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Search Results for " 离子通道 "

Targets

184

Compounds

31

Natural Products

6

Libraries

Cat No. Product Name Synonyms Targets
T10674 Potassium Channel Activator 1 ZINC34634569 Potassium Channel
Potassium Channel Activator 1 can be used in studies about the treatment of disorders or conditions wherein the dopaminergic system is disrupted such as mood disorders ADHD, schizophrenia, and other psychotic states.
T10101 Calcium channel-modulator-1 Others , Calcium Channel
Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.
T2604 1-EBIO 1-EBIO Calcium Channel
1-EBIO (1-EBIO) is a calium channel agonist.
T4669 Fantofarone SR 33557 Calcium Channel , Parasite
Fantofarone (SR 33557) is a highly potent antagonist of Calcium Channel.
T10852 CNS-5161 hydrochloride CNS 5161A NMDAR
CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel. It interacts with the NMDA receptor/ion channel site to produce a noncompetitive blockade of the actions of glutamate.
T10566 BMS-191095 Potassium Channel
BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.
T22537 9-Phenanthrol TRP/TRPV Channel
9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.
T10307 AMPA receptor modulator-1 iGluR
AMPA receptor modulator-1 can be activated by glutamate, thereby modulating ion channels.
T22353 Lanthanum(III) chloride heptahydrate Calcium Channel
Lanthanum(III) chloride is an inorganic compound which used in biochemical research to block the activity of divalent cation channels, especially calcium channels.
T7182 Metaflumizone BAS-320I Sodium Channel , Parasite
Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.
T1422 Nilvadipine FK235,FR34235,ARC029 Calcium Channel
Nilvadipine (FK235), a calcium channel blocker (CCB), is utilized for treatment of hypertension.
T2342 Raxatrigine CNV1014802,CNV 1014802,GSK-1014802,CNV-1014802 Sodium Channel
Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.
T64561 DPhPC Others
DPhPC is a synthetic liposome used to synthesize liposomes commonly used in artificial membrane matrices.DPhPC bilayers do not allow ion leakage in the absence of pore/ion channels.DPhPC can be used to study channel prot...
T0231 Amlodipine Besylate Amlodipine benzenesulfonate Calcium Channel
Amlodipine Besylate(Amlodipine benzenesulfonate) is a long-lasting calcium channel blocker.
T12608 QX-314 chloride Sodium Channel
QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.
T15053 Darodipine PY-108068,PY 108-068 Calcium Channel
Darodipine (PY-108068) is a dihydropyridine type Ca+2 antagonist.
T15233 Endovion NS3728 Chloride channel
Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.
T16346 NS1652 Chloride channel
NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.
T5183 AUT1 Potassium Channel
AUT1 (AUT-1) is a novel specific modulator of Kv3 channels (EC50: 4.7 and 4.9 uM for Kv3.1b and Kv3.2a).
T16110 ML418 Potassium Channel
ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.
T0121 Azelnidipine CS 905,UR-12592 Calcium Channel
Azelnidipine (UR-12592) is a dihydropyridine used as calcium channel blocker.
T0193 Manidipine dihydrochloride Manidipine 2HCl,CV-4093 Calcium Channel
Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).
TQ0014 GNE-131 Sodium Channel
GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).
T1385 Amlodipine UK-48340 Calcium Channel
Amlodipine (UK-48340) is a synthetic dihydropyridine and a calcium channel blocker with antihypertensive and antianginal properties.
T12032 Mibefradil dihydrochloride Ro 40-5967 (dihydrochloride) Calcium Channel
Mibefradil dihydrochloride (Ro 40-5967 (dihydrochloride)) is an blocker of calcium channel with moderate selectivity for T-type Ca2+ channels (T-type and L-type currents with IC50s of 2.7 μM and 18.6 μM, respectively).
T10979 DCPIB Potassium Channel , Chloride channel
DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM, demonstrating at least 100-fold higher affinity over TREK1...
T0693 Niflumic acid Nifluril,Forenol,Landruma Others , Phospholipase , Chloride channel , COX , Monocarboxylate transporter , UGT
Niflumic acid (Nifluril) is a Ca2+-activated Cl- channel blocker and an analgesic and anti-inflammatory agent used in the therapy of rheumatoid arthritis.
T0946 Mepivacaine hydrochloride Mepivacaine HCl Sodium Channel
Mepivacaine hydrochloride (Mepivacaine HCl) is the hydrochloride salt form of mepivacaine, an amide derivative with local anesthetic properties.
T68143 Solpecainol Sodium Channel
solpecainol is a sodium channel blocker used in the study of neurological and cardiovascular diseases.
T3303 ML277 ML-277,CID-53347902 Potassium Channel
ML277 (CID-53347902) was identified as a potent activator of KCNQ1 channels (EC(50)=260 nM).
T8617 GMQ hydrochloride NSC 403387 hydrochloride Others
GMQ hydrochloride (NSC-403387 hydrochloride) is a potent and selective acid-sensing ion channel (ASIC) modulator. It activates ASIC3 channels under neutral pH and blocks acid-induced maximal peak current.
T4330 CaCCinh-A01 Chloride channel
CaCCinh-A01 is an inhibitor of the calcium-activated chloride channel (CaCC, 10 μM) and TMEM16A (IC50: 2.1 μM).
TQ0033 Zegocractin CM-4620,N-(5-(6-Chloro-2,2-difluorobenzo[d][1,3]dioxol-5-yl)pyrazin-2-yl)-2-fluoro-6-methylbenzamide,CM4620 Calcium Channel
Zegocractin (CM-4620) is a calcium-release activated calcium-channel (CRAC channel) inhibitor.
T7547 Ralfinamide mesylate FCE-26742A (mesylate) Sodium Channel
Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.
T68038 Celivarone Potassium Channel
Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and atrial fibrillation.
T13047 Synta66 Calcium Channel
Synta66 is a store-operated calcium entry channel Orai inhibitor, and used for the research of neurological disease.
T0008 Phenytoin sodium 5,5-Diphenylhydantoin sodium salt,Diphantoine,Dilantin sodium,Diphenylhydantoin Sodium Virus Protease , Sodium Channel
Phenytoin sodium (Diphantoine) is an inactive stabilizer for voltage-gated sodium channel .
T0386 Ropivacaine hydrochloride Ropivacaine monohydrochloride Potassium Channel , Sodium Channel
Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activity.
T10884 CRAC intermediate 1 5-(S)-Fluorowillardiine Calcium Channel
CRAC intermediate 1 (5-(S)-Fluorowillardiine) is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.
T2711 Chembridge-5861528 TCS 5861528 TRP/TRPV Channel
Chembridge-5861528 (TCS 5861528) is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx with IC50 values of 14.3 and 18.7 μM, respectively.
T1406 Amantadine hydrochloride 1-adamantanamine HCl,1-Adamantanamine hydrochloride,Symmetrel,CI-719,Amantadine HCl,1-Adamantylamine hydrochloride Dopamine Receptor , Influenza Virus
Amantadine hydrochloride (CI-719) is an antiviral that is used in the prophylactic or symptomatic treatment of influenza A and Parkinson disease.
TP1300 GsMTx4 TFA (1209500-46-8 free base) GsMTx4 TFA Piezo Channel
GsMTx4 TFA (1209500-46-8 free base) (GsMTx4 TFA) is a spider venom peptide that selectively inhibits cationic permeable mechanically-sensitive channels (MSCs) belonging to the Piezo and TRP channel families.
T28020 Mesendogen TRP/TRPV Channel
Mesendogen is an inhibitor of TRPM6. Mesendogen alters magnesium homeostasis, promotes mesoderm and definitive endoderm differentiation.
T4059 Selamectin UK-124114 Chloride channel , P-gp , Parasite
Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in nematodes. In an H. contortus larval development assay, sel...
T10690 Cav 2.2 blocker 1 Calcium Channel
Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
T8401 Efonidipine hydrochloride monoethanolate NZ-105 hydrochloride monoethanolate Calcium Channel
Efonidipine hydrochloride monoethanolate (NZ-105 hydrochloride monoethanolate) is a Ca(2+)-channel Blocker, Enhances the Production of Dehydroepiandrosterone Sulfate in NCI-H295R Human Adrenocortical Carcinoma Cells
T0386L Ropivacaine LEA-103 HCl Potassium Channel , Sodium Channel
Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.
T13059 T16Ainh-A01 Chloride channel
T16Ainh-A01 is a potent inhibitor of TMEM16A Chloride channel, inhibiting TMEM16A-mediated chloride currents (IC50 of 1 µM),and functions as a calcium-activated chloride channel (CaCC).
T6645 Ropivacaine hydrochloride monohydrate Ropivacaine HCl,Ropivacaine HCl monohydrate,LEA 103,LEA-103 HCl Potassium Channel , Sodium Channel
Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction in nerve fibres through inhibiting sodium ion influx reversibly.
T3651 YM-58483 YM 58483,BTP2 Calcium Channel
YM-58483 (BTP2) is a specific and effective inhibitor of CRAC channels and subsequent Ca2+ signals.

Compounds

Potassium Channel Activator 1
T10674
Synonym: ZINC34634569
Target: Potassium Channel
Calcium channel-modulator-1
T10101
Synonym:
Target: Others, Calcium Channel
1-EBIO
T2604
Synonym: 1-EBIO
Target: Calcium Channel
Fantofarone
T4669
Synonym: SR 33557
Target: Calcium Channel, Parasite
CNS-5161 hydrochloride
T10852
Synonym: CNS 5161A
Target: NMDAR
BMS-191095
T10566
Synonym:
Target: Potassium Channel
9-Phenanthrol
T22537
Synonym:
Target: TRP/TRPV Channel
AMPA receptor modulator-1
T10307
Synonym:
Target: iGluR
Lanthanum(III) chloride heptahydrate
T22353
Synonym:
Target: Calcium Channel
Metaflumizone
T7182
Synonym: BAS-320I
Target: Sodium Channel, Parasite
Nilvadipine
T1422
Synonym: FK235,FR34235,ARC029
Target: Calcium Channel
Raxatrigine
T2342
Synonym: CNV1014802,CNV 1014802,GSK-1014802,CNV-1014802
Target: Sodium Channel
DPhPC
T64561
Synonym:
Target: Others
Amlodipine Besylate
T0231
Synonym: Amlodipine benzenesulfonate
Target: Calcium Channel
QX-314 chloride
T12608
Synonym:
Target: Sodium Channel
Darodipine
T15053
Synonym: PY-108068,PY 108-068
Target: Calcium Channel
Endovion
T15233
Synonym: NS3728
Target: Chloride channel
NS1652
T16346
Synonym:
Target: Chloride channel
AUT1
T5183
Synonym:
Target: Potassium Channel
ML418
T16110
Synonym:
Target: Potassium Channel
Azelnidipine
T0121
Synonym: CS 905,UR-12592
Target: Calcium Channel
Manidipine dihydrochloride
T0193
Synonym: Manidipine 2HCl,CV-4093
Target: Calcium Channel
GNE-131
TQ0014
Synonym:
Target: Sodium Channel
Amlodipine
T1385
Synonym: UK-48340
Target: Calcium Channel
Mibefradil dihydrochloride
T12032
Synonym: Ro 40-5967 (dihydrochloride)
Target: Calcium Channel
DCPIB
T10979
Synonym:
Target: Potassium Channel, Chloride channel
Niflumic acid
T0693
Synonym: Nifluril,Forenol,Landruma
Target: Others, Phospholipase, Chloride channel, COX, Monocarboxylate transporter, UGT
Mepivacaine hydrochloride
T0946
Synonym: Mepivacaine HCl
Target: Sodium Channel
Solpecainol
T68143
Synonym:
Target: Sodium Channel
ML277
T3303
Synonym: ML-277,CID-53347902
Target: Potassium Channel
GMQ hydrochloride
T8617
Synonym: NSC 403387 hydrochloride
Target: Others
CaCCinh-A01
T4330
Synonym:
Target: Chloride channel
Zegocractin
TQ0033
Synonym: CM-4620,N-(5-(6-Chloro-2,2-difluorobenzo[d][1,3]dioxol-5-yl)pyrazin-2-yl)-2-fluoro-6-methylbenzamide,CM4620
Target: Calcium Channel
Ralfinamide mesylate
T7547
Synonym: FCE-26742A (mesylate)
Target: Sodium Channel
Celivarone
T68038
Synonym:
Target: Potassium Channel
Synta66
T13047
Synonym:
Target: Calcium Channel
Phenytoin sodium
T0008
Synonym: 5,5-Diphenylhydantoin sodium salt,Diphantoine,Dilantin sodium,Diphenylhydantoin Sodium
Target: Virus Protease, Sodium Channel
Ropivacaine hydrochloride
T0386
Synonym: Ropivacaine monohydrochloride
Target: Potassium Channel, Sodium Channel
CRAC intermediate 1
T10884
Synonym: 5-(S)-Fluorowillardiine
Target: Calcium Channel
Chembridge-5861528
T2711
Synonym: TCS 5861528
Target: TRP/TRPV Channel
Amantadine hydrochloride
T1406
Synonym: 1-adamantanamine HCl,1-Adamantanamine hydrochloride,Symmetrel,CI-719,Amantadine HCl,1-Adamantylamine hydrochloride
Target: Dopamine Receptor, Influenza Virus
GsMTx4 TFA (1209500-46-8 free base)
TP1300
Synonym: GsMTx4 TFA
Target: Piezo Channel
Mesendogen
T28020
Synonym:
Target: TRP/TRPV Channel
Selamectin
T4059
Synonym: UK-124114
Target: Chloride channel, P-gp, Parasite
Cav 2.2 blocker 1
T10690
Synonym:
Target: Calcium Channel
Efonidipine hydrochloride monoethanolate
T8401
Synonym: NZ-105 hydrochloride monoethanolate
Target: Calcium Channel
Ropivacaine
T0386L
Synonym: LEA-103 HCl
Target: Potassium Channel, Sodium Channel
T16Ainh-A01
T13059
Synonym:
Target: Chloride channel
Ropivacaine hydrochloride monohydrate
T6645
Synonym: Ropivacaine HCl,Ropivacaine HCl monohydrate,LEA 103,LEA-103 HCl
Target: Potassium Channel, Sodium Channel
YM-58483
T3651
Synonym: YM 58483,BTP2
Target: Calcium Channel
1 2 3 4
Cat No. Product Name Synonyms Targets
T8040 Cholesterol myristate Cholesteryl myristate,Cholesteryl tetradecanoate Others , Potassium Channel , GABA Receptor , Endogenous Metabolite , AChR
Cholesterol myristate (Cholesteryl myristate) is a natural steroid present in traditional Chinese medicine. Cholesterol myristate binds to several ion channels such as GABAA receptor, the nicotinic acetylcholine receptor...
T1381 Milbemycin oxime Others , Antibiotic , Parasite
Milbemycin oxime is a broad spectrum antiparasitic, used as a veterinary drug.
T2996 Tetrandrine NSC-77037,d-Tetrandrine,Hanfangchin A,Fanchinine,Sinomenine A Potassium Channel , Calcium Channel
Tetrandrine (Sinomenine A) is a natural, bis-benzylisoquinoline alkaloid isolated from the root of the plant. Tetrandrine non-selectively inhibits calcium channel activity and induces G1 blockade of the G1 phase of the c...
T2807 Caffeic Acid Lipoxygenase , Endogenous Metabolite , TRP/TRPV Channel
Caffeic Acid is an orally bioavailable, hydroxycinnamic acid derivative and polyphenol, with potential anti-oxidant, anti-inflammatory, and antineoplastic activities.
T2782 Catharanthine (+)-3, 4-Didehydrocoronaridine,(+)-3,4-Didehydrocoronaridine Calcium Channel , AChR
Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).
TN1081 Hirsuteine Dopamine Receptor
Hirsuteine is a natural product. It non-competitively antagonizes nicotine-mediated dopamine release by blocking ion permeation through nicotinic receptor channel complexes.
T3S0156 Atractyloside potassium salt Atractyloside Dipotassium Salt Others
1. Atractyloside potassium salt (Atractyloside Dipotassium Salt) inhibits oxidative phosphorylation by blocking the transfer of adenosine nucleotides through the mitochondrial membrane.
T16535 Picrotoxinin Chloride channel , GABA Receptor
Picrotoxinin is a blocker of chloride channel and a noncompetitive antagonist of GABAA with an IC50 of 1.15 μM for α1β2γ2L GABAA. Picrotoxinin shows convulsant properties.
T2720 Ginsenoside Rc Panaxoside Rc Others , TNF , GABA Receptor , Interleukin
Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.
T3013 Catharanthine tartrate Catharanthine hemitartrate Others , Calcium Channel
Catharanthine tartrate (Catharanthine hemitartrate) is an alkaloid from periwinkle that inhibits voltage-gated L-type calcium channels and has antitumor and hypotensive activities.
T1130 Gramicidin Gramicidinum,Gramicidine,Gramicidina MRP , Antibacterial , Antibiotic
A group of peptide antibiotics from BACILLUS brevis. Gramicidin (Gramicidine) C or S is a cyclic, ten-amino acid polypeptide and gramicidins A, B, D are linear. Gramicidin is one of the two principal components of TYROTH...
T4S1876 3-Deoxyaconitine Sodium Channel
3- Deoxyaconitine is a derivative of Aconitine (A189875), which activates tetrodotoxin-sensitive Na+ channels, inducing presynaptic depolarization, thus blocking the nerve action potential which, in turn, blocks the rele...
TN1035 Irisolidone IL Receptor , NF-κB , Chloride channel
Irisolidone is a potent volume-regulated anion channel (VRAC) current inhibitor, it exhibits high efficacy for VRAC blockade with IC50s of 5-13 μM.
T0690 Quinine 奎宁 Potassium Channel , Platelet aggregation , Parasite
Quinine is a natural cinchona alkaloid that has been used for centuries in the prevention and therapy of malaria. Quinine is also used for idiopathic muscle cramps. Quinine therapy has been associated with rare instances...
TWS1563 Incensole Others
1. Incensole has a protective or stimulating effect on β-cells of the rat pancreas, it also can increase the insulin secretion, which evidenced by a significant increase both in body weight and in liver glycogen.
T1131 Ivermectin MK-933 Mitophagy , GluCls , P2X Receptor , SARS-CoV , HIV Protease , Antibiotic , Parasite , Autophagy , HSV
Ivermectin (MK-933) is a glutamate-gated chloride channel (GluCls) activator, with antiparasitic activity.
T6856 Halofuginone Tempostatin,empostatin,RU-19110 Calcium Channel , DNA/RNA Synthesis , Sodium Channel , Parasite , TGF-beta/Smad
Halofuginone (RU-19110), the competitive inhibitor of prolyl-tRNA synthetase(Ki=18.3 nM), could also down-regulate Smad3 and blocked TGF-β signaling at 10 ng/ml in the mammal.
T1125 Shikonin NSC 252844,Isoarnebin 4,(+)-Shikonin,Alkanna Red,C.I. 75535,Anchusa acid TNF , NF-κB , Chloride channel , HIV Protease , PKM
Shikonin (Anchusa acid) is an TMEM16A chloride channel inhibitor (IC50: 6.5 μM). Shikonin is also a selective PKM2 inhibitor and can also suppress activation of the NF-κB pathway and inhibit TNF-α. Shikonin decreases exo...
T7177 Capsazepine Apoptosis , TRP/TRPV Channel
Capsazepine is an antagonist of TRPV1 receptor ( IC50 : 562 nM). Capsazepine blocks the painful sensation of heat caused by capsaicin (the active ingredient of chilli pepper) which activates the TRPV1 ion channel. It is ...
T2994 (E)-Cardamonin Alpinetin chalcone,Cardamomin,Cardamonin,(E)-Cardamoni Apoptosis , TRP/TRPV Channel
(E)-Cardamonin (Alpinetin chalcone) is a chalconoid that has been isolated from several plants including Alpinia katsumadai and Alpinia conchigera. It is a novel antagonist of hTRPA1 cation channel with an IC50 of 454 nM...
T1407 (-)-Menthol L-Menthol,Levomenthol,Menthomenthol,Menthacamphor Opioid Receptor , Endogenous Metabolite , TRP/TRPV Channel
(-)-Menthol (Levomenthol) is a levo isomer of menthol, an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local anesthetic properties. When added to pharmaceuticals and foo...
T4808 Agmatine sulfate Agmatine sulfate salt Endogenous Metabolite , NO Synthase , Imidazoline Receptor
Agmatine sulfate (Agmatine sulfate salt) is a bioactive metabolite of the arginine amino acid. It exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide sy...
T23735 Jamaicin An-Co-A4,AnCoA-4,An Co A4,AnCoA4 Calcium Channel
Jamaicin (AnCoA4), an isoflavone derived from the chickweed plant, is an inhibitor of the STIM1-Orai1 channel that blocks calcium influx, reduces its interaction with STIM1, and inhibits T-cell activation.
T4S0969 Obtusifolin Antioxidant , NF-κB
1. Obtusifolin has antioxidant properties and improves chemically induced diabetes and its complications by modulation of oxidative stress. 2. Obtusifolin suppresses phthalate esters-mediated bone resorption, thus may be...
T3243 Betaine Abromine,glycine betaine,oxyneurine,trimethylglycine,lycine Others , Endogenous Metabolite
Betaine (trimethylglycine) is a methyl derivative of glycine first isolated from sugar beets. It has been shown to have potential benefits for fighting heart disease, improving body composition, and helping promote muscl...
T5065 GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD Monosodium-GMP,cGMP sodium salt,Cyclic GMP PKA
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) , also known as cGMP, is a cellular regulatory agent and has been described as a second messenger. Its levels increase in response to a variety of hormones, inc...
T82764 Cd1a β-TRTX-cd1a,β-Theraphotoxin-cd1a
Cd1a, a β-toxin from the African spider Ceratogyrus darlingi, modulates calcium ion channels and inhibits human calcium ion channels (Ca v 2.2)(IC 50 2.6 μM) as well as mouse sodium ion channels (Na v 1.7). This compound...
T75722 Chlorotoxin TFA
Chlorotoxin TFA is a peptide isolated from the venom of the scorpion Leiurus quinquestriatus , acts as a chloride channel blocker [1] . Anti-cancer activity [2] .
T36439 Gramicidin A Antibacterial , HIF , Parasite
Gramicidin A is a peptide antibiotic isolated from B. brevis.Gramicidin A is a highly hydrophobic channel-forming ion carrier that forms monovalent cation-permeable channels in artificial membranes.Gramicidin A induces t...
T38484 Englerin A (-)-Englerin A TRP/TRPV Channel
Englerin A, a TRPC4 and TRPC5 channel agonist, is a compound from the East African plant Phyllanthus engleri with analgesic, anti-inflammatory, and anticancer activities that induces necrosis in human renal cancer cells.
T75333 Quinine hemisulfate hydrate
Quinine hemisulfate hydrate, an alkaloid derived from the bark of the cinchona tree, acts as an anti-malaria agent. Quinine hemisulfate hydrate is a potassium channel inhibitor that inhibits WT mouse Slo3 (K Ca 5.1) chan...

Natural Products

Cholesterol myristate
T8040
Synonym: Cholesteryl myristate,Cholesteryl tetradecanoate
Target: Others, Potassium Channel, GABA Receptor, Endogenous Metabolite, AChR
Milbemycin oxime
T1381
Synonym:
Target: Others, Antibiotic, Parasite
Tetrandrine
T2996
Synonym: NSC-77037,d-Tetrandrine,Hanfangchin A,Fanchinine,Sinomenine A
Target: Potassium Channel, Calcium Channel
Caffeic Acid
T2807
Synonym:
Target: Lipoxygenase, Endogenous Metabolite, TRP/TRPV Channel
Catharanthine
T2782
Synonym: (+)-3, 4-Didehydrocoronaridine,(+)-3,4-Didehydrocoronaridine
Target: Calcium Channel, AChR
Hirsuteine
TN1081
Synonym:
Target: Dopamine Receptor
Atractyloside potassium salt
T3S0156
Synonym: Atractyloside Dipotassium Salt
Target: Others
Picrotoxinin
T16535
Synonym:
Target: Chloride channel, GABA Receptor
Ginsenoside Rc
T2720
Synonym: Panaxoside Rc
Target: Others, TNF, GABA Receptor, Interleukin
Catharanthine tartrate
T3013
Synonym: Catharanthine hemitartrate
Target: Others, Calcium Channel
Gramicidin
T1130
Synonym: Gramicidinum,Gramicidine,Gramicidina
Target: MRP, Antibacterial, Antibiotic
3-Deoxyaconitine
T4S1876
Synonym:
Target: Sodium Channel
Irisolidone
TN1035
Synonym:
Target: IL Receptor, NF-κB, Chloride channel
Quinine
T0690
Synonym: 奎宁
Target: Potassium Channel, Platelet aggregation, Parasite
Incensole
TWS1563
Synonym:
Target: Others
Ivermectin
T1131
Synonym: MK-933
Target: Mitophagy, GluCls, P2X Receptor, SARS-CoV, HIV Protease, Antibiotic, Parasite, Autophagy, HSV
Halofuginone
T6856
Synonym: Tempostatin,empostatin,RU-19110
Target: Calcium Channel, DNA/RNA Synthesis, Sodium Channel, Parasite, TGF-beta/Smad
Shikonin
T1125
Synonym: NSC 252844,Isoarnebin 4,(+)-Shikonin,Alkanna Red,C.I. 75535,Anchusa acid
Target: TNF, NF-κB, Chloride channel, HIV Protease, PKM
Capsazepine
T7177
Synonym:
Target: Apoptosis, TRP/TRPV Channel
(E)-Cardamonin
T2994
Synonym: Alpinetin chalcone,Cardamomin,Cardamonin,(E)-Cardamoni
Target: Apoptosis, TRP/TRPV Channel
(-)-Menthol
T1407
Synonym: L-Menthol,Levomenthol,Menthomenthol,Menthacamphor
Target: Opioid Receptor, Endogenous Metabolite, TRP/TRPV Channel
Agmatine sulfate
T4808
Synonym: Agmatine sulfate salt
Target: Endogenous Metabolite, NO Synthase, Imidazoline Receptor
Jamaicin
T23735
Synonym: An-Co-A4,AnCoA-4,An Co A4,AnCoA4
Target: Calcium Channel
Obtusifolin
T4S0969
Synonym:
Target: Antioxidant, NF-κB
Betaine
T3243
Synonym: Abromine,glycine betaine,oxyneurine,trimethylglycine,lycine
Target: Others, Endogenous Metabolite
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD
T5065
Synonym: Monosodium-GMP,cGMP sodium salt,Cyclic GMP
Target: PKA
Cd1a
T82764
Synonym: β-TRTX-cd1a,β-Theraphotoxin-cd1a
Target:
Chlorotoxin TFA
T75722
Synonym:
Target:
Gramicidin A
T36439
Synonym:
Target: Antibacterial, HIF, Parasite
Englerin A
T38484
Synonym: (-)-Englerin A
Target: TRP/TRPV Channel
Quinine hemisulfate hydrate
T75333
Synonym:
Target:
Cat No. Product Name
L2300 Ion Channel Inhibitor Library

946 compounds
A unique collection of 946 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;
L7300 Potassium Channel Blocker Library

160 compounds
A unique collection of 160 potassium channel blockers and agonists for high throughput and high content screening;
L7400 Sodium Channel Blocker Library

128 compounds
A unique collection of 128 sodium channel blockers and agonists for high throughput and high content screening;
L7200 Calcium Channel Compound Library

143 compounds
A unique collection of 143 calcium channel blockers and agonists for high throughput and high content screening;
L2800 Serotonin Receptor-Targeted Compound Library

275 compounds
A unique collection of 275 compounds targeting serotonin receptors for high throughput screening and high content screening;
L9420 Exosome Compound Library

80 compounds
80 exosome-related compounds that can be used for high-throughput and high-content screening.
TargetMol