Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T37792	A2A receptor antagonist 1	443103-97-7	99.76%
T37792	A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
T6979	SCH 58261	160098-96-4	99.75%
T6979	SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.
T1825	Reversine	656820-32-5	99.75%
T1825	Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).
TN2247	Swertisin	6991-10-2	99.74%
TN2247	Swertisin, a novel herbal biomolecule, shows a strong antihyperglycemic action. Swertisin is an adenosine A1 receptor antagonist, is known to have antidiabetic, ...
T16378	Ogerin	1309198-71-7	99.7%
T16378	Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and a...
T27323	FK-453	121524-18-3	99.69%
T27323	FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.
T1083	Theophylline	58-55-9	99.65%
T1083	Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervo...
T28881	Sulmazole	73384-60-8	99.64%
T28881	Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.Sulma...
T28861	ST-1535	496955-42-1	99.64%
T28861	ST 1535 is a potent and orally active antagonist of A2A adenosine receptor with antiparkinsonian activity and antitremorigenic effects. ST 1535 exhibits the pote...
T14944	CGS 15943	104615-18-1	99.63%
T14944	CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Rec...
T4265	AZD4635	1321514-06-0	99.61%
T4265	AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).
T12159	APNEA	89705-21-5	99.58%
T12159	APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.
T2671	Regadenoson	313348-27-5	99.57%
T2671	Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadeno...
T10822	Cirsimarin	13020-19-4	99.55%
T10822	Cirsimarin (Cirsitakaoside) is a flavonoid isolated from Microtea debilis. It shows a potent antilipogenic effect and decreases adipose tissue deposition in mice...
T17117	Tonapofylline	340021-17-2	99.52%
T17117	Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about hea...
T4006	Pentostatin	53910-25-1	99.47%
T4006	Pentostatin (CI-825) is an extremely effective and irreversible inhibitor of adenosine deaminase (Ki: 2.5 pM).
T6884	Namodenoson	163042-96-4	99.4%
T6884	Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
T10248	Adenosine antagonist-1	431040-19-6	99.37%
T10248	Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
T28748	Selodenoson	110299-05-3	99.33%
T28748	Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.
T7736	2-Chloroadenosine	146-77-0	99.24%
T7736	2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively)...