Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T16158	PF-02575799	863491-70-7	98%
T16158	PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
TQ0136	GR79236	124555-18-6	98%
TQ0136	GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
T16281	Nelonicline	1026134-63-3	98%
T16281	Nelonicline is a selective agonist of neuronal nicotinic receptors.
T13008	ST3932	1246018-21-2	98%
T13008	ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
T11762	Kira8 Hydrochloride	2250019-92-0	98%
T11762	Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
T21620	2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine	133240-06-9	98%
T21620	2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine is an adenosine receptor antagonist.
T8613	1-Ethyl-6-aminouracil	41862-09-3	98%
T8613	1-Ethyl-6-aminouracil is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosi...
T10248	Adenosine antagonist-1	431040-19-6	98%
T10248	Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
T9180	LUF6096	1116652-18-6	98%
T9180	LUF6096 is a potent allosteric enhancer of the adenosine A3 receptor. LUF6096 is able to allosterically enhance agonist binding. LUF6096 shows low orthosteric af...
T0665	Xanthine	69-89-6	98%
T0665	Xanthine is a product on the pathway of purine degradation. Xanthine is subsequently converted to uric acid by the action of the Xanthine oxidase enzyme. Xanthin...
T27076	8-Cyclopentyl-1,3-dimethylxanthine	35873-49-5	98%
T27076	8-Cyclopentyl-1,3-dimethylxanthine is a potent antagonist of adenosine A1 receptor.
T14127	Adenosine A1 receptor activator T62	40312-34-3	98%
T14127	Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also r...
T23016	MRS1220	183721-15-5	98%
T23016	MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...
T27629	ISAM-140	932191-62-3	98%
T27629	ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
T16140	MRS 1754	264622-58-4	98%
T16140	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
T5081	Adenine monohydrochloride hemihydrate	6055-72-7	98%
T5081	Adenine is a high affinity adenine receptor agonist (Ki = 18 nM at rat adenine receptor). It inhibits forskolin-stimulated cAMP formation in CHO cells transfecte...
T23518	VUF 5574	280570-45-8	98%
T23518	VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.
T23535L	Xanthine amine congener trihydrochloride	2459963-12-1	98%
T23535L	Xanthine amine congener trihydrochloride is a potent adenosine antagonist that reverses the reduction in urine flow, sodium excretion and heart rate produced by ...
T16136	MRS-1706	264622-53-9	98%
T16136	MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B ...
T7320	Tozadenant	870070-55-6	98%
T7320	Tozadenant is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)