T13325 |
VU 0365114
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1208222-39-2
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VU 0365114 is a positive allosteric modulator of mAChR M5 (EC50: 2.7 μM).
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T9787 |
Suvn-911
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2414674-71-6
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suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.
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PDK0015 |
4-Hydroxycoumarin
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1076-38-6
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4-Hydroxycoumarin is a coumarin derivative and one of the versatile heterocyclic scaffolds with electrophilic and nucleophilic properties.
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T1179 |
Tiotropium bromide
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136310-93-5
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Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD). T...
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T1007 |
Nanofin
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504-03-0
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Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.
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T0594 |
Diphenmanil methylsulfate
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62-97-5
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Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors and thus decreases secretory exc...
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T6301 |
Tosedostat
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238750-77-1
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Tosedostat (CHR-2797) is an orally bioavailable inhibitor of the M1 family of aminopeptidases with potential antineoplastic activity. Tosedostat is converted int...
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T3S1612 |
Kuwanon G
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75629-19-5
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1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective ...
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TN1544 |
D-Menthol
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15356-60-2
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D-Menthol ((+)-MENTHOL) is a common compound in pharmaceutical and commercial products and a popular additive to cigarettes, it attenuates α±7 mediated Ca 2+ tra...
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TP2063 |
α-Conotoxin MII
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175735-93-0
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α-Conotoxin MII is a highly potent and selective competitive antagonist for α3β2 subunit-containing nicotinic receptors (IC50 = 0.5 - 3.5 nM at α3β2 expressed in...
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T8725 |
A 582941 HCl (848591-90-2(free base))
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T8725
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A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties
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T2555 |
Aclidinium bromide
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320345-99-1
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Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis or ...
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T0401 |
Benzethonium chloride
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121-54-0
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Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.
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T0296 |
Pempidine
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79-55-0
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Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.
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T8702 |
SKF-83566
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99295-33-7
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SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 n...
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T12201 |
Nebracetam hydrochloride
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1177279-49-0
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Nebracetam hydrochloride (WEB 1881 FU hydrochloride) is an agonist nootropic M1-muscarinic. Nebracetam hydrochloride induces a rise of intracellular Ca2+ concent...
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T1072 |
Loxeen
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6856-31-1
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Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.
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T22016 |
A-582941 dihydrochloride
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848591-90-2
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A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial
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T0976 |
Propoxur
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114-26-1
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Propoxur (Propoxure) is an insecticide used to control cockroaches, flies, mosquitoes, and lawn and turf insects. Acute (short-term) exposure of humans to propox...
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T0098 |
Ipratropium bromide monohydrate
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66985-17-9
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Ipratropium bromide monohydrate (Ipratropium bromide hydrate) is a muscarinic antagonist structurally related to ATROPINE but often considered safer and more eff...
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