Home Tools
Log in
Cart

AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TN2217 Sophoflavescenol 216450-65-6 99.65%
Sophoflavescenol
Sophoflavescenol is a mixed inhibitor of PDE5 with a K(i) value of 0.005 microM. Sophoflavescenol has antioxidant, anti-inflammatory, and apoptotic effects , the...
TN1798 Isorosmanol 93780-80-4 98.85%
Isorosmanol
Isorosmanol possesses antioxidant, neuroprotective and neurotrophic effects, it might be useful in ageing disorders such as the declining of cognitive functions ...
T0346 Camylofine 54-30-8 98%
Camylofine
Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.
TN1519 (S)-Coclaurine 486-39-5 97.72%
(S)-Coclaurine
(S)-Coclaurine (Coclaurine) is an antagonist of nAChR isolated from Sarcopetalum harveyanum.
T8702 SKF-83566 99295-33-7 95.00%
SKF-83566
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 n...
T68019 Ursulcholic acid 88426-32-8 100%
Ursulcholic acid
Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
T1236 Pentolinium Tartrate 52-62-0
Pentolinium Tartrate
Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.
T0218 Biperiden 514-65-8
Biperiden
Biperiden (Bipariden) is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteri...
T13129 Terodiline hydrochloride 7082-21-5 98%
Terodiline hydrochloride
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bl...
T6721 Vinblastine 865-21-4 98%
Vinblastine
Vinblastine inhibits microtubule formation and suppresses nAChR activity with IC50 of 8.9 μM, used to treat certain kinds of cancer.
TN4837 Pseudotaraxasterol 464-98-2 98%
Pseudotaraxasterol
Pseudotaraxasterol shows cytotoxic activity against MOLT-4 cells.
TN3696 Conodurine 2665-57-8 98%
Conodurine
Conodurine shows leishmanicidal and antibacterial activities, it shows inhibition activity for acetyl (AChE) and butyrylcholinesterase (BuChE).
TN1559 Dehydrodicentrine 19843-03-9 98%
Dehydrodicentrine
Dehydrodicentrine showed strong acetylcholinesterase (AChE) inhibitory effects with the IC50 value of 2.98 μM.
T12020 Metixene hydrochloride 1553-34-0 98%
Metixene hydrochloride
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
TN1645 Flavokawain C 56798-34-6 98%
Flavokawain C
Flavokawain C is a melanogenesis inhibitor, it inhibited melanogenesis with IC50 values of 6.9 μM. Flavokawain C has anti-tumor activity, it inhibited cell cycle...
TN1653 Fustin 20725-03-5 98%
Fustin
Fustin is the phytogenic flavanol component of the plant Rhus verniciflua Stokes. Fustin shows protective effects on 6-hydroxydopamine-induced neuronal cell deat...
TN3380 Alloisoimperatorin 35214-83-6 98%
Alloisoimperatorin
Alloisoimperatorin is a candidate of AChE inhibitors, it displays potent antioxidant effects against the DPPH radical and against renal epithelial cell injury by...
T13713 GP531 142344-87-4 98%
GP531
GP531 is a second-generation adenosine regulating agent. It is pharmacologically silent under basal conditions but increases localized endogenous adenosine durin...
TN2505 1,5-Diphenylpentan-1-one 39686-51-6 98%
1,5-Diphenylpentan-1-one
1,5-Diphenylpentan-1-one shows poor insecticidal and acetylcholinesterase inhibitory activities.
TN4652 Niazimicin 147821-49-6 98%
Niazimicin
Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in...
Sophoflavescenol
TN2217
Sophoflavescenol is a mixed inhibitor of PDE5 with a K(i) value of 0.005 microM. Sophoflavescenol has antioxidant, anti-inflammatory, and apoptotic effects , the...
Isorosmanol
TN1798
Isorosmanol possesses antioxidant, neuroprotective and neurotrophic effects, it might be useful in ageing disorders such as the declining of cognitive functions ...
Camylofine
T0346
Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.
(S)-Coclaurine
TN1519
(S)-Coclaurine (Coclaurine) is an antagonist of nAChR isolated from Sarcopetalum harveyanum.
SKF-83566
T8702
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 n...
Ursulcholic acid
T68019
Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
Pentolinium Tartrate
T1236
Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.
Biperiden
T0218
Biperiden (Bipariden) is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteri...
Terodiline hydrochloride
T13129
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bl...
Vinblastine
T6721
Vinblastine inhibits microtubule formation and suppresses nAChR activity with IC50 of 8.9 μM, used to treat certain kinds of cancer.
Pseudotaraxasterol
TN4837
Pseudotaraxasterol shows cytotoxic activity against MOLT-4 cells.
Conodurine
TN3696
Conodurine shows leishmanicidal and antibacterial activities, it shows inhibition activity for acetyl (AChE) and butyrylcholinesterase (BuChE).
Dehydrodicentrine
TN1559
Dehydrodicentrine showed strong acetylcholinesterase (AChE) inhibitory effects with the IC50 value of 2.98 μM.
Metixene hydrochloride
T12020
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
Flavokawain C
TN1645
Flavokawain C is a melanogenesis inhibitor, it inhibited melanogenesis with IC50 values of 6.9 μM. Flavokawain C has anti-tumor activity, it inhibited cell cycle...
Fustin
TN1653
Fustin is the phytogenic flavanol component of the plant Rhus verniciflua Stokes. Fustin shows protective effects on 6-hydroxydopamine-induced neuronal cell deat...
Alloisoimperatorin
TN3380
Alloisoimperatorin is a candidate of AChE inhibitors, it displays potent antioxidant effects against the DPPH radical and against renal epithelial cell injury by...
GP531
T13713
GP531 is a second-generation adenosine regulating agent. It is pharmacologically silent under basal conditions but increases localized endogenous adenosine durin...
1,5-Diphenylpentan-1-one
TN2505
1,5-Diphenylpentan-1-one shows poor insecticidal and acetylcholinesterase inhibitory activities.
Niazimicin
TN4652
Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in...
1 2 3 4 5 ... 21
TargetMol