (PARP) inhibitors have been developed that potentiate the cytotoxicity of...
T63522 Anticancer agent 64
Anticancer agent 64 (化合物 5m) 对 CCRF-CEM 细胞具有细胞毒性，其IC50为2.4 μM。Anticancer agent 64 通过诱导细胞凋亡表现出良好的抗癌活性。Anticancer agent 64...
T73403 Aviculin
Aviculin 是一种木聚糖苷，是一种有效的抗癌剂 (anticanceragent)。Aviculin 可降低 MCF-7 细胞代谢活性到 50% 以下，IC50为 75.47 μM。Aviculin 通过内在凋亡途径诱导乳腺癌细胞凋亡...
T64223 RMS5
RMS5 是一种汉防己碱类似物，是一种有效的 P-糖蛋白 (P-gp) 抑制剂。RMS5 对癌细胞具有显着的抗增殖和细胞毒作用。RMS5 略微降低抗凋亡 Bcl-2 家族蛋白 Bcl-XL 和 Mcl-1 的表达。RMS3 导致 PARP ...
APX2014
T70732
synonym:
Target:
pNP-ADPr
T41083
synonym: pNP-ADPr,ADP-ribose-pNP
Target:
INO-1001 methanesulfonate
T69185
synonym:
Target:
Venadaparib hydrochloride
T39147
synonym: IDX-1197 hydrochloride
Target:
6(5H)-Phenanthridinone
T72017
synonym:
Target:
Antitumor agent-72
T63001
synonym:
Target:
GPI-15427
T68663
synonym:
Target:
L-2286
T68878
synonym:
Target:
CSRM617
T10896
synonym:
Target:
Olaparib-d5
T12292
synonym: AZD2281 D5,KU0059436 D5,Olaparib D5
Target:
SC-10914
T71757
synonym:
Target:
JPI-547 HCl
T69955
synonym:
Target:
INO-1001
T62527
synonym:
Target:
6-Methoxypurine-9-β-D-5’(R)-C-methylriboside
T75074
synonym:
Target:
N-Descyclopropanecarbaldehyde Olaparib
T36571
synonym:
Target:
WP-1034
T68536
synonym:
Target:
NU1085
T71908
synonym:
Target:
Anticancer agent 64
T63522
synonym:
Target:
Aviculin
T73403
synonym:
Target:
RMS5
T64223
synonym:
Target:
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