AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.

Cat. No.	Product name	CAS No.	Purity
T3324	Lycorine	476-28-8	98.71%
T3324	Lycorine (Narcissine) inhibits protein synthesis and may inhibit ascorbic acid biosynthesis, although studies on the latter are controversial and inconclusive.
T1049	Oxybutynin chloride	1508-65-2	98.71%
T1049	Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties. It competitively antagonizes the M1, M2, ...
T3720	Tebanicline hydrochloride	203564-54-9	98.71%
T3720	Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.
T67790	Biricodar dicitrate	174254-13-8	98.67%
T67790	Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.
T10066	2',5'-Dideoxyadenosine	6698-26-6	98.66%
T10066	2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
T4494	CLOZAPINE N-OXIDE	34233-69-7	98.65%
T4494	Clozapine N-oxide is the major metabolite of Clozapine and is blood-brain barrier permeable. Clozapine N-oxide is an agonist of DREADDs and activates the DREADD ...
T34573	SCH-900271	915210-50-3	98.64%
T34573	SCH-900271 is a potent nicotinic acid receptor for the treatment of dyslipidaemia and is commonly used in the study of mixed hyperlipidaemia and primary hypercho...
T21532	Anisodamine	55869-99-3	98.63%
T21532	Anisodamine (6-beta-Hydroxyhyoscyamine) is an antagonist of muscarinic and nicotinic cholinoceptor with similar affinities at the muscarinic receptor as scopolam...
T11366	Garcinol	78824-30-3	98.59%
T11366	Garcinol also inhibits histone acetyltransferases (HATs, IC50= 7 μM) and p300/CPB-associated factor (PCAF, IC50 = 5 μM). Garcinol has anti-inflammatory and anti-...
T10914	Cyclodrine hydrochloride	78853-39-1	98.59%
T10914	Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of neurologica...
T1475	Fesoterodine fumarate	286930-03-8	98.55%
T1475	Fesoterodine fumarate (Toviaz) is the fumarate salt form of fesoterodine, a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasm...
T11004	Desformylflustrabromine hydrochloride	951322-11-5	98.51%
T11004	Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.48...
T13066	TAK-071	1820812-16-5	98.47%
T13066	TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).
T12820	S16961	153874-14-7	98.43%
T12820	S16961 (S169611) is an agonist of nicotinic receptor.
T22329	Ethyl (triphenylphosphoranylidene) acetate	1099-45-2	98.43%
T22329	Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.
T7780	Blarcamesine	195615-83-9	98.42%
T7780	Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.
T6607	Nitenpyram	150824-47-8	98.42%
T6607	Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.
T8193	α-Thujone	546-80-5	98.41%
T8193	α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.
T7079	Batefenterol	743461-65-6	98.4%
T7079	Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic an...
T27679	JNJ-39393406	953428-73-4	98.36%
T27679	JNJ-39393406 is an α7 nicotinic acetylcholine receptor positive allosteric modulator for the study of tobacco dependence and Alzheimer's disease.