AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.

Cat. No.	Product name	CAS No.	Purity
T0268	Lobeline hydrochloride	134-63-4	99.65%
T0268	Lobeline hydrochloride (α-Lobeline hydrochloride) is a nicotinic receptor agonist, acting as an effective antagonist at both α4β2 and α3β2 neuronal nicotinic rec...
T16881L	SIB 1553A	191611-76-4	99.64%
T16881L	SIB 1553A is an orally available and selective agonist of nicotinic acetylcholine receptors (nAChRs), which are subtype-selective ligands for nicotinic acetylcho...
T0703	Flavoxate hydrochloride	3717-88-2	99.64%
T0703	Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.
T0364	Dibucaine	85-79-0	99.64%
T0364	Dibucaine (Cinchocaine), a local anesthetic of the amide type, is now usually used for surface anesthesia.
T6744	Methylbenactyzium Bromide	3166-62-9	99.63%
T6744	Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.
T0051	Urethane	51-79-6	99.63%
T0051	Urethane (Ethylurethane) was an antineoplastic agent .Now is used for other medicinal purposes.
T28722	SCH 57790	221660-80-6	99.62%
T28722	SCH 57790 is a novel and selective muscarinic M(2) receptor antagonist that releases acetylcholine and enhances cognition in experimental animals for the treatme...
T1542	Pirenzepine dihydrochloride	29868-97-1	99.62%
T1542	Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.
T4960	VASICINE	6159-55-3	99.62%
T4960	Vasicine is oxytocic and abortifacient agents.Vasicine, a potential natural cholinesterase inhibitor, has been in development for treatment of Alzheimer's diseas...
T36640	Xanomeline	131986-45-3	99.61%
T36640	Xanomeline (LY-246708) is a functionally selective M1/M4 activator used in the study of neurological disorders such as schizophrenia and has shown promising trea...
T7056	Dronedarone	141626-36-0	99.58%
T7056	Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
T2939	Forskolin	66575-29-9	99.57%
T2939	Forskolin (Coleonol) is a natural product, an adenylate cyclase activator (EC50=0.5 μM). Forskolin increases cAMP levels, activates PXR and FXR, and induces auto...
T29687	Afacifenacin	877606-63-8	99.57%
T29687	Afacifenacin (SMP-986) fumarate is an M3 muscarinic receptor-selective antagonist used in the study of ischemic heart disease, urinary incontinence and cystitis ...
T15658	KH7	330676-02-3	99.56%
T15658	KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific. It has IC50s of 3-10 μM toward both recombinant purified human sACt protein and heterologously exp...
T6426	Buclizine dihydrochloride	129-74-8	99.56%
T6426	Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and anti...
T2782	Catharanthine	2468-21-5	99.55%
T2782	Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).
TN3500	Beta-Amyrone	638-97-1	99.55%
TN3500	beta-Amyrone (β-Amyron) has antifungal activity against Chikungunya virus replication with an EC50 of 86 uM. beta-Amyrone has anti-inflammatory activity through ...
T23513	VU10010	633283-39-3	99.54%
T23513	VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.
T1328	DL-trihexyphenidyl hydrochloride	58947-95-8	99.53%
T1328	DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.
T22380	Nor-benzetimide	19315-71-0	99.53%
T22380	Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.