T0216 |
Eletriptan hydrobromide
|
177834-92-3
|
97.8%
|
|
Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor.
|
T12596 |
(4E)-SUN9221
|
222318-55-0
|
97.79%
|
|
(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in hypertens...
|
T22520 |
5-Carboxamidotryptamine maleate
|
74885-72-6
|
97.77%
|
|
5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.
|
T38507 |
Renzapride
|
112727-80-7
|
97.76%
|
|
Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist.Renzapride can be used in the study of constipation-pr...
|
T72322 |
R 59-022 hydrochloride
|
93076-98-3
|
97.7%
|
|
R 59-022 hydrochloride (DKGI-I hydrochloride) is a 5-HT Receptor antagonist that activates protein kinase C (PKC).R 59-022 hydrochloride is a DGK inhibitor (IC50...
|
T3046 |
BMY 7378 dihydrochloride
|
21102-95-4
|
97.67%
|
|
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
|
T14526 |
Bemesetron
|
40796-97-2
|
97.37%
|
|
Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.
|
T27795L |
(Iso)-Landipirdine
|
1000308-09-7
|
97.27%
|
|
(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist. (Iso)-Landipirdine has a significant effect on the hERG pharmacophore and can be...
|
T7521 |
Azaphen
|
24853-80-3
|
97.12%
|
|
Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.
|
T39161 |
Ro60-0175
|
169675-08-5
|
97.09%
|
|
Ro60-0175 a selective agonist for both the 5-hydroxytryptamine 2B (5-HT2B) and 5-hydroxytryptamine 2C (5-HT2C)serotonin receptor subtypes, commonly used as fumar...
|
T10989 |
Dehydroaripiprazole
|
129722-25-4
|
97.05%
|
|
Dehydroaripiprazole (DM-14857) is the active metabolite of aripiprazole. Aripiprazole is an antipsychotic drug, which is metabolized by CYP3A4 and CYP2D6 and mai...
|
T0076 |
Paliperidone
|
144598-75-4
|
96.98%
|
|
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically,...
|
T31592 |
E6801
|
528859-04-3
|
96.66%
|
|
E6801 is a novel selective 5-HT6 receptor agonist with a wide range of biological activities.E6801 can be used in the study of dementia, Parkinson's disease, dep...
|
T0965 |
Histamine
|
51-45-6
|
96.63%
|
|
Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial s...
|
T22833 |
H-9 dihydrochloride
|
116700-36-8
|
96.57%
|
|
H-9 dihydrochloride is a potent protein kinase (PKA) inhibitor.H-9 Dihydrochloride significantly reduces the excitatory response to 5-HT at low concentrations.H-...
|
T23325 |
SB 699551 dihydrochloride
|
864741-95-7
|
96.53%
|
|
SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.
|
T15034 |
Roluperidone
|
359625-79-9
|
96.46%
|
|
Roluperidone (CYR-101) is a novel cyclic amide derivative. It has high equipotent affinities for 5-HT2A and σ2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A an...
|
T35841 |
5-Benzyloxygramine
|
1453-97-0
|
96.33%
|
|
5-Benzyloxygramine is a N protein PPI orthosteric stabilizer that exhibits both antiviral and N-NTD protein-stabilizing activities[1].
5-benzyloxygramine stabili...
|
T3341 |
Elemicin
|
487-11-6
|
96.27%
|
|
Elemicin (Elemicine) is a constituent of several plant species' essential oils with anticholinergic effects in human.
|
T67851 |
Rac Desmethyl Citalopram Hydrochloride
|
97743-99-2
|
96.14%
|
|
rac Desmethyl Citalopram Hydrochloride is a 5-hydroxy tryptamine uptake inhibitor with IC50 value of 0.013 μM.
|