T8236 |
RHC 80267
|
83654-05-1
|
98%
|
|
RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)
|
T1519L |
Rimonabant
|
168273-06-1
|
98%
|
|
Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1. It is an anorectic anti-obesity drug produced and marketed by Sanofi-Aventis. Its m...
|
T0504 |
Cyclandelate
|
456-59-7
|
98%
|
|
Cyclandelate (BS 572), a direct-acting smooth muscle relaxant, is used to dilate blood vessels.
|
T73350 |
BAY-3827
|
2377576-35-5
|
100%
|
|
BAY-3827 is a potent and selective AMPK inhibitor with potential antitumor activity, showing antiproliferative activity in an androgen-dependent prostate cancer ...
|
T10035 |
10,12-Tricosadiynoic acid
|
66990-30-5
|
|
|
10,12-Tricosadiynoic acid is a highly selective and orally active inhibitor of acyl-CoA oxidase-1 (ACOX1). It can treat the high-fat diet- or obesity-induced met...
|
T11733 |
K-604 dihydrochloride
|
217094-32-1
|
98%
|
|
K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.
|
T23521 |
VULM 1457
|
228544-65-8
|
98%
|
|
VULM 1457 is a potent ACAT inhibitor. VULM 1457 has remarkable hypolipidaemic activity and improves the overall myocardial ischaemia-reperfusion injury outcomes....
|
T14523 |
Beauvericin
|
26048-05-5
|
98%
|
|
Beauvericin, a Fusarium mycotoxin, inhibits acyl-CoA:cholesterol acyltransferase (ACAT) in rat liver microsomal enzyme assays with an IC50 value of 3 μM.
|
T6365 |
A 922500
|
959122-11-3
|
98%
|
|
A 922500 (DGAT-1 Inhibitor 4a) is an inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively, good selectivity over related acyltransferas...
|
T5544 |
2-Furoic acid
|
88-14-2
|
98%
|
|
2-Furoic acid (Furan-2-carboxylic acid) 2-Furoic acid can reduce serum cholesterol and triglyceride levels and has anti-lipidemic effects.
|
T4681 |
T863
|
701232-20-4
|
98%
|
|
T-863(DGAT-1 inhibitor) is an orally active, selective and potent DGAT1 (Acyl-CoA:diacylglycerol acyltransferase 1) inhibitor that interacts with the acyl-CoA bi...
|
T13373 |
YM17E
|
124900-72-7
|
98%
|
|
YM17E is an inhibitor of ACAT with IC50 of 44 nM in rabbit liver microsomes in vitro.
|
T10503 |
ACAT-IN-1 cis isomer
|
145961-79-1
|
98%
|
|
ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.
|