TN2131 |
Questin
|
3774-64-9
|
98%
|
|
Questin is an antimicrobial agent derived from Aspergillus florescens with an antimicrobial activity profile that inhibits V. harveyi, V. anguillarum, V. cholera...
|
T17312 |
(+)-Phenserine
|
116839-68-0
|
98%
|
|
(+)-Phenserine is a novel selective inhibitor of cholinesterase non-competitive (IC50: 45.3 μM).
|
T16353 |
Meseclazone
|
29053-27-8
|
98%
|
|
Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.
|
TN4426 |
Leojaponin
|
864817-63-0
|
98%
|
|
Leojaponin is a prolyl oligopeptidase (POP) inhibitor. Leojaponin exhibits significant cytoprotective activities against glutamate-induced toxicity at concentrat...
|
TN3285 |
8-Hydroxypinoresinol
|
81426-17-7
|
98%
|
|
8-Hydroxypinoresinol has antioxidant activity,it and phillygenin significantly reduce the cell injury by 3-morpholinosydnonimine (SIN-1), a ONOO- generator, may ...
|
TN4492 |
Mangostanol
|
184587-72-2
|
98%
|
|
Mangostanol is an acetylcholinesterase (AChE) selective inhibitor.Mangostanol has anti-cancer activity, it shows significant activities against the CEM-SS cell l...
|
TL0018 |
Lobelin
|
90-69-7
|
98%
|
|
Inhalation challenge with capsaicin and rapid intravenous injection of Lobelin and alinamin indicated that peripheral c-fiber receptors were involved in the indu...
|
TN5193 |
Tubotaiwine
|
6711-69-9
|
98%
|
|
Tubotaiwine shows selective activity against L. infantum. Tubotaiwine and apparicine have affinity for adenosine receptors in the micromolar range and also have ...
|
T14966 |
Cimetropium Bromide
|
51598-60-8
|
98%
|
|
Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.
|
T12825 |
Timepidium bromide
|
35035-05-3
|
98%
|
|
Timepidium bromide is an agent of anticholinergic.
|
TN3287 |
8-Lavandulylkaempferol
|
883859-83-4
|
98%
|
|
8-Lavandulylkaempferol exhibits significant inhibitory effects with IC(50) values of 7.10 and 8.11 microM for butyrylcholinesterase and acetylcholinesterase, res...
|
T12766 |
RPR121056
|
181467-56-1
|
98%
|
|
RPR121056 is a Irinotecan metabolite, which is generated by CYP3A4. Irinotecan is an antineoplastic agent that inhibits topoisomerase type I.
|
TN3550 |
Buxbodine B
|
390362-51-3
|
98%
|
|
Buxbodine B has weak anti-AChE activity with IC50 values in the range of 10.8-98μM.
|
T12136 |
N-0861 racemate
|
121241-87-0
|
98%
|
|
N-0861 racemate is the racemate of N-0861.
|
TN3812 |
Dehydrovomifoliol
|
39763-33-2
|
98%
|
|
Dehydrovomifoliol could be a marker of Polish heather honey. Dehydrovomifoliol exhibits moderate acetylcholinesterase (AChE) inhibitory activities. Dehydrovomifo...
|
TN4286 |
Isodunnianol
|
139726-30-0
|
98%
|
|
Isodunnianol exhibits anti-AChE activity with an IC50 value of 13.0 uM; it also exhibits neurite outgrowth-promoting activity at the concentration ranging from 0...
|
T8306 |
Epiberberine chloride
|
889665-86-5
|
98%
|
|
Epiberberine chloride (Epiberberine (chloride)) is an alkaloid isolated from Coptis chinensis, acts as a potent AChE and BChE inhibitor, and a non-competitive BA...
|
T19933 |
GTS-21
|
148372-04-7
|
98%
|
|
GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.
|
TN4600 |
Myrianthic acid
|
89786-84-5
|
98%
|
|
Myrianthic acid shows anticancer activity, it shows inhibitory activities on foam cell formation in human monocyte-derived macrophages induced by acetylated low-...
|
TN3744 |
Cyclomorusin
|
62596-34-3
|
98%
|
|
Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of s...
|