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AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T16563 Pozanicline 161417-03-4 98%
Pozanicline
Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
TN1790 Isopteropodine 5171-37-9 98%
Isopteropodine
Isopteropodine (Uncarine E) is an isoyohimbine-type octindole alkaloid isolated from Hamelia patens micropropagated and has antimicrobial activity and stimulates...
TN3875 Dipterocarpol 471-69-2 98%
Dipterocarpol
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng. Dipterocarpol A shows moderate acetylcholinesterase inhibitory a...
TN2067 Picfeltarraegenin X 1391826-61-1 98%
Picfeltarraegenin X
Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
T12525 Pozanicline dihydrochloride 161416-61-1 98%
Pozanicline dihydrochloride
Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)
T12191 NBTGR 13153-27-0 98%
NBTGR
NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
T19623 α-Muricholic acid 2393-58-0 98%
α-Muricholic acid
α-Muricholic acid is the most abundant primary bile acid in rodents.
TN2504 1,5-Dihydroxyxanthone 14686-65-8 98%
1,5-Dihydroxyxanthone
1,5-Dihydroxyxanthone exhibits the epidermal growth factor receptor (EGFR) -tyrosine kinase inhibitory activity, with the IC50 value of 90.34 nM. It may have ant...
TN4812 Pluviatolide 28115-68-6 98%
Pluviatolide
(-)-Pluviatolide can inhibit electrically-induced and acetylcholine-induced contraction in the isolated guinea-pig ileum.
T16417 Oxitropium Bromide 30286-75-0 98%
Oxitropium Bromide
Oxitropium bromide is a mAChR antagonist. It is used as an anticholinergic bronchodilator drug for the treatment of asthma and chronic obstructive pulmonary dise...
T13256 UP202-56 163838-04-8 98%
UP202-56
UP202-56 is an adenosinergic agonist and is an adenosine analog.
TN4456 Lucidadiol 252351-95-4 98%
Lucidadiol
Lucidadiol exhibits butyrylcholinesterase-inhibitory activity at concentrations up to 200 uM, it also possesses inhibitory activity against acetylcholinesterase ...
T12868 Sch412348 377727-26-9 98%
Sch412348
Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
TN1409 Asimilobine 6871-21-2 98%
Asimilobine
(-)-Asimilobine shows antioxidative, anti-acetylcholinesterase (AChE), anti-α±-glucosidase, anti-leishmanial and anti-fungal activities; it displays weak inhibit...
T10731 CDD0102 146422-58-4 98%
CDD0102
CDD0102 is a potent agonist of M1 Muscarinic receptor.
T12446 Phenserine 101246-66-6 98%
Phenserine
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
T5476 MAChr-in-1 119391-56-9 98%
mAChr-in-1
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
T13772 MHP 133 147340-43-0 98%
MHP 133
MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
TP2065L α-Conotoxin PIA acetate 98%
α-Conotoxin PIA acetate
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.
T8868 4BP-TQS 360791-49-7 99.99%
4BP-TQS
4BP-TQS is an allosteric agonist of α7 nAChRs.
Pozanicline
T16563
Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
Isopteropodine
TN1790
Isopteropodine (Uncarine E) is an isoyohimbine-type octindole alkaloid isolated from Hamelia patens micropropagated and has antimicrobial activity and stimulates...
Dipterocarpol
TN3875
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng. Dipterocarpol A shows moderate acetylcholinesterase inhibitory a...
Picfeltarraegenin X
TN2067
Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
Pozanicline dihydrochloride
T12525
Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)
NBTGR
T12191
NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
α-Muricholic acid
T19623
α-Muricholic acid is the most abundant primary bile acid in rodents.
1,5-Dihydroxyxanthone
TN2504
1,5-Dihydroxyxanthone exhibits the epidermal growth factor receptor (EGFR) -tyrosine kinase inhibitory activity, with the IC50 value of 90.34 nM. It may have ant...
Pluviatolide
TN4812
(-)-Pluviatolide can inhibit electrically-induced and acetylcholine-induced contraction in the isolated guinea-pig ileum.
Oxitropium Bromide
T16417
Oxitropium bromide is a mAChR antagonist. It is used as an anticholinergic bronchodilator drug for the treatment of asthma and chronic obstructive pulmonary dise...
UP202-56
T13256
UP202-56 is an adenosinergic agonist and is an adenosine analog.
Lucidadiol
TN4456
Lucidadiol exhibits butyrylcholinesterase-inhibitory activity at concentrations up to 200 uM, it also possesses inhibitory activity against acetylcholinesterase ...
Sch412348
T12868
Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
Asimilobine
TN1409
(-)-Asimilobine shows antioxidative, anti-acetylcholinesterase (AChE), anti-α±-glucosidase, anti-leishmanial and anti-fungal activities; it displays weak inhibit...
CDD0102
T10731
CDD0102 is a potent agonist of M1 Muscarinic receptor.
Phenserine
T12446
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
mAChr-in-1
T5476
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
MHP 133
T13772
MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
α-Conotoxin PIA acetate
TP2065L
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.
4BP-TQS
T8868
4BP-TQS is an allosteric agonist of α7 nAChRs.
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TargetMol