TN2116 |
Pteropodine
|
5629-60-7
|
98%
|
|
Pteropodine acts as a positive modulator of muscarinic M(1) and 5-HT(2) receptors. Pteropodine shows antigenotoxic, antioxidant and lymphocyte induction effects,...
|
T10996 |
Deramciclane
|
120444-71-5
|
98%
|
|
Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors. It acts as an antagonist in both receptor subtypes and has inverse agonist properties for 5-HT2C ...
|
T17253 |
WAY 163909
|
428868-32-0
|
98%
|
|
WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).
|
T15552 |
Iferanserin
|
58754-46-4
|
98%
|
|
Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors. Iferanserin has the potential fo...
|
T22921 |
LE 300
|
274694-98-3
|
98%
|
|
dopamine D1 receptor antagonist
|
TN1755 |
Hyperforin
|
11079-53-1
|
98%
|
|
Hyperforin acts as an angiogenesis inhibitor, it as a possible antidepressant component of hypericum extracts.
|
T22340 |
Granisetron
|
109889-09-0
|
98%
|
|
Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.
|
T10192 |
7-Desmethyl-3-hydroxyagomelatine
|
166527-00-0
|
98%
|
|
7-Desmethyl-3-hydroxyagomelatine is a metabolite of Agomelatine and has less activity than Agomelatine. Agomelatine is a melatonergic (MT1 and MT2) agonist and 5...
|
T26622 |
Ampreloxetine
|
1227056-84-9
|
98%
|
|
Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.
|
T16399 |
Opiranserin
|
1441000-45-8
|
98%
|
|
Opiranserin is a development as an injectable agent for the treatment of postoperative pain. Opiranserin is a non-opioid and non-NSAID analgesic candidate and is...
|
T10294 |
AM9405
|
T10294
|
98%
|
|
AM9405 is a novel peripherally active cannabinoid type 1 (CB1) and serotonin type 3 receptor agonist. AM9405 inhibits twitch contraction of the ileum and the col...
|
T12843 |
SB-399885 hydrochloride
|
402713-81-9
|
98%
|
|
SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.
|
T16556 |
PNU-142633
|
187665-65-2
|
98%
|
|
PNU-142633 has anti-migraine efficacy. PNU-142633 is a high affinity and selective 5-HT1D receptor agonist (Kis of 6 nM and > 18 000 nM for human 5-HT1D receptor...
|
T10611 |
Brexpiprazole S-oxide D8
|
2748605-29-8
|
98%
|
|
Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium labeled Brexpiprazole S-oxide. Brexpiprazole S-oxide is a main metabolite of Brexpiprazole. Brexpiprazole is...
|
T10344 |
AP521
|
151227-08-6
|
98%
|
|
AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).
|
TN1790 |
Isopteropodine
|
5171-37-9
|
98%
|
|
Isopteropodine (Uncarine E) is an isoyohimbine-type octindole alkaloid isolated from Hamelia patens micropropagated and has antimicrobial activity and stimulates...
|
T21360 |
Asenapine
|
65576-45-6
|
98%
|
|
Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, dopamine receptor, and histamine receptor antagonist with antipsychotic effects that is used to tre...
|
T12631 |
(R)-Mirtazapine D3
|
T12631
|
98%
|
|
(R)-Mirtazapine D3 is a deuterium labeled (R)-Mirtazapine.(R)-Mirtazapine is a antagonist of 5-HT3 receptor.
|
T10267 |
Agomelatine (L(+)-Tartaric acid)
|
824393-18-2
|
98%
|
|
Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and ...
|
T10498 |
5-HT2A antagonist 1
|
204643-75-4
|
98%
|
|
5-HT2A antagonist 1 is a 5-HT2A antagonist. It may be useful in the treatment of gastrointestinal disorders circulatory disorders.
|