AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.

Cat. No.	Product name	CAS No.	Purity
TN3243	7-O-Methyleriodictyol	51857-11-5	99.38%
TN3243	7-O-Methyleriodictyol is a flavanone isolated from Artemisia monosperma and shows biological effects on rat isolated smooth muscles.
T68599	Orphenadrine	83-98-7	99.38%
T68599	Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner, producin...
T0130	Physostigmine Salicylate	57-64-7	99.36%
T0130	Physostigmine, a parasympathomimetic alkaloid, is a reversible cholinesterase inhibitor. It extracts from the Calabar bean.
T1266	Terfenadine	50679-08-8	99.36%
T1266	Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist...
T0786	Clidinium bromide	3485-62-9	99.36%
T0786	Clidinium bromide (Ro 2-3773) , a synthetic anticholinergic agent, has been shown in experimental and clinical researchers to have a pronounced antisecretory and...
T7695	PNU-282987 S enantiomer free base	737727-12-7	99.35%
T7695	PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).
T14065	9-Ethyladenine	2715-68-6	99.35%
T14065	9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].
T68154	TC-2216	646055-67-6	99.33%
T68154	TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.
T8448	ZSET1446	887603-94-3	99.32%
T8448	ZSET1446 (ST-101) is a T-type calcium channel activator potentially for the treatment of learning deficits in various types of Alzheimer disease (AD) models.
T0804	Pilocarpine Hydrochloride	54-71-7	99.29%
T0804	Pilocarpine Hydrochloride (NSC 5746 HCl) , a nonselective muscarinic acetylcholine receptor agonist, is utilized to produce an experimental model of epilepsy.
TP2058L	Catestatin acetate	TP2058L	99.28%
TP2058L	Catestatin acetate is a non-competitive antagonist of nAChR and inhibits catecholamine release. Catestatin acetate regulates cardiac function and blood pressure....
T68953	Arecoline	63-75-2	99.28%
T68953	Arecoline is a natural alkaloid derived from areca nut in the palm family and is a potent nicotine and partial agonist of muscarinic acetylcholine receptors. Are...
T7224	Anabasine	494-52-0	99.27%
T7224	Anabasine ((S)-Anabasine) is an alkaloid extracted from tobacco. Anabasine is a full agonist of nicotinic acetylcholine receptors (nAChRs) with insecticidal acti...
T0166	Pancuronium dibromide	15500-66-0	99.27%
T0166	Pancuronium dibromide (Pavulon), a competitive AChR antagonist (IC50 = 5.5 nM), acts as a skeletal muscle relaxant. Pancuronium dibromide(Pancuronium bromide) bl...
T9018	JHU37160	2369979-68-8	99.25%
T9018	JHU37160 (JHU 37160) is a Designer Receptors Exclusively Activated by Designer Drug (DREADD) agonist with Ki of 1.9 nM and 3.6 nM for human muscarinic acetylchol...
T29123	VU0152099	612514-42-8	99.24%
T29123	VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).
T7052	Gnetol	86361-55-9	99.21%
T7052	Gnetol competitivity inhibits butyrylcholinesterase (IC50: 1.3 uM). Gnetol has a strong inhibitory effect on murine tyrosinase activity. Gnetol significantly sup...
T4246	Varenicline dihydrochloride	866823-63-4	99.21%
T4246	Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.
T0794	Mepenzolate Bromide	76-90-4	99.21%
T0794	Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.
T0086	Galanthamine hydrobromide	1953-04-4	99.19%
T0086	Galanthamine hydrobromide (Galantamine hydrobromide), a long-acting and centrally active AChE inhibitor (IC50:410 nM), is an allosteric potentiator at neuronal n...