Search Result

Search Results for " 泛素化 "

Targets

138

Compounds

Natural Products

Libraries

Cat No.	Product Name	Synonyms	Targets
T9884	EN523		Others
	EN523 targets non-catalytic allosteric cysteine C23 in K48 ubiquitin-specific deuquitinase OTUB1.		Others
T12579	RAMB4	PTP1B-IN-9	Proteasome
	RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.		Proteasome
T16974	TAK-243	MLN7243	Apoptosis , E1/E2/E3 Enzyme , NF-κB
	TAK-243 (MLN7243) is a selective inhibitor of the ubiquitin-activating enzyme UAE (IC50=1 nM). TAK-243 blocks ubiquitin binding and disrupts mono-ubiquitin signaling as well as overall protein ubiquitination. TAK-243 exh...		Apoptosis , E1/E2/E3 Enzyme , NF-κB
T22922	Lenalidomide hemihydrate		TNF , Ligand for E3 Ligase , Molecular Glues
	Lenalidomide hemihydrate is a TNF-α secretion inhibitor (IC50 = 13 nM). Lenalidomide hemihydrate could bound endogenous CRBN and recombinant CRBN-DNA damage binding protein-1 (DDB1) complexes.		TNF , Ligand for E3 Ligase , Molecular Glues
T1642	Lenalidomide	CC-5013	Apoptosis , TNF , Ligand for E3 Ligase , Molecular Glues
	Lenalidomide (CC-5013) is a potent inhibitor of TNF-α that, at 10 μM, alters gene expression and cell viability in a range of cancer cell lines.		Apoptosis , TNF , Ligand for E3 Ligase , Molecular Glues
T1932	B-AP15	NSC 687852	Apoptosis , DUB
	B-AP15 (NSC-687852)(NSC-687852) is a selective inhibitor of the deubiquitinating enzymes Usp14 and UCHL5 of the 26S proteasome. It blocks the deubiquitinating activity of the 26S proteasome.		Apoptosis , DUB
T3110	PRT4165	NSC600157,PRT 4165	BMI-1 , Others , E1/E2/E3 Enzyme
	PRT4165 (NSC600157) is a potent PRC1-mediated H2A ubiquitylation inhibitor.		BMI-1 , Others , E1/E2/E3 Enzyme
T16904	Smurf1-IN-A01	A01	Others
	Smurf1-IN-A01 (A01) is a ubiquitin ligase Smad ubiquitination regulatory factor-1 inhibitor (kd: 3.664 nM). It increases BMP-2 responsiveness by inhibiting Smurf1-mediated Smad1/5 degradation.		Others
T25465	GS143	GS-143,GS 143	IκB/IKK , E1/E2/E3 Enzyme , NF-κB
	GS143 is a selective IκBα ubiquitination inhibitor with an IC50 of 5.2 μM for SCFβTrCP1-mediated IκBα ubiquitylation. GS143 suppresses NF-κB activation and transcription of target genes and does not inhibit protea...		IκB/IKK , E1/E2/E3 Enzyme , NF-κB
T6697	TCID	UCH-L3 Inhibitor	DUB
	TCID (UCH-L3 Inhibitor)(IC50=0.6 μM) is a DUB inhibitor of ubiquitin C-terminal hydrolase L3. It has the 125-fold selectivity to L1.		DUB
T17879	E3 ligase Ligand 8		Others , Ligand for E3 Ligase
	E3 ligase Ligand 8 is a ligand for E3 ubiquitin ligase. The E3 ligase Ligand 8 can be linked to protein ligands through linkers to form PROTACs, which are inducers of ubiquitination-mediated degradation of cancer-promoti...		Others , Ligand for E3 Ligase
T21773	SP-141	SP 141	Mdm2
	SP 141 is a MDM2 inhibitor.SP-141 promotes MDM2 auto-ubiquitination and degradation, with anticancer activity.		Mdm2
T12024	MF-094		DUB
	MF-094 is a potent and selective inhibitor of USP30 (IC50 of 120 nM).		DUB
T21527	HBX 41108	HBX-41108	DUB , p53
	HBX 41108 (HBX-41108) is a non-competitive, reversible inhibitor of USP7 with an IC50 of 424nM. HBX 41108 inhibited deubiquitination of p53 mediated by USP7 in a dose-dependent manner with an IC50 of 0.8μM.		DUB , p53
T6629	PYR-41	PYR41,PYR 41	Apoptosis , E1/E2/E3 Enzyme
	PYR-41 is the first cell-permeable inhibitor of ubiquitin-activating enzyme E1, with no activity at E2.		Apoptosis , E1/E2/E3 Enzyme
T1919	Tenovin-1	Tenovin 1	Mdm2 , Dehydrogenase , Sirtuin , p53 , Autophagy
	Tenovin-1 inhibits protein-deacetylating activities of SirT1 and SirT2 and protects against MDM2-mediated p53 degradation, which involves ubiquitination.		Mdm2 , Dehydrogenase , Sirtuin , p53 , Autophagy
T1757	ML-323	ML323	DUB
	ML323 is a reversible and effective USP1-UAF1 inhibitor in a Ub-Rho assay (IC50: 76 nM) and in orthogonal gel-based assays using K63-linked diubiquitin (di-Ub) (IC50: 174 nM 820 nM)and monoubiquitinated PCNA (Ub-PCNA) (I...		DUB
T27240	Eeyarestatin I		Apoptosis
	Eeyarestatin I is an inhibitor that inhibits the degradation and translocation of ER-associated proteins. Eeyarestatin I is associated with the p97 deubiquitination process and inhibits atx3 deubiquitination. Eeyarestati...		Apoptosis
T6910	NSC59984		p53
	NSC59984, a p53 pathway activator, induces mutant p53 protein degradation and p73 activation.		p53
T3088	N-Ethylmaleimide	1-Ethyl-1H-pyrrole-2,5-dione,Ethylmaleimide,NEM	Cysteine Protease , DUB
	N-Ethylmaleimide (NEM) is a sulfhydryl reagent that is widely used in experimental biochemical studies.		Cysteine Protease , DUB
T5199	COH000		E1/E2/E3 Enzyme
	COH000 is a covalent and irreversible inhibitor of small ubiquitin-like modifier (SUMO)-activating enzyme and inhibited SUMOylation (IC50: ~ 0.2 μM in vitro).		E1/E2/E3 Enzyme
T13349	WS-383		E1/E2/E3 Enzyme
	WS-383 is a selective, potent and reversible DCN1-UBC12 interaction inhibitor(IC50 of 11 nM).		E1/E2/E3 Enzyme
TP1186	Cyclo(Phe-Pro)	A-64863,Cyclo(phenylalanylprolyl)	Others
	Cyclo(Phe-Pro) (A-64863) known as a secondary metabolite of some bacteria and fungi, is also produced by Vibrio vulnificus.		Others
T11209	EOAI3402143		DUB
	EOAI3402143 inhibits Usp9x and Usp24 activity, increases tumor cell apoptosis. EOAI3402143 phenocopies the FAS induction and apoptotic sensitization of Usp5 knockdown and fully blocks melanoma tumor growth.		DUB
T60130	USP5-IN-1		DUB
	USP5-IN-1 (compound 64) is a potent deubiquitinase USP5 inhibitor, which binds to the USP5 ZnF-UBD with a KD of 2.8 μM and is selective over nine proteins containing structurally similar ZnF-UBD domains. USP5-IN-1 inhibi...		DUB
T11485	GSK2643943A		DUB
	GSK2643943A is a deubiquitylating enzyme (DUB) inhibitor, with an IC 50 of 160 nM for USP20/Ub-Rho. GSK2643943A has anti-tumor efficacy.		DUB
T13244	Ubiquitination-IN-1		Others
	Ubiquitination-IN-1 is an inhibitor of ubiquitination and Cksl-Skp2 protein-protein interaction (IC50: 0.17 μM).		Others
T22263	Bavdegalutamide	ARV-110	Androgen Receptor
	Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR). Bavdegalutamide can be used in studies about prostate cancer. Bavdegalutamide shows oral activity and selectivity and facilitates the ubiquitinati...		Androgen Receptor
T1372	2-Methoxybenzylamine		Others
	2-Methoxybenzylamine is widely used in the synthesis of other compounds such as dyes, fragrances and plastics; it can also be used in the synthesis of bioactive compounds such as antibiotics and antifungals.		Others
T0922	Zoxazolamine	NSC 24995,Contrazole	Others
	Zoxazolamine (NSC-24995) is a uricosuric and muscle relaxant. Zoxazolamine acts centrally as a muscle relaxant, but the mechanism of its action is not understood.		Others
T36682	USP30 inhibitor 18		DUB
	USP30 inhibitor 18 is a selective USP30 inhibitor with an IC50 of 0.02 μM. USP30 inhibitor 18 increases protein ubiquitination and accelerates mitophagy[1]. [1]. Arthur F Kluge, et al. Novel highly selective inhibitors o...		DUB
T61477	DCeMM2		Molecular Glues
	dCeMM2 is a glue degrader. dCeMM2 prompts an interaction of CDK12-cyclin K with a CRL4B ligase complex, leading to the ubiquitination and degradation of cyclin K.		Molecular Glues
T6743	(E/Z)-4-Hydroxytamoxifen	Afimoxifene,4-Hydroxytamoxifen	Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeutic and chemopreventive treatment of breast cancer.		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T67876	USP8-IN-2		DUB
	USP8-IN-2 is a potent inhibitor of the deubiquitinating enzymes USP7 and USP8, with an IC50 of 4.0 μM against USP8D. USP8-IN-2 is a potential compound for the treatment of cancer and viral infections.		DUB
T8951	JTP 0819958 - HOIPIN-1		IκB/IKK
	JTP-0819958 is a selective linear ubiquitin chain assembly complex (LUBAC) inhibitor with an IC50 of 2.8 μM[1]. JTP-0819958 suppress LUBAC-mediated NF-kB activation in vitro[2].		IκB/IKK
T73560	I-138		DUB
	I-138 is an orally active and potent reversible inhibitor of USP1-UAF1.I-138 induces mono-ubiquitination of FANCD2 and PCNA and inhibits USP1 auto-cleavage in cells.		DUB
T10765	Eragidomide	CC-90009,Cereblon modulator 1	Apoptosis , Ligand for E3 Ligase , Molecular Glues
	Eragidomide (CC-90009; Cereblon modulator 1) is a cereblon (CRBN) E3 ligase modulator. Eragidomide specifically binds to CRBN, thereby affecting the activity of the ubiquitin E3 ligase complex.		Apoptosis , Ligand for E3 Ligase , Molecular Glues
T6300	Degrasyn	WP1130	Apoptosis , JAK , Bcr-Abl , DUB , Autophagy
	Degrasyn (WP1130) (WP1130), a specific deubiquitinase (DUB: USP5, UCH-L1, USP9x, USP14, and UCH37) inhibitor, also inhibits Bcr/Abl, which is a JAK2 transducer (without affecting 20S proteasome) and activator of transcri...		Apoptosis , JAK , Bcr-Abl , DUB , Autophagy
T37042	SCH529074	SCH 529074	p53
	SCH529074 is a selective activator of p53 (Ki = 1 μM) and can be used in studies about non-small-cell lung carcinoma. SCH529074 restores mutant p53 function and interrupts HDM2-mediated ubiquitination of wild Type p53.		p53
T8773	MID-1		Others , IGF-1R
	MID-1 is an inhibitor of MG53-IRS-1 (Mitsugumin 53-Insulin Receptor Substrate-1) interaction. It disrupts molecular association of MG53 with IRS-1 and abolishes MG53-induced IRS-1 ubiquitination and degradation in skelet...		Others , IGF-1R
T0424	Bismuth Subsalicylate	Bismuth subsalicylat,Bismuth(III) salicylate basic,Bismuth oxysalicylate	COX , PGE Synthase
	Bismuth Subsalicylate (Bismuth subsalicylat) is the active ingredient in the popular medication Pepto-Bismol that is used to treat nausea, heartburn, indigestion, upset stomach, diarrhea, and other temporary discomforts ...		COX , PGE Synthase
T64339	Apcin A HCL		APC
	Apcin A HCL is an Apcin derivative. Apcin A HCL is an anaphase-promoting complex (APC) inhibitor. Apcin-A HCL interacts strongly with Cdc20, and inhibits the ubiquitination of Cdc20 substrates. Apcin-A HCL can be used to...		APC
T1902	BAY 11-7082	BAY 11-7821	Apoptosis , Others , IκB/IKK , DUB , Autophagy
	BAY 11-7082 (BAY 11-7821) is an NF-κB inhibitor that inhibits TNFα-induced IκBα phosphorylation (IC50=10 μM). BAY 11-7082 is also an inhibitor of the ubiquitin-specific proteases USP7 and USP21 (IC50=0.19/0.96 μM).		Apoptosis , Others , IκB/IKK , DUB , Autophagy
T63790	Cbl-b-IN-3		E1/E2/E3 Enzyme
	Cbl-b-IN-3 is a potent proto-oncogene-B (CPL-B) inhibitor of casitas B-series lymphoma (ic50 < 1 nM). Cpl-b, a cyclic E3 ubiquitin protein ligase, is involved in the setting of T lymphocyte activation thresholds. Cpl-b n...		E1/E2/E3 Enzyme
T5461	GNE-6640		DUB
	GNE-6640 is a non-covalent inhibitor targeting ubiquitin specific peptidase 7 (USP7), exhibiting IC50 values of 0.75 μM for full-length USP7, 0.43 μM for the USP7 catalytic domain, 20.3 μM for full-length USP43, and 0.23...		DUB
T17187	TZ9		Apoptosis , E1/E2/E3 Enzyme
	TZ9 is a selective and potent Rad6 inhibitor with anticancer and anti-tumor activity.TZ9 inhibits Rad6B-induced ubiquitination of histone H2A.TZ9 induces cell cycle arrest and apoptosis.		Apoptosis , E1/E2/E3 Enzyme
T8488	GMB-475		Bcr-Abl
	GMB-475 is a BCR-ABL1 tyrosine kinase degrader based on PROTAC, overcoming BCR-ABL1-dependent drug resistance. GMB-475 targets BCR-ABL1 protein and recruits the E3 ligase Von Hippel Lindau (VHL).resulting in ubiquitinati...		Bcr-Abl
T15069	DBCO-PEG4-Biotin	ADIBO-NH-PEG2-Biotin	Others
	DBCO-PEG4-Biotin (ADIBO-NH-PEG2-Biotin) is an azadibenzocyclooctyne-biotin derivative containing a biotin moiety and 4 PEGs.DBCO-PEG4-Biotin is a versatile biotinylation reagent that introduces a portion of biotin into ...		Others
T66491	4-(1-Phenylethyl)resorcinol	4-(1-Phenylethyl)benzene-1,3-diol,Phenylethyl resorcinol	Others
	4-(1-Phenylethyl)resorcinol (4-(1-Phenylethyl)benzene-1,3-diol) is a skin brightening agent that is a cosmetic additive. It works by inhibiting melanin production, reducing the appearance of dark spots, hyperpigmentation...		Others
T67873	USP8-IN-3		DUB
	USP8-IN-3 is a potent inhibitor of the deubiquitinating enzymes USP7 and USP8, with IC50 of 4.0 μM against USP8D. USP8-IN-3 inhibited the proliferation of GH3 and H1957 cells with GI50 values of 37.03 μM and 6.01 μM, res...		DUB

Compounds

Target: Apoptosis, E1/E2/E3 Enzyme, NF-κB

Lenalidomide hemihydrate

T22922

Synonym:

Target: TNF, Ligand for E3 Ligase, Molecular Glues

Lenalidomide

T1642

Synonym: CC-5013

Target: Apoptosis, TNF, Ligand for E3 Ligase, Molecular Glues

B-AP15

T1932

Synonym: NSC 687852

Target: Apoptosis, DUB

PRT4165

T3110

Synonym: NSC600157,PRT 4165

Target: BMI-1, Others, E1/E2/E3 Enzyme

Synonym: GS-143,GS 143

Target: IκB/IKK, E1/E2/E3 Enzyme, NF-κB

TCID

T6697

Synonym: UCH-L3 Inhibitor

Target: Others, Ligand for E3 Ligase

Synonym: PYR41,PYR 41

Target: Apoptosis, E1/E2/E3 Enzyme

Tenovin-1

T1919

Synonym: Tenovin 1

Target: Mdm2, Dehydrogenase, Sirtuin, p53, Autophagy

Synonym: 1-Ethyl-1H-pyrrole-2,5-dione,Ethylmaleimide,NEM

Target: Cysteine Protease, DUB

COH000

T5199

Synonym:

Target: E1/E2/E3 Enzyme

WS-383

T13349

Synonym:

Target: E1/E2/E3 Enzyme

Cyclo(Phe-Pro)

TP1186

Synonym: A-64863,Cyclo(phenylalanylprolyl)

Target: Androgen Receptor

Synonym: NSC 24995,Contrazole

Target: Molecular Glues

(E/Z)-4-Hydroxytamoxifen

T6743

Synonym: Afimoxifene,4-Hydroxytamoxifen

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor

JTP 0819958 - HOIPIN-1

Synonym: CC-90009,Cereblon modulator 1

Target: Apoptosis, Ligand for E3 Ligase, Molecular Glues

Degrasyn

T6300

Synonym: WP1130

Target: Apoptosis, JAK, Bcr-Abl, DUB, Autophagy

Target: Others, IGF-1R

Bismuth Subsalicylate

T0424

Synonym: Bismuth subsalicylat,Bismuth(III) salicylate basic,Bismuth oxysalicylate

Target: COX, PGE Synthase

Target: Apoptosis, Others, IκB/IKK, DUB, Autophagy

Cbl-b-IN-3

T63790

Synonym:

Target: E1/E2/E3 Enzyme

Target: Apoptosis, E1/E2/E3 Enzyme

Synonym: ADIBO-NH-PEG2-Biotin

Target: Others

4-(1-Phenylethyl)resorcinol

T66491

Synonym: 4-(1-Phenylethyl)benzene-1,3-diol,Phenylethyl resorcinol

Cat No.	Product Name	Synonyms	Targets
T1059	Retinyl palmitate	Retinol palmitate,Vitamin A palmitate,Retinyl (Vitamin A) Palmitate	Others , Endogenous Metabolite
	Retinyl palmitate (Vitamin A palmitate) is a naturally-occurring phenyl analogue of retinol, with potential antineoplastic and chemopreventive activities.		Others , Endogenous Metabolite
T8201	Gambogenic acid		Histone Methyltransferase
	Gambogenic acid is a natural product,is an effective inhibitor of EZH2,with anticancer activity.		Histone Methyltransferase
T1558	Resveratrol	trans-Resveratrol,SRT 501	Apoptosis , Mitophagy , IκB/IKK , Lipoxygenase , Sirtuin , COX , NADPH , DNA/RNA Synthesis , Nrf2 , Antibacterial , Antibiotic , Autophagy , Antifungal
	Resveratrol (SRT 501) is a polyphenolic natural product, a plant antitoxin with antioxidant and chemopreventive activities. Resveratrol has a wide range of targets including COX, SIRT, LOC, etc. Resveratrol induces autop...
T3S0137	Bavachalcone		Antibacterial , Antibiotic
	Bavachalcone is a major bioactive compounds isolated from Psoralea corylifolia L. it may be useful as a therapeutic drug for bone resorption-associated diseases.Bavachalcone can protect the endothelial function by increa...		Antibacterial , Antibiotic
T4970	LANOSTEROL	3β-Hydroxy-8,24-lanostadiene,8,24-Lanostadien-3β-ol	Endogenous Metabolite
	Lanosterol (3β-Hydroxy-8,24-lanostadiene) is a tetracyclic triterpenoid which is the compound from which all steroids are derived.		Endogenous Metabolite
T22417	Rutin hydrate	Rutoside,Sophorin,Quercetin-3-O-rutinoside	Beta Amyloid , Others , Autophagy
	Rutin hydrate (Sophorin), a kind of glycoside, widely exists in many plants including citrus fruit.		Beta Amyloid , Others , Autophagy
T5813	BYAKANGELICIN		Reductase
	BYAKANGELICIN,a main furanocoumarin constituent isolated and characterized as an aldose reductase inhibitor,and is effective for the treatment of sugar cataracts and diabetic neuropathy and hence might be useful as a lea...		Reductase
T6S1780	Protosappanin B	Q-100961,FT-0689654	Apoptosis
	1. Protosappanin B (Q-100961) significantly increases cell viability, inhibits cell apoptosis and up-regulates the expression of growth-associated protein 43. 2. Protosappanin B induces the degradation of p53 protein, vi...		Apoptosis
T3254	PHYTOL	trans-Phytol,(E)-Phytol	Antibacterial , PPAR , Parasite
	PHYTOL (trans-Phytol) , a diterpene alcohol from chlorophyll widely used as a food additive and in medicinal fields, shows antinociceptive and antioxidant activities as well as anti-inflammatory and antiallergic effects....		Antibacterial , PPAR , Parasite
T65269	L-Aspartic acid potasium salt	Aspartic acid potasium salt,Potassium L-aspartate	Others
	L-aspartic acid potasium salt（VX-548） is an amino acid widely found in plants and animals.L-aspartic acid potasium salt drives the production of nitrogen oxides, which promotes phagocytosis and contributes to fish surviv...		Others
T78486	Cis-Nerolidol
	cis-Nerolidol, a sesquiterpene alcohol present in numerous plants, exhibits antioxidant and antibacterial properties. Additionally, it can potentiate the effects of antibiotics [1].
T75743	HA Peptide TFA
	HA Peptide (TFA), a nine amino acid sequence derived from human influenza hemagglutinin (HA), is widely employed in cell biology and biochemistry for the isolation, purification, detection, and tracking of target protein...
T83437	18-O-Demethylpederin
	18-O-Demethylpederin, a pederin analogue, is a natural polyketide first isolated from Paederus. This compound is a non-protein insect toxin and exhibits a range of biological activities, such as antibacterial, antiviral,...
T79941	Antimycin A2c		Apoptosis
	Anticancer Agent 141 (Compound AE), an antimycin alkaloid, exhibits inhibitory potential against HPV-infected cervical cancer. It impedes HeLa cell proliferation by arresting the cell cycle at the S phase and induces cas...		Apoptosis
T78506	α-Lactose hydrate	α-D-Lactose hydrate
	α-Lactose (hydrate) (α-D-Lactose (hydrate)), the main carbohydrate in mammalian milk, comprises two sugar units: glucose and galactose, and occurs as two anomers, α and β. It serves multiple roles in the food and pharmac...

Natural Products

Retinyl palmitate

T1059

Synonym: Retinol palmitate,Vitamin A palmitate,Retinyl (Vitamin A) Palmitate

Target: Others, Endogenous Metabolite

Gambogenic acid

T8201

Synonym:

Target: Histone Methyltransferase

Resveratrol

T1558

Synonym: trans-Resveratrol,SRT 501

Target: Apoptosis, Mitophagy, IκB/IKK, Lipoxygenase, Sirtuin, COX, NADPH, DNA/RNA Synthesis, Nrf2, Antibacterial, Antibiotic, Autophagy, Antifungal

Bavachalcone

T3S0137

Synonym:

Target: Antibacterial, Antibiotic

LANOSTEROL

T4970

Synonym: 3β-Hydroxy-8,24-lanostadiene,8,24-Lanostadien-3β-ol

Target: Endogenous Metabolite

Rutin hydrate

T22417

Synonym: Rutoside,Sophorin,Quercetin-3-O-rutinoside

Target: Beta Amyloid, Others, Autophagy

Synonym: Q-100961,FT-0689654

Target: Apoptosis

PHYTOL

T3254

Synonym: trans-Phytol,(E)-Phytol

Target: Antibacterial, PPAR, Parasite

L-Aspartic acid potasium salt

T65269

Synonym: Aspartic acid potasium salt,Potassium L-aspartate

Synonym: α-D-Lactose hydrate

Target:

Cat No.	Product Name
L8600	Ubiquitination Compound Library	214 compounds
	A unique collection of 214 ubiquitination related small chemicals can be used for high throughput and high content screening；
L9820	Beta-Lactam Compound Library	105 compounds
	A unique collection of 105 beta-lactam compounds, can be used in HTS and HCS;
L3300	Histamine & Melatonin Receptor-Targeted Compound Library	155 compounds
	A unique collection of 155 compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS) for new drugs;
L7300	Potassium Channel Blocker Library	160 compounds
	A unique collection of 160 potassium channel blockers and agonists for high throughput and high content screening;
L6140	Saccharide and Glycoside Natural Product Library	364 compounds
	A unique collection of 364 saccharides and glycosides compounds can be used for HTS and HCS；
L4710	Nonsteroidal Anti-Inflammatory Compound Library	530 compounds
	530 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening.
L8200	Anti-Aging Compound Library	3324 compounds
	A unique collection of 3324 anti-aging compounds for high throughput screening (HTS) and high content screening (HCS);
L4020	NO PAINS Compound Library	9555 compounds
	TargetMol created the L4020 NO-PAINS Compound Library that applied the PAINS filter, remaining 9555 small molecules that are suitable for new drug development, signaling pathway research, drug repurposing and other resea...
L3500	Histone Modification Compound Library	480 compounds
	A unique collection of 480 histone modification related compounds for high throughput screening (HTS) and high content screening (HCS);
L6750	PBCRBS Traditional Chinese Medicine Compound Library	588 compounds
	A unique collection of 588 compounds derived from traditional Chinese medicines (TCMs) for promoting blood circulation and removing blood stasis.
L2800	Serotonin Receptor-Targeted Compound Library	275 compounds
	A unique collection of 275 compounds targeting serotonin receptors for high throughput screening and high content screening;
L8300	Chromatin Modification Compound Library	256 compounds
	A unique collection of 256 compounds targeting chromatin remodeling pathway for high throughput screening (HTS) and high content screening (HCS);
L9300	Macrocyclic Compound Library	216 compounds
	216 macrocyclic compounds of known activity for high-throughput, high-content screening;
DO1200	SmartTM Library	53200 compounds

L1300	PI3K-AKT-mTOR Compound Library	425 compounds
	A unique collection of 425 compounds targeting PI3K/Akt/mTOR signaling for research in PI3K/Akt/mTOR signaling, and drug discovery in diseases involved with PI3K/Akt/mTOR signaling;
L6110	Alkaloid Natural Product Library	468 compounds
	A unique collection of 468 natural alkaloids can be used for high throughput and high content screening；
L7200	Calcium Channel Compound Library	143 compounds
	A unique collection of 143 calcium channel blockers and agonists for high throughput and high content screening;
L9600	Peptide Compound Library	800 compounds
	800 peptides can be used in peptide drug development and signaling transduction and mechanism study;
L5510	Drug-induced Liver Injury (DILI) Compound Library	1040 compounds
	A unique collection of 1040 hepatotoxicity causing compounds, a powerful tool for drug toxicity study, can be used for HTS and HCS screening；
L6820	Tobacco Monomer Library	750 compounds
	A unique collection of 750 tobacco monomer compounds for high throughput screening and high content screening;