5-HT Receptor

5-hydroxytryptamine receptors or 5-HT receptors, or serotonin receptors, are a group of G protein-coupled receptor and ligand-gated ion channels found in the central and peripheral nervous systems. They mediate both excitatory and inhibitory neurotransmission.

Cat. No.	Product name	CAS No.	Purity
T20828	Citalopram	59729-33-8	99.89%
T20828	Citalopram (Lu 10-171 is an orally active, selective serotonin reuptake inhibitor (SSRI), a selective 5-hydroxytryptamine reuptake inhibitor, and a racemic mixtu...
T27117	DA-6886	1645260-76-9	99.89%
T27117	DA-6886 is an agonist 5-Hydroxytryptamine receptor 4 (5-HT4). DA-6886 induced relaxation of the rat oesophagus preparation in a 5-HT4 receptor antagonist-sensiti...
T2874	Tetrahydroberberine	522-97-4	99.89%
T2874	Tetrahydroberberine (Canadine) is an isoquinoline alkaloid isolated from corydalis tuber, has a micromolar affinity for dopamine D(2) receptors.
T6602	Naratriptan hydrochloride	143388-64-1	99.89%
T6602	Naratriptan Hydrochloride is the hydrochloride salt form of naratriptan, a sulfonamide with selective serotonin (5-HT) 1 receptor agonistic activity and anti-mig...
T16759	Ritanserin	87051-43-2	99.89%
T16759	Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine ...
T1042	Granisetron hydrochloride	107007-99-8	99.88%
T1042	Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy pati...
T23310	SB-203186 hydrochloride	207572-69-8	99.88%
T23310	SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist
T6597	Mosapride Citrate	112885-42-4	99.88%
T6597	Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.
T7135	Phenylbiguanide	102-02-3	99.87%
T7135	Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)
T0678	Amitriptyline hydrochloride	549-18-8	99.87%
T0678	Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive ...
T24421	LY-2624803	879409-35-5	99.87%
T24421	LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.
T22379L	NLX-204 hydrochloride（2170405-10-2 free base）	T22379L	99.87%
T22379L	NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).
T1580	Desvenlafaxine	93413-62-8	99.86%
T1580	Desvenlafaxine (O-Desmethylvenlafaxine) is a cyclohexanol and phenol derivative and metabolite of venlafaxine that functions as a serotonin and noradrenaline reu...
T2589	Dolasetron Mesylate hydrate	878143-33-0	99.86%
T2589	Dolasetron Mesylate hydrate (Dalasetron Mesylate Hydrate) , a selective serotonin receptor antagonist, competitively blocks the action of serotonin at 5HT3 recep...
T23312	SB 204741	152239-46-8	99.86%
T23312	SB 204741 is a 5-HT2B receptor antagonist.
T10169	5-HT4 antagonist 1	261766-73-8	99.86%
T10169	5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).
T2209	Serotonin hydrochloride	153-98-0	99.86%
T2209	Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (COMT...
T1445	Agomelatine	138112-76-2	99.86%
T1445	Agomelatine (Valdoxan) is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-...
TN1032	Geissoschizine methyl ether	60314-89-8	99.86%
TN1032	Geissoschizine methyl ether, a major indole alkaloid found in Uncaria hook, is a major active component of Yokukansan with psychotropic effects. Geissoschizine m...
T0482	Sertraline hydrochloride	79559-97-0	99.86%
T0482	Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.