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Search Results for " resistance "

412

Compounds

92

Natural Products

183

Recombinant Proteins

15

Libraries

Cat No. Product Name Synonyms Targets
T83892 33-BCRP Inhibitor 33-Breast Cancer Resistance Protein Inhibitor
33-BCRP inhibitor is a compound that blocks the action of breast cancer resistance protein (BCRP), enhancing the susceptibility of mitoxantrone-resistant H460/MX20 lung cancer cells to the cytotoxic effects of mitoxantro...
TQ0186 Ko 143 BCRP , ABC
Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).
T9982 PU23 MRP
PU 23 is an inhibitor of multidrug-resistant protein 4 (MRP4).
T21876 DC_AC50 Apoptosis , Others
DC_AC50 is a dual inhibitor of Atox1 and CCS (copper chaperones). Inhibiting intracellular copper chaperones as a means of reducing/preventing acquired chemotherapy resistance.DC_AC50 binding to Atox1 and CCS and reducin...
T13383 Zamicastat BIA 5-1058 BCRP , Hydroxylase , P-gp
Zamicastat (BIA 5-1058) is an inhibitor of dopamine β-hydroxylase (DBH), and is also a concentration-dependent dual inhibitor of P-gp and BCRP(IC50 values of 73.8 μM and 17.0 μM, respectively).
T4595 YHO-13177 YHO 13177,YHO13177 BCRP
YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells and no effect on P-glycoprotein–mediated paclitaxel resistance in MDR1-transduced human leukemia K562 cells.
T3581 KS176 Potassium Channel , BCRP
KS176 is a potent and selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter, showing no inhibitory activity against P-gp or MRP1.
T3971 CASIN Pirl1-related Compound 2 CDK , STAT , Ras
CASIN (Pirl1-related Compound 2) is a specific inhibitor of GTPase Cdc42 (IC50: 2 uM).
T8157 Centhaquin PMZ-2010,Centhaquine Others
Centhaquin (Centhaquine)e is an adrenergic receptor potentially for the treatment of postoperative pain and for the resuscitation of hypovolemic shock
T1248 Sulfanitran Antibacterial , Autophagy
Sulfanitran is a sulfonamide antibiotic used in the poultry industry.
T27617 Inz-1 P450
Inz-1 is an effective and fungal-selective inhibitor of mitochondrial cytochrome bc1 with IC50s of 8.092 and 45.320 μM for yeast and human. Inz-1 reverses Fluconazole or other triazole antifungals’ resistance in the path...
T12832 Amcenestrant SAR439859 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Amcenestrant (SAR439859) is an orally active, nonsteroidal and selective degrader of estrogen receptor (SERD). SAR439859 is a potent antagonist of ER (with an EC50 of 0.2 nM for ERα degradation).
T4628 Seladelpar MBX 8025 PPAR
Seladelpar (MBX 8025) has been used in trials studying the treatment of Hyperlipidemia.
T21955 GQ-16 PPAR
GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.
T7656 Apelin-13
Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor angiotensin II protein J (APJ), with an EC50 value of 0.37 ...
T38400 Triclabendazole sulfoxide TCBZ-SO BCRP , Parasite
Triclabendazole sulfoxide (TCBZ-SO) is a main plasma metabolite of Triclabendazole. Triclabendazole sulfoxide inhibits membrane transporter ABCG2/BCRP and exhibits anti-parasite effects.
T8596 Ceefourin 1 MRP
Ceefourin 1 is a highly selective multidrug resistance protein 4 (MRP4) inhibitor.
T2680 NVP-BVU972 c-Met/HGFR
NVP-BVU972 is a selective and potent Met inhibitor with IC50 of 14 nM.
T12341 P-gp inhibitor 1 Others , P-gp
P-gp inhibitor 1 inhibits reversing P-glycoprotein-mediated multidrug resistance with an EC50 of 57.9 nM (K562/A02 cells).
T8426 Encequidar HM30181,HM30181A P-gp
Encequidar (HM30181A) is a potent and selective P-glycoprotein inhibitor.
T3071 Olverembatinib GZD 824 Bcr-Abl
Olverembatinib (GZD 824) is an orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT, IC50: 0.34 nM) and Bcr-Abl(T315I, IC50: 0.68 nM).
T22459 Xanthinol Nicotinate Angioamin,Complamin Others
Xanthinol Nicotinate (Complamin) is a potent vasodilator that can easily enter the cell and causes an increase in glucose metabolism resulting in an increased energy.
T4337 PCI 29732 PCI29732,PCI-29732 Others , BCRP , BTK
PCI 29732 is a selective and irreversible Btk inhibitor with IC50 of 8.2 nM in a FRET based biochemical enzymology assay.
T2620 G-749 G749 Apoptosis , FLT , c-RET , TAM Receptor , Aurora Kinase
G-749, a new-type FLT3 inhibitor, exhibits effective and sustained inhibition of the FLT3 wild type and mutants.
T16561 Polyoxyethylene stearate POES Antibacterial , P-gp
Polyoxyethylene stearate (POES) is an agent of non-ionic emulsifying.
T6287 Tariquidar XR9576 P-gp
Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.
T11071 Dofequidar fumarate MS-209 P-gp
Dofequidar fumarate (MS-209)(MS-209 fumarate), a quinoline-based compound administered orally, is known for counteracting multidrug resistance (MDR) through the inhibition of ABCB1/P-glycoprotein (P-gp) and ABCC1/MDR-ass...
T2657 Elacridar GW0918,GW120918,GF120918,GG918 BCRP , P-gp
Elacridar (GG918) (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor.
T9179 CLP-3094 2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE Androgen Receptor
CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a selective and potent GP...
T0351 Risperidone Risperidal,R 64 766 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , P-gp
Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
T1275 Phentolamine mesylate Phentolamine methanesulfonate,Phentolamine mesilate Adrenergic Receptor
Phentolamine mesylate (Phentolamine methanesulfonate) is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, vasospasm of RAYNAUD DISEAS...
T15735 Leptomycin B CI 940,LMB CRM1 , Antibiotic , Antifungal
Leptomycin B (LMB) is a potent inhibitor of the nuclear export of proteins and is a potent antifungal antibiotic blocking the eukaryotic cell cycle. Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a ...
T7714 Temocapil Tyrosinase
Temocapril is an inhibitor of tyrosine kinase.
T4059 Selamectin UK-124114 Chloride channel , P-gp , Parasite
Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in nematodes. In an H. contortus larval development assay, sel...
T8389 Trifluoperazine trifluoroperazine CaMK , Dopamine Receptor , Influenza Virus , Adrenergic Receptor , P-gp , Autophagy
Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
T13416 ZX-29 ALK
ZX-29 is a potent and selective inhibitor of ALK(IC50 of 2.1 nM, 1.3 nM and 3.9 nM for ALK, ALK L1196M and ALK G1202R mutations, respectively), and also induces protective autophagy and has antitumor effect.
T11578L Encequidar mesylate HM30181 mesylate,HM30181A mesylate P-gp
Encequidar mesylate (HM30181A mesylate) is a competitive P-glycoprotein inhibitor.
T2429 Olverembatinib dimesylate GZD824 Dimesylate,HQP1351 Bcr-Abl
Olverembatinib dimesylate (GZD824 Dimesylate) is a novel orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT) and Bcr-Abl(T315I).
T1967 AZD-3463 ALK/IGF1R inhibitor Apoptosis , IGF-1R , ALK , Autophagy
AZD-3463 (ALK/IGF1R inhibitor) , an orally bioavailable ALK inhibitor (Ki: 0.75 nM), can inhibit IGF1R with equivalent potency.
T16028 IMB-XH1 Mcl1-IN-2 BCL , Antibacterial
IMB-XH1 (Mcl1-IN-2) is a myeloid cell factor 1 (Mcl-1) inhibitor.
T0100L Atazanavir Zrivada,Reyataz,Latazanavir,BMS-232632 P450 , SARS-CoV , HIV Protease , P-gp
Atazanavir (BMS-232632)(BMS-232632) is an highly effective HIV-1 protease inhibitor.
T1634 Glibenclamide Glyburide Potassium Channel , Mitochondrial Metabolism , CFTR , P-gp , Autophagy
Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.
T20656 Verapamil NSC 135784,NSC-135784,CP-16533-1,(±)-Verapamil P450 , Calcium Channel , P-gp
Verapamil (CP-16533-1) is a calcium channel blocker and an orally active and effective inhibitor of P-gp. Verapamil inhibits CYP3A4 and can be used in studies about the treatment of high blood pressure, heart arrhythmias...
T10353 APX-115 free base Ewha-18278 free base NADPH-oxidase , NADPH
APX-115 free base (Ewha-18278 free base) (Ewha-18278 free base) is a potent, orally active pan NADPH oxidase (Nox) inhibitor (Kis: 1.08 μM, 0.57 μM, and 0.63 μM for Nox1, Nox2, and Nox4). APX-115 effectively prevents kid...
T2330 Rilpivirine TMC278,R278474,DB08864 HIV Protease , Reverse Transcriptase
Rilpivirine (R278474) is a diarylpyrimidine derivative and reverse transcriptase inhibitor with antiviral activity against HIV-1 that is used in the treatment of HIV infections.
T16339 Norverapamil hydrochloride (±)-Norverapamil hydrochloride,D591 hydrochloride Calcium Channel , P-gp , Drug Metabolite
Norverapamil hydrochloride (D591 hydrochloride) ((±)-Norverapamil hydrochloride) is an N-demethylated metabolite of Verapamil and it is an L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor.
T14364 AZ-Dyrk1B-33 3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine DYRK
AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.
T1010 Verapamil hydrochloride Manidon,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride P450 , Calcium Channel , P-gp
Verapamil hydrochloride (Verapamil HCl) is a calcium channel blocker that is a class IV anti-arrhythmia agent.
T0100 Atazanavir sulfate BMS-232632,BMS-232632 sulfate P450 , SARS-CoV , HIV Protease , P-gp
Atazanavir sulfate (BMS-232632 sulfate) is an azapeptide and HIV-PROTEASE INHIBITOR that is used in the treatment of HIV INFECTIONS and AIDS in combination with other ANTI-HIV AGENTS.
T1222 Trifluoperazine dihydrochloride Trifluoperazine 2HCl,SKF5019,Urinox CaMK , Dopamine Receptor , Influenza Virus , Adrenergic Receptor , P-gp , Autophagy
Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.

Compounds

33-BCRP Inhibitor
T83892
Synonym: 33-Breast Cancer Resistance Protein Inhibitor
Target:
Ko 143
TQ0186
Synonym:
Target: BCRP, ABC
PU23
T9982
Synonym:
Target: MRP
DC_AC50
T21876
Synonym:
Target: Apoptosis, Others
Zamicastat
T13383
Synonym: BIA 5-1058
Target: BCRP, Hydroxylase, P-gp
YHO-13177
T4595
Synonym: YHO 13177,YHO13177
Target: BCRP
KS176
T3581
Synonym:
Target: Potassium Channel, BCRP
CASIN
T3971
Synonym: Pirl1-related Compound 2
Target: CDK, STAT, Ras
Centhaquin
T8157
Synonym: PMZ-2010,Centhaquine
Target: Others
Sulfanitran
T1248
Synonym:
Target: Antibacterial, Autophagy
Inz-1
T27617
Synonym:
Target: P450
Amcenestrant
T12832
Synonym: SAR439859
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Seladelpar
T4628
Synonym: MBX 8025
Target: PPAR
GQ-16
T21955
Synonym:
Target: PPAR
Apelin-13
T7656
Synonym:
Target:
Triclabendazole sulfoxide
T38400
Synonym: TCBZ-SO
Target: BCRP, Parasite
Ceefourin 1
T8596
Synonym:
Target: MRP
NVP-BVU972
T2680
Synonym:
Target: c-Met/HGFR
P-gp inhibitor 1
T12341
Synonym:
Target: Others, P-gp
Encequidar
T8426
Synonym: HM30181,HM30181A
Target: P-gp
Olverembatinib
T3071
Synonym: GZD 824
Target: Bcr-Abl
Xanthinol Nicotinate
T22459
Synonym: Angioamin,Complamin
Target: Others
PCI 29732
T4337
Synonym: PCI29732,PCI-29732
Target: Others, BCRP, BTK
G-749
T2620
Synonym: G749
Target: Apoptosis, FLT, c-RET, TAM Receptor, Aurora Kinase
Polyoxyethylene stearate
T16561
Synonym: POES
Target: Antibacterial, P-gp
Tariquidar
T6287
Synonym: XR9576
Target: P-gp
Dofequidar fumarate
T11071
Synonym: MS-209
Target: P-gp
Elacridar
T2657
Synonym: GW0918,GW120918,GF120918,GG918
Target: BCRP, P-gp
CLP-3094
T9179
Synonym: 2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE
Target: Androgen Receptor
Risperidone
T0351
Synonym: Risperidal,R 64 766
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, P-gp
Phentolamine mesylate
T1275
Synonym: Phentolamine methanesulfonate,Phentolamine mesilate
Target: Adrenergic Receptor
Leptomycin B
T15735
Synonym: CI 940,LMB
Target: CRM1, Antibiotic, Antifungal
Temocapil
T7714
Synonym:
Target: Tyrosinase
Selamectin
T4059
Synonym: UK-124114
Target: Chloride channel, P-gp, Parasite
Trifluoperazine
T8389
Synonym: trifluoroperazine
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
ZX-29
T13416
Synonym:
Target: ALK
Encequidar mesylate
T11578L
Synonym: HM30181 mesylate,HM30181A mesylate
Target: P-gp
Olverembatinib dimesylate
T2429
Synonym: GZD824 Dimesylate,HQP1351
Target: Bcr-Abl
AZD-3463
T1967
Synonym: ALK/IGF1R inhibitor
Target: Apoptosis, IGF-1R, ALK, Autophagy
IMB-XH1
T16028
Synonym: Mcl1-IN-2
Target: BCL, Antibacterial
Atazanavir
T0100L
Synonym: Zrivada,Reyataz,Latazanavir,BMS-232632
Target: P450, SARS-CoV, HIV Protease, P-gp
Glibenclamide
T1634
Synonym: Glyburide
Target: Potassium Channel, Mitochondrial Metabolism, CFTR, P-gp, Autophagy
Verapamil
T20656
Synonym: NSC 135784,NSC-135784,CP-16533-1,(±)-Verapamil
Target: P450, Calcium Channel, P-gp
APX-115 free base
T10353
Synonym: Ewha-18278 free base
Target: NADPH-oxidase, NADPH
Rilpivirine
T2330
Synonym: TMC278,R278474,DB08864
Target: HIV Protease, Reverse Transcriptase
Norverapamil hydrochloride
T16339
Synonym: (±)-Norverapamil hydrochloride,D591 hydrochloride
Target: Calcium Channel, P-gp, Drug Metabolite
AZ-Dyrk1B-33
T14364
Synonym: 3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine
Target: DYRK
Verapamil hydrochloride
T1010
Synonym: Manidon,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride
Target: P450, Calcium Channel, P-gp
Atazanavir sulfate
T0100
Synonym: BMS-232632,BMS-232632 sulfate
Target: P450, SARS-CoV, HIV Protease, P-gp
Trifluoperazine dihydrochloride
T1222
Synonym: Trifluoperazine 2HCl,SKF5019,Urinox
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
1 2 3 4 5 6 7 8 9
Cat No. Product Name Synonyms Targets
T10815 Cinnamoylglycine Endogenous Metabolite
Cinnamoylglycine is a glycine conjugate of cinnamic acid and a urinary metabolite in humans. It is used as a potential urinary biomarker.
T3881 Vaccarin Integrin , Akt , PERK , AMPK
Vaccarin is a major flavonoid glycoside in Vaccariae semen, its biotransformation pathways involves methylation, hydroxylation, glycosylation and deglycosylation.
TN1651 Furanodiene Apoptosis , PARP , Reactive Oxygen Species , Caspase , CDK , P-gp
Furanodiene has anti-inflammatory and antioxidant activities, it is active against gram-positive bacteria and Candida albicans.
T3S0012 Coniferyl ferulate P-gp , GST
Coniferyl ferulate is a strong inhibitor of glutathione S-transferase (GST) isolated from Radix Angelicae sinensis. It shows strong inhibition of human placental GST (IC50: 0.3 μM). It also reverses multidrug resistance ...
T6670 Silymarin Silybin B SARS-CoV
Silymarin (Silybin B) (Silybin B) is a polyphenolic flavonoid that extracts from the milk thistle or seeds of Silybum marianum. It is used in the prevention and treatment of liver diseases.
T2S0223 Isosinensetin 6-Demethoxynobiletin Antioxidant , HIV Protease , Antibacterial , P-gp
1. Isosinensetin (6-Demethoxynobiletin) shows antioxidant and HIV-1 protease inhibiting activities.
TN4761 Phellamurin P-gp
Phellamurin inhibits intestinal P-glycoprotein in a dose-dependent manner, there is a serious interaction occurred between Phellamurin with cyclosporin, to ensure the efficacy of cyclosporin, we suggest that the coadmini...
T2869 Emodin Frangula emodin SARS-CoV , Casein Kinase , Autophagy
Emodin (Frangula emodin) is a naturally occurring anthraquinone present in the roots and barks of numerous plants; exerts antiproliferative effects in Y cells that are regulated by different signaling pathways.
TJS1159 Chrysosplenetin Chrysosptertin B P450 , Ferroptosis , P-gp
Chrysosplenetin is a metabolic inhibitor of artemisinin.
T2S0271 Voacamine Voacanginine Cannabinoid Receptor , P-gp
Voacamine (Voacanginine) is an indole alkaloid. Voacamine exhibits potent cannabinoid CB1 receptor antagonistic activity. Voacamine also inhibits P-glycoprotein (P-gp) action in multidrug-resistant tumor cells.Voacangini...
T3002 Piperine 1-Piperoylpiperidine,Bioperine P450 , Endogenous Metabolite , P-gp , Autophagy
Piperine (Bioperine) , a alkaloid, has been used in trials studying the treatment of multiple myeloma and deglutition disorders.
T19458 N-Hydroxypipecolic acid 1-Hydroxy-2-piperidinecarboxylic acid,NHP Others
N-Hydroxypipecolic acid (NHP) is a plant metabolite and a systemic acquired resistance (SAR) regulator.
TL0006 Cichoric Acid Dicaffeoyltartaric acid,Chicoric Acid Reactive Oxygen Species , HIV Protease
Cichoric Acid (Dicaffeoyltartaric acid) is a potent inhibitor of human immunodeficiency virus type-1 (HIV-1) integrase and the replication in tissues. It also a class of cannabinomimetics with CB2 receptor-dependent and ...
T2S1200 Sinapine Antioxidant , P-gp , AChE
1. Sinapine, an alkaloid from seeds of the cruciferous species, can be used as an effective natural compound for chemo-resistance. 2. Sinapine has antioxidant and radio-protective activities.
T4034 Solamargine Solamargin,δ-Solanigrine Apoptosis , p38 MAPK , P-gp , STAT
Solamargine (δ-Solanigrine) is a major steroidal alkaloid glycoside extracted from a traditional Chinese medicine herb, Solanum nigrum L. (SNL); has been shown to inhibit growth and induce apoptosis of various cancer cel...
T3392 Sinapine thiocyanate P-gp , AChE
Sinapine Thiocyanate, is a derivative of Sinapine (S486605), an alkaloidal amine found in black mustard seeds. It is the choline ester of Sinapic Acid (S486800). It is also a phenolic-chloine conjugates, acting as anti-o...
T2799 (20S)-Protopanaxadiol 20-Epiprotopanaxadiol,20(S)-APPD Apoptosis , Reactive Oxygen Species , P-gp
(20S)-Protopanaxadiol (20-Epiprotopanaxadiol) (20-Epiprotopanaxadiol), an apoptosis inducer, is an aglycon metabolic derivative of the protopanaxadiol-type ginseng saponin.
TN1525 Convallatoxin NF-κB , P-gp , PPAR
Convallatoxin is a natural product
TN1757 Hypophyllanthin Potassium Channel , Calcium Channel , P-gp
Hypophyllanthin and phyllanthin have antitumour effects against Ehrlich Ascites Carcinoma in mice.
T19768 γ-Tocotrienol gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol Others
γ-Tocotrienol (Plastochromanol) is one of the four types of tocotrienol, a type of vitamin E. Itl is also a radioprotector, antioxidant. It shows antitumor and antihypertensive effects in vivo.
T4085 Paris saponin VII Chonglou Saponin VII,Polyphyllin-VII,Dioscinin,Paris saponin-VII Apoptosis , BCL , Others , PARP , p38 MAPK , Akt , Caspase , P-gp , Autophagy
Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.
TCS2336 Evodine P-gp
1. Evodine has antinociceptive activity.
T15355 Fumitremorgin C 12α-Fumitremorgin C BCRP , Antibacterial , Antibiotic , ABC
Fumitremorgin C (12α-Fumitremorgin C) is a mycotoxin and inhibits ABCG2/BRCP.
TN3150 6,8-Diprenylnaringenin Senegalensin,Lonchocarpol A BCRP , ABC
6,8-Diprenylnaringenin (Senegalensin) is a natural product from hop Humulus lupulus. 6,8-Diprenylnaringenin is a breast cancer resistance protein(BCRP) inhibitor with some estrogenicity.
TN6339 (R)-5-Hydroxy-1,7-diphenylheptan-3-one (5R)-Dihydroyashabushiketol Others
(R)-5-Hydroxy-1,7-diphenylheptan-3-one ((5R)-Dihydroyashabushiketol) is extracted from the rhizomes of Alpinia officinarum, a Chinese medicinal herb. (R)-5-Hydroxy-1,7-diphenylheptan-3-one inhibits melanogenesis in theop...
T2831 Glycocholic acid Glycocholate,cholylglycine Others , Endogenous Metabolite
Glycocholic acid (Glycocholate) is a bile acid with anticancer activity. Glycocholic acid targets against pump resistance-related and non-pump resistance-related pathways.
T3S2019 Lathyrol Others
1.Lathyrol diterpenes is a modulator of P-glycoprotein dependent multidrug resistance.
T3S2381 Perillene 3-Isohexenylfuran,Perillen Others , Antibacterial
Perillene (3-Isohexenylfuran) is an actiive constituent in the drug which promotes enterocinesia. Perillen demonstrates strong resistance activity against staphylococcus aureus and E.coli.
T4461 3,5-Diiodo-L-thyronine Diiodothyronine Thyroid hormone receptor(THR) , Endogenous Metabolite
3,5-Diiodo-L-thyronine (Diiodothyronine) is an iodinated thyronine hormone that regulates gene activity affecting processes such as homeostasis, lipid metabolism and insulin resistance.
T4797 DEHP Bis(2-ethylhexyl) phthalate Others , Endogenous Metabolite
DEHP (Bis(2-ethylhexyl) phthalate) is used to impart softness and flexibility to PVC products. DEHP has been implicated in obesity and insulin resistance. DEHP inhibits prostaglandin synthesis and adversely affects the e...
T5777 Phaseoloidin Others
Phaseoloidin, a homogentisic acid glucoside from Nicotiana attenuata trichomes, contributes to the plant's resistance against lepidopteran herbivores.
T6S1842 Tenacissoside G Tenacissimoside A Others
Tenacissoside G, a C21 steroid derived from the stems of Marsdenia tenacissima, can reverse multidrug resistance in cancer cells exhibiting overexpression of P-glycoprotein.
T2A2486 3',​4',​5',​5,​7-​Pentamethoxyflavone 5,7,3',4',5'-Pentamethoxyflavone Nrf2
3',4',5',5,7-Pentamethoxyflavone is a naturally occurring brassinosteroid compound from the Rutaceae family that exhibits resistance to cancer cells by inhibiting the Nrf2 pathway to overcome chemotherapeutically active ...
T4A2399 Cinobufotalin IL Receptor , Akt , MRP , P-gp
Cinobufotalin is a main cardiac toxin in toad, it is a novel anti-HCC agent, it induces growth inhibition and apoptosis in cultured HCC cells through ceramide production. Cinobufotalin is also an effective reversal agent...
T15091 Decoyinine Decynylene,Angustmycin A
Decoyinine (Decynylene), a selective inhibitor of GMP synthase, is a novel potential microbial insecticide, a secondary metabolite produced by Streptomyces hygroscopicus.Decoyinine induces resistance in rice to the small...
T0950 Neomycin sulfate Framycin sulfate Phospholipase , ribosome , Antibacterial , Antibiotic
Neomycin sulfate (Framycin sulfate) is a broad-spectrum aminoglycoside antibiotic that blocks the synthesis of bacterial proteins in order to exert antimicrobial activity. Neomycin sulfate is commonly used to screen prok...
T4785 Oxfenicine 4-Hydroxy-L-phenylglycine Others
Oxfenicine (4-Hydroxy-L-phenylglycine) is a carnitine palmitoyltransferase-1 inhibitor. Oxfenicine improves whole-body glucose tolerance and insulin sensitivity in high-fat diet-induced obese mouse with insulin resistanc...
T6S0095 Genkwanin 7-O-Methylapigenin,Puddumetin,Apigenin 7-methyl ether Virus Protease
1. Genkwanin (Apigenin 7-methyl ether) exerts its anti-inflammatory effect mainly through the regulation of the miR-11/MKP-1/MAPK pathway. 2. Genkwanin is transported by both passive diffusion and multidrug resistance pr...
T3208 Brevianamide F Cyclo-L-tryptophyl-L-proline,cyclo-(L-Trp-L-Pro),Cyclo(L-Pro-L-Trp) BCRP , PI3K , Antibacterial
Brevianamide F (Cyclo(L-Pro-L-Trp)), also known as cyclo-(L-Trp-L-Pro), belongs to a class of naturally occurring 2,5-diketopiperazines. Brevianamide F possess interesting breast cancer resistance protein inhibitory acti...
T2S0265 Robinin NSC 9222 TLR
Flavone glycoside from Robinia with antibacterial and diuretic properties; derived from kaempferol.The ability of robinin to reverse the multidrug resistance of the human colon cancer cell line Colo 320 expreβing MDR1/LR...
TN1921 Meloside A Isovitexin 2''-O-glucoside,Isovitexin 2''-O-β-D-glucoside Others
Meloside A (Isovitexin 2''-O-β-D-glucoside) is a phenylpropanoid extracted from barley. Meloside A exhibits antioxidant and protective properties against excess UV-B radiation and has been linked to resistance to pathoge...
T1181 Gefitinib ZD1839 EGFR , Tyrosine Kinases , Autophagy
Gefitinib (ZD1839) is an EGFR first-generation inhibitor with oral activity that inhibits the EGFR 19 Del and L858R mutations. Gefitinib has antitumor activity and is used for the treatment of EGFR-mutated non-small-cell...
TN2256 Taccalonolide B Microtubule Associated
Taccalonolide B is effective in vitro against cell lines that overexpress P-glycoprotein (Pgp) and multidrug-resistance protein (MRP7). Taccalonolide B inhibits growth of SK-OV-3 cells with an IC50 of 208 nM.
T1273 Diacerein Diacerhein,Fisiodar,Diacetylrhein IL Receptor , Interleukin
Diacerein (Fisiodar) is a prodrug which is metabolized to rhein. It is currently approved in France for the treatment of osteoarthritis although the use of diacerein is restricted due to the side effects including sevre ...
T6S1885 Benzoylmesaconine Mesaconine 14-benzoate Others
Benzoylmesaconine (Mesaconine 14-benzoate) is the most abundant component of Wutou decoction, which is widely used in China because of its therapeutic effect on rheumatoid arthritis. Benzoylmesconine has analgesic activi...
T4S2128 Bilobetin PKA , PPAR
Bilobetin ameliorates insulin resistance by PKA-mediated phosphorylation of PPARα in rats fed a high-fat diet.
T1022 Hygromycin B Hygrovetine ribosome , Antibacterial , Antibiotic , Antifungal
Hygromycin B (Hygrovetine) is an aminoglycoside antibiotic that inhibits protein synthesis by interfering with translocation and causing mistranslation of the 70S ribosome. Hygromycin B can be used to screen prokaryotic ...
T5S1286 (+)-Columbianetin (S)-Columbianetin,Columbianetin Antifungal
(+)-Columbianetin ((S)-Columbianetin) is a new phytoalexin associated with celery (Apium graveolens) resistance to pathogens during storage, it also has antifungal activity. (+)-Columbianetin has anti-inflammatory effect...
Fr13883 3-Methoxyphenylacetic acid Others
3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid...
T6S0232 Eriodictyol Huazhongilexone Influenza Virus , DNA/RNA Synthesis , Nrf2 , Endogenous Metabolite
1. Eriodictyol (Huazhongilexone) is a flavonoid with anti-inflammatory and antioxidant activities. 2. Eriodictyol may possess antidiabetic properties through increasing glucose uptake and improving insulin resistance. 3....
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Natural Products

Cinnamoylglycine
T10815
Synonym:
Target: Endogenous Metabolite
Vaccarin
T3881
Synonym:
Target: Integrin, Akt, PERK, AMPK
Furanodiene
TN1651
Synonym:
Target: Apoptosis, PARP, Reactive Oxygen Species, Caspase, CDK, P-gp
coniferyl ferulate
T3S0012
Synonym:
Target: P-gp, GST
Silymarin
T6670
Synonym: Silybin B
Target: SARS-CoV
Isosinensetin
T2S0223
Synonym: 6-Demethoxynobiletin
Target: Antioxidant, HIV Protease, Antibacterial, P-gp
Phellamurin
TN4761
Synonym:
Target: P-gp
Emodin
T2869
Synonym: Frangula emodin
Target: SARS-CoV, Casein Kinase, Autophagy
Chrysosplenetin
TJS1159
Synonym: Chrysosptertin B
Target: P450, Ferroptosis, P-gp
Voacamine
T2S0271
Synonym: Voacanginine
Target: Cannabinoid Receptor, P-gp
Piperine
T3002
Synonym: 1-Piperoylpiperidine,Bioperine
Target: P450, Endogenous Metabolite, P-gp, Autophagy
N-Hydroxypipecolic acid
T19458
Synonym: 1-Hydroxy-2-piperidinecarboxylic acid,NHP
Target: Others
Cichoric Acid
TL0006
Synonym: Dicaffeoyltartaric acid,Chicoric Acid
Target: Reactive Oxygen Species, HIV Protease
Sinapine
T2S1200
Synonym:
Target: Antioxidant, P-gp, AChE
Solamargine
T4034
Synonym: Solamargin,δ-Solanigrine
Target: Apoptosis, p38 MAPK, P-gp, STAT
Sinapine thiocyanate
T3392
Synonym:
Target: P-gp, AChE
(20S)-Protopanaxadiol
T2799
Synonym: 20-Epiprotopanaxadiol,20(S)-APPD
Target: Apoptosis, Reactive Oxygen Species, P-gp
Convallatoxin
TN1525
Synonym:
Target: NF-κB, P-gp, PPAR
Hypophyllanthin
TN1757
Synonym:
Target: Potassium Channel, Calcium Channel, P-gp
γ-Tocotrienol
T19768
Synonym: gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol
Target: Others
Paris saponin VII
T4085
Synonym: Chonglou Saponin VII,Polyphyllin-VII,Dioscinin,Paris saponin-VII
Target: Apoptosis, BCL, Others, PARP, p38 MAPK, Akt, Caspase, P-gp, Autophagy
Evodine
TCS2336
Synonym:
Target: P-gp
Fumitremorgin C
T15355
Synonym: 12α-Fumitremorgin C
Target: BCRP, Antibacterial, Antibiotic, ABC
6,8-Diprenylnaringenin
TN3150
Synonym: Senegalensin,Lonchocarpol A
Target: BCRP, ABC
(R)-5-Hydroxy-1,7-diphenylheptan-3-one
TN6339
Synonym: (5R)-Dihydroyashabushiketol
Target: Others
Glycocholic acid
T2831
Synonym: Glycocholate,cholylglycine
Target: Others, Endogenous Metabolite
Lathyrol
T3S2019
Synonym:
Target: Others
Perillene
T3S2381
Synonym: 3-Isohexenylfuran,Perillen
Target: Others, Antibacterial
3,5-Diiodo-L-thyronine
T4461
Synonym: Diiodothyronine
Target: Thyroid hormone receptor(THR), Endogenous Metabolite
DEHP
T4797
Synonym: Bis(2-ethylhexyl) phthalate
Target: Others, Endogenous Metabolite
Phaseoloidin
T5777
Synonym:
Target: Others
Tenacissoside G
T6S1842
Synonym: Tenacissimoside A
Target: Others
3',​4',​5',​5,​7-​Pentamethoxyflavone
T2A2486
Synonym: 5,7,3',4',5'-Pentamethoxyflavone
Target: Nrf2
Cinobufotalin
T4A2399
Synonym:
Target: IL Receptor, Akt, MRP, P-gp
Decoyinine
T15091
Synonym: Decynylene,Angustmycin A
Target:
Neomycin sulfate
T0950
Synonym: Framycin sulfate
Target: Phospholipase, ribosome, Antibacterial, Antibiotic
Oxfenicine
T4785
Synonym: 4-Hydroxy-L-phenylglycine
Target: Others
Genkwanin
T6S0095
Synonym: 7-O-Methylapigenin,Puddumetin,Apigenin 7-methyl ether
Target: Virus Protease
Brevianamide F
T3208
Synonym: Cyclo-L-tryptophyl-L-proline,cyclo-(L-Trp-L-Pro),Cyclo(L-Pro-L-Trp)
Target: BCRP, PI3K, Antibacterial
Robinin
T2S0265
Synonym: NSC 9222
Target: TLR
Meloside A
TN1921
Synonym: Isovitexin 2''-O-glucoside,Isovitexin 2''-O-β-D-glucoside
Target: Others
Gefitinib
T1181
Synonym: ZD1839
Target: EGFR, Tyrosine Kinases, Autophagy
Taccalonolide B
TN2256
Synonym:
Target: Microtubule Associated
Diacerein
T1273
Synonym: Diacerhein,Fisiodar,Diacetylrhein
Target: IL Receptor, Interleukin
Benzoylmesaconine
T6S1885
Synonym: Mesaconine 14-benzoate
Target: Others
Bilobetin
T4S2128
Synonym:
Target: PKA, PPAR
Hygromycin B
T1022
Synonym: Hygrovetine
Target: ribosome, Antibacterial, Antibiotic, Antifungal
(+)-Columbianetin
T5S1286
Synonym: (S)-Columbianetin,Columbianetin
Target: Antifungal
3-Methoxyphenylacetic acid
Fr13883
Synonym:
Target: Others
Eriodictyol
T6S0232
Synonym: Huazhongilexone
Target: Influenza Virus, DNA/RNA Synthesis, Nrf2, Endogenous Metabolite

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPJ-00871 BAR Protein, S. hygroscopicus, Recombinant Streptomyces hygroscopicus E. coli
Phosphinothricin N-acetyltransferase (PAT) is an enzyme that acetylates the free NH2 group of L-phosphinothricin (L-PPT) in the presence of acetyl-CoA as a co-substrate. It is highly specific for L-PPT and does not acety...
TMPY-05556 Adiponectin Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
Adiponectin (ADIPOQ), or 30 kDa adipocyte complement-related protein (Acrp30) is a protein secreted by adipose tissue, which acts to reduce insulin resistance and atherogenic damage, but it also exerts actions in other t...
TMPY-02848 Adiponectin Protein, Human, Recombinant (hFc) Human HEK293
Adiponectin (ADIPOQ), or 30 kDa adipocyte complement-related protein (Acrp30) is a protein secreted by adipose tissue, which acts to reduce insulin resistance and atherogenic damage, but it also exerts actions in other t...
TMPY-01146 Insulin Receptor Protein, Human, Recombinant (long isoform, His) Human HEK293
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to the protein kinase superfamily and exists as a tetramer consisting of two alpha subunits and two beta...
TMPY-01009 TGFBI Protein, Human, Recombinant (His) Human HEK293
TGFBI is an RGD-containing protein that binds to type I, II and IV collagens. The RGD motif is found in many extracellular matrix proteins modulating cell adhesion and serves as a ligand recognition sequence for several ...
TMPY-04069 Neurotrophin 3 Protein, Human, Recombinant Human E. coli
NTF3 (Neurotrophin 3) is a Protein Coding gene. The protein encoded by this gene is a member of the neurotrophin family, that controls the survival and differentiation of mammalian neurons. This protein is closely relate...
TMPY-00971 CEACAM6 Protein, Human, Recombinant (His) Human HEK293
Carcinoembryonic antigen-related cell adhesion molecule 6 (CEACAM6), also known as nonspecific crossreacting antigen (NCA) and CD66c, is one of seven human CEACAM family members within the immunoglobulin superfamily. It ...
TMPY-05850 CEACAM6 Protein, Cynomolgus, Recombinant (His) Cynomolgus HEK293
Carcinoembryonic antigen-related cell adhesion molecule 6 (CEACAM6), also known as nonspecific crossreacting antigen (NCA) and CD66c, is one of seven human CEACAM family members within the immunoglobulin superfamily. It ...
TMPY-05151 CD39 Protein, Cynomolgus, Rhesus, Recombinant (His) Cynomolgus,Rhesus Baculovirus-Insect Cells
CD39, also known as ENTPD1, belongs to the GDA1/CD39 NTPase family. It is expressed primarily on activated lymphoid cells and can also be detected in endothelial tissues. The vascular isoform and the placental isoform II...
TMPY-01567 RBP4 Protein, Mouse, Recombinant (His) Mouse HEK293
Retinol-binding protein 4 (RBP4) is the specific carrier for retinol (also known as vitamin A), and is responsible for the conversion of unstable and insoluble retinol in aqueous solution into stable and soluble complex ...
TMPY-02808 CD39 Protein, Mouse, Recombinant (His) Mouse Baculovirus-Insect Cells
CD39, also known as ENTPD1, belongs to the GDA1/CD39 NTPase family. It is expressed primarily on activated lymphoid cells and can also be detected in endothelial tissues. The vascular isoform and the placental isoform II...
TMPY-00907 RBP4 Protein, Human, Recombinant (His) Human HEK293
Retinol-binding protein 4 (RBP4) is the specific carrier for retinol (also known as vitamin A), and is responsible for the conversion of unstable and insoluble retinol in aqueous solution into stable and soluble complex ...
TMPY-06935 FGF-21 Protein, Human, Recombinant Human E. coli
Fibroblast growth factor 21 (FGF21) is a member of the fibroblast growth factor (FGF) family. FGF family members possess broad mitogenic and cell survival activities and are involved in a variety of biological processes ...
TMPY-01007 VEGFC Protein, Human, Recombinant (His) Human HEK293
Vascular endothelial growth factor C (VEGF-C) is a member of the VEGF family. Upon biosynthesis, VEGF-C protein is secreted as a non-covalent momodimer in an anti-parellel fashion. VEGF-C protein is a dimeric glycoprotei...
TMPY-03156 VEGFC Protein, Mouse/Rat, Recombinant (aa 108-223, His) Mouse,Rat HEK293
Vascular endothelial growth factor C (VEGF-C) is a member of the VEGF family. Upon biosynthesis, VEGF-C protein is secreted as a non-covalent momodimer in an anti-parellel fashion. VEGF-C protein is a dimeric glycoprotei...
TMPY-01126 CD39 Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
CD39, also known as ENTPD1, belongs to the GDA1/CD39 NTPase family. It is expressed primarily on activated lymphoid cells and can also be detected in endothelial tissues. The vascular isoform and the placental isoform II...
TMPY-02938 REG4 Protein, Rat, Recombinant (His) Rat HEK293
Regenerating islet-derived protein 4, also known as REG-like protein, REG4, GISP and RELP, a member of the regenerating gene family belonging to the calcium (C-type) dependent lectin superfamily, has been found to be inv...
TMPY-02412 ENO1 Protein, Human, Recombinant (His) Human E. coli
The ENO1 gene encodes a multifunctional enzyme that has been identified as a key component of the glycolytic pathway. ENO1 overexpression and post-translational modifications could be of diagnostic and prognostic value ...
TMPY-00566 CCL18 Protein, Human, Recombinant (His) Human Yeast
CCL18 is a chemotactic cytokine involved in the pathogenesis and progression of various disorders, including cancer. Proof showed high levels of CCL18 in the serum of epithelial ovarian carcinoma patients suggesting its...
TMPY-01725 Leptin Receptor Protein, Human, Recombinant (His) Human HEK293
Leptin Receptor or CD295 belongs to the gp130 family of cytokine receptors that are known to stimulate gene transcription via activation of cytosolic STAT proteins. This protein is a receptor for leptin (an adipocyte-spe...
TMPY-01474 PAI-1 Protein, Human, Recombinant (His) Human HEK293
Plasminogen activator inhibitor 1, also known as PAI-1, Endothelial plasminogen activator inhibitor, SerpinE1 and PLANH1, is a secreted glycoprotein that belongs to the serpin family. SerpinE1 is the primary physiologica...
TMPH-00009 OGT Protein, Human, Recombinant (His & SUMO) Human E. coli
Catalyzes the transfer of a single N-acetylglucosamine from UDP-GlcNAc to a serine or threonine residue in cytoplasmic and nuclear proteins resulting in their modification with a beta-linked N-acetylglucosamine (O-GlcNAc...
TMPH-03473 UspA Protein, Salmonella typhi, Recombinant (His) Salmonella typhi E. coli
Required for resistance to DNA-damaging agents.
TMPH-02762 LPL Protein, Mouse, Recombinant Mouse E. coli
Involved in disease resistance and abiotic stress tolerance signaling pathways. Acts as a positive regulator of drought, salt and cold tolerance. Negatively modulates pathogenesis-related (PR) gene expression and broad-s...
TMPH-00678 Peptide deformylase Protein, E. coli O157:H7, Recombinant (His & SUMO) E. coli E. coli
TetR is the repressor of the tetracycline resistance element; its N-terminal region forms a helix-turn-helix structure and binds DNA. Binding of tetracycline to TetR reduces the repressor affinity for the tetracycline re...
TMPH-00691 IscS Protein, E. coli O6:K15:H31, Recombinant (His & Myc & SUMO) E. coli E. coli
Required for resistance to DNA-damaging agents.
TMPH-02133 DDX39B Protein, Human, Recombinant (GST) Human E. coli
Confers resistance to the different beta-lactams antibiotics (penicillin, cephalosporin and carbapenem) via the hydrolysis of the beta-lactam ring. Does not confer resistance to the polymixin colistin or the fluoroquinol...
TMPH-00711 BioH Protein, E. coli, Recombinant (His & Myc) E. coli E. coli
Involved in disease resistance.
TMPH-03029 MetAP Protein, Mycoplasma pneumoniae, Recombinant (His & SUMO) Mycoplasma pneumoniae E. coli
Prothymosin alpha may mediate immune function by conferring resistance to certain opportunistic infections.
TMPH-03135 Pla l 1 Protein, Plantago lanceolata, Recombinant (His & SUMO) Plantago lanceolata E. coli
Required for resistance to DNA-damaging agents.
TMPH-00677 OmpX Protein, E. coli O157:H7, Recombinant (His & Myc) E. coli E. coli
TetR is the repressor of the tetracycline resistance element; its N-terminal region forms a helix-turn-helix structure and binds DNA. Binding of tetracycline to TetR reduces the repressor affinity for the tetracycline re...
TMPH-03717 YopE Protein, Yersinia enterocolitica, Recombinant (His) Yersinia enterocolitica in vitro E. coli expression system
Essential virulence determinant; cytotoxic effector, involved in resistance to phagocytosis.
TMPH-01662 Merlin Protein, Human, Recombinant (His) Human E. coli
Parathymosin may mediate immune function by blocking the effect of prothymosin alpha which confers resistance to certain opportunistic infections.
TMPH-02131 SKP2 Protein, Human, Recombinant (His & SUMO) Human E. coli
SHV enzymes hydrolyze broad spectrum cephalosporins notably cefotaxime and ceftazidime. SHV-5 causes particularly high levels of resistance to aztreonam and ceftazidime.
TMPH-03175 Porin P Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPH-03519 ACP Protein, S. aureus, Recombinant (His) Staphylococcus aureus Yeast
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPH-03149 Porcine circovirus 2 (PCV2) Capsid Protein (E. coli, His) PCV2 E. coli
Confers resistance to the different beta-lactams antibiotics (penicillin, cephalosporin and carbapenem) via the hydrolysis of the beta-lactam ring.
TMPH-03518 ACP Protein, S. aureus, Recombinant (GST) Staphylococcus aureus E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPH-03177 RhlR Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO) Pseudomonas aeruginosa E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPH-03608 Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His) Streptomyces viridochromogenes Yeast
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance.
TMPH-02215 TCN1 Protein, Human, Recombinant (His) Human Yeast
Binds and compacts DNA (95 to 150 base pairs) to form nucleosome-like structures that contain positive DNA supercoils. Increases the resistance of DNA to thermal denaturation.
TMPH-00654 Methionine aminopeptidase Protein, E. coli, Recombinant (His & SUMO) E. coli E. coli
Not part of a putrescine export system. Very similar to a S.typhimurium protein implicated in antimicrobial peptide resistance, but the SapBCDF operon in E.coli is implicated in putrescine export.
TMPH-00539 Epstein-Barr virus (strain B95-8) BDLF3 Protein (His & Myc) EBV E. coli
TEM-type are the most prevalent beta-lactamases in enterobacteria; they hydrolyze the beta-lactam bond in susceptible beta-lactam antibiotics, thus conferring resistance to penicillins and cephalosporins. TEM-3 and TEM-4...
TMPH-00538 Epstein-Barr virus (strain GD1) EBNA3 Protein (His & Myc) EBV E. coli
Broad spectrum beta-lactamase which confers resistance to penicillins, as well as first, second and third-generation cephalosporins.
TMPH-03488 Metallo-beta-lactamase type 2 Protein, Serratia marcescens, Recombinant (His & Myc) Serratia marcescens E. coli
Confers resistance to the different beta-lactams antibiotics (penicillin, cephalosporin and carbapenem) via the hydrolysis of the beta-lactam ring.
TMPH-03571 WalK Protein, S. aureus, Recombinant (His & Myc) Staphylococcus aureus E. coli
Member of the two-component regulatory system WalK/WalR that regulates genes involved in cell wall metabolism, virulence regulation, biofilm production, oxidative stress resistance and antibiotic resistance via direct or...
TMPH-03176 LasA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPH-03520 ACP Protein, S. aureus, Recombinant (His & SUMO) Staphylococcus aureus E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPH-03604 Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His) Streptomyces hygroscopicus E. coli
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. Can also acetylate demethylphosphinothricin but not PTT or glutamate. This enzyme is an effector of phosphinothricin tripeptide (PTT or b...
TMPH-03260 Carboxypeptidase A1 Protein, Rat, Recombinant (His & Myc) Rat E. coli
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance.
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BAR Protein, S. hygroscopicus, Recombinant
TMPJ-00871
Species: Streptomyces hygroscopicus
Expression System: E. coli
Adiponectin Protein, Human, Recombinant (His)
TMPY-05556
Species: Human
Expression System: Baculovirus-Insect Cells
Adiponectin Protein, Human, Recombinant (hFc)
TMPY-02848
Species: Human
Expression System: HEK293
Insulin Receptor Protein, Human, Recombinant (long isoform, His)
TMPY-01146
Species: Human
Expression System: HEK293
TGFBI Protein, Human, Recombinant (His)
TMPY-01009
Species: Human
Expression System: HEK293
Neurotrophin 3 Protein, Human, Recombinant
TMPY-04069
Species: Human
Expression System: E. coli
CEACAM6 Protein, Human, Recombinant (His)
TMPY-00971
Species: Human
Expression System: HEK293
CEACAM6 Protein, Cynomolgus, Recombinant (His)
TMPY-05850
Species: Cynomolgus
Expression System: HEK293
CD39 Protein, Cynomolgus, Rhesus, Recombinant (His)
TMPY-05151
Species: Cynomolgus,Rhesus
Expression System: Baculovirus-Insect Cells
RBP4 Protein, Mouse, Recombinant (His)
TMPY-01567
Species: Mouse
Expression System: HEK293
CD39 Protein, Mouse, Recombinant (His)
TMPY-02808
Species: Mouse
Expression System: Baculovirus-Insect Cells
RBP4 Protein, Human, Recombinant (His)
TMPY-00907
Species: Human
Expression System: HEK293
FGF-21 Protein, Human, Recombinant
TMPY-06935
Species: Human
Expression System: E. coli
VEGFC Protein, Human, Recombinant (His)
TMPY-01007
Species: Human
Expression System: HEK293
VEGFC Protein, Mouse/Rat, Recombinant (aa 108-223, His)
TMPY-03156
Species: Mouse,Rat
Expression System: HEK293
CD39 Protein, Human, Recombinant (His)
TMPY-01126
Species: Human
Expression System: Baculovirus-Insect Cells
REG4 Protein, Rat, Recombinant (His)
TMPY-02938
Species: Rat
Expression System: HEK293
ENO1 Protein, Human, Recombinant (His)
TMPY-02412
Species: Human
Expression System: E. coli
CCL18 Protein, Human, Recombinant (His)
TMPY-00566
Species: Human
Expression System: Yeast
Leptin Receptor Protein, Human, Recombinant (His)
TMPY-01725
Species: Human
Expression System: HEK293
PAI-1 Protein, Human, Recombinant (His)
TMPY-01474
Species: Human
Expression System: HEK293
OGT Protein, Human, Recombinant (His & SUMO)
TMPH-00009
Species: Human
Expression System: E. coli
UspA Protein, Salmonella typhi, Recombinant (His)
TMPH-03473
Species: Salmonella typhi
Expression System: E. coli
LPL Protein, Mouse, Recombinant
TMPH-02762
Species: Mouse
Expression System: E. coli
Peptide deformylase Protein, E. coli O157:H7, Recombinant (His & SUMO)
TMPH-00678
Species: E. coli
Expression System: E. coli
IscS Protein, E. coli O6:K15:H31, Recombinant (His & Myc & SUMO)
TMPH-00691
Species: E. coli
Expression System: E. coli
DDX39B Protein, Human, Recombinant (GST)
TMPH-02133
Species: Human
Expression System: E. coli
BioH Protein, E. coli, Recombinant (His & Myc)
TMPH-00711
Species: E. coli
Expression System: E. coli
MetAP Protein, Mycoplasma pneumoniae, Recombinant (His & SUMO)
TMPH-03029
Species: Mycoplasma pneumoniae
Expression System: E. coli
Pla l 1 Protein, Plantago lanceolata, Recombinant (His & SUMO)
TMPH-03135
Species: Plantago lanceolata
Expression System: E. coli
OmpX Protein, E. coli O157:H7, Recombinant (His & Myc)
TMPH-00677
Species: E. coli
Expression System: E. coli
YopE Protein, Yersinia enterocolitica, Recombinant (His)
TMPH-03717
Species: Yersinia enterocolitica
Expression System: in vitro E. coli expression system
Merlin Protein, Human, Recombinant (His)
TMPH-01662
Species: Human
Expression System: E. coli
SKP2 Protein, Human, Recombinant (His & SUMO)
TMPH-02131
Species: Human
Expression System: E. coli
Porin P Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03175
Species: Pseudomonas aeruginosa
Expression System: E. coli
ACP Protein, S. aureus, Recombinant (His)
TMPH-03519
Species: Staphylococcus aureus
Expression System: Yeast
Porcine circovirus 2 (PCV2) Capsid Protein (E. coli, His)
TMPH-03149
Species: PCV2
Expression System: E. coli
ACP Protein, S. aureus, Recombinant (GST)
TMPH-03518
Species: Staphylococcus aureus
Expression System: E. coli
RhlR Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO)
TMPH-03177
Species: Pseudomonas aeruginosa
Expression System: E. coli
Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His)
TMPH-03608
Species: Streptomyces viridochromogenes
Expression System: Yeast
TCN1 Protein, Human, Recombinant (His)
TMPH-02215
Species: Human
Expression System: Yeast
Methionine aminopeptidase Protein, E. coli, Recombinant (His & SUMO)
TMPH-00654
Species: E. coli
Expression System: E. coli
Epstein-Barr virus (strain B95-8) BDLF3 Protein (His & Myc)
TMPH-00539
Species: EBV
Expression System: E. coli
Epstein-Barr virus (strain GD1) EBNA3 Protein (His & Myc)
TMPH-00538
Species: EBV
Expression System: E. coli
Metallo-beta-lactamase type 2 Protein, Serratia marcescens, Recombinant (His & Myc)
TMPH-03488
Species: Serratia marcescens
Expression System: E. coli
WalK Protein, S. aureus, Recombinant (His & Myc)
TMPH-03571
Species: Staphylococcus aureus
Expression System: E. coli
LasA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03176
Species: Pseudomonas aeruginosa
Expression System: E. coli
ACP Protein, S. aureus, Recombinant (His & SUMO)
TMPH-03520
Species: Staphylococcus aureus
Expression System: E. coli
Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His)
TMPH-03604
Species: Streptomyces hygroscopicus
Expression System: E. coli
Carboxypeptidase A1 Protein, Rat, Recombinant (His & Myc)
TMPH-03260
Species: Rat
Expression System: E. coli
Cat No. Product Name
L2190 Anti-Lung Cancer Compound Library

1735 compounds
A unique collection of 1735 compounds with anti-lung cancer therapeutic activity or targeting lung cancer’s major signaling pathways, can be used for anti-lung cancer drug discovery and mechanism study;
L4510 Anti-Parasitic Compound Library

420 compounds
420 well-chosen unique anti-parasitic small molecules;
L4520 Anti-Bacterial Compound Library

921 compounds
A unique collection of 921 antibacterial bioactive compounds, a powerful tool for antibacterial drug development;
L3900 DNA Damage & Repair Compound Library

937 compounds
A unique collection of 937 DNA Damage & Repair related compounds for high throughput screening (HTS) and high content screening (HCS);
L4400 Antibiotics Library

708 compounds
A unique collection of 708 compounds with antibiotic activity for new antibacterial drug screening;
L3980 DNA Damage and Repair Compound Library Plus

667 compounds
Well-chosen 667 compounds with unique structures targeting DNA damage & repair;
L7110 Anti-Hypertension Compound Library

719 compounds
719 hypertension-related small molecules for high-throughput and high-content screening.
L6730 Anti-virus Traditional Chinese Medicine Monomer Library

270 compounds
A collection of 270 TCM monomers with anti-virus activity. An effective tool for drug development and pharmacological studies.
L9300 Macrocyclic Compound Library

216 compounds
216 macrocyclic compounds of known activity for high-throughput, high-content screening;
L6610 Anti-infective Natural Product Library

1070 compounds
A unique collection of 1070 species of natural products with anti-infective activity for high throughput screening (HTS) and high content screening (HCS);
L2140 Cancer Cell Differentiation Compound Library

413 compounds
A unique collection of 413 cancer cell differentiation inducing compounds for high throughput and high content screening;
L2130 Anti-Cancer Metabolism Compound Library

1280 compounds
A unique collection of 1280 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS);
L9700 Endoplasmic Reticulum Stress Compound Library

193 compounds
A unique collection of 193 endoplasmic reticulum stress (ER stress) related compounds used for high throughput screening (HTS) and high content screening (HCS);
L2540 Gut Microbial Metabolite Library

614 compounds
A unique collection of 614 gut microbial metabolites which can be used for HTS and HCS;
L9410 Covalent Inhibitor Library

1949 compounds
A unique collection of 1949 covalent Inhibitors and other molecules with common warheads like chloroacetyl,2-Chloropropionyl,Acryloyl,sulfonyl fluoride, alkyne,acrylamide, ketocarbonyl,disulfide bond, etc.
TargetMol