Home Tools

Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T8551	Nitrobenzylthioinosine	38048-32-7	98.83%
T8551	Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
T6441	CGS 21680 Hydrochloride	124431-80-7	98.81%
T6441	CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.
T27800	LAS38096	851371-22-7	98.71%
T27800	LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .
T22234	Alloxazine	490-59-5	98.68%
T22234	Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.
T5S1895	Norisoboldine	23599-69-1	98.64%
T5S1895	1. Norisoboldine ((+)-Laurelliptine) might be a potential therapeutic agent for rheumatoid arthritis, and it functions through protecting joint destruction as we...
T6552	Istradefylline	155270-99-8	98.57%
T6552	Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in...
T26641L	Apadenoson TFA		98.40%
T26641L	Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
T12160	N6-Cyclohexyladenosine	36396-99-3	98.31%
T12160	N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm. N6-Cyclohexyladenosine exerts anticonvulsant effects and protects against...
T7683	Adenosine amine congener	96760-69-9	98.29%
T7683	Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
T6115	Fostamatinib	901119-35-5	98.24%
T6115	Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.
T22031	ANR 94	634924-89-3	98.21%
T22031	ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows ...
T8512	BAY-545	1699717-32-2	98.05%
T8512	BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).
T9238	KI-7	1489263-00-4	98.03%
T9238	KI-7 is an adenosine A2B receptor positive allosteric modulator.
T7183	CPI-444	1202402-40-1	98%
T7183	CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.
T7509	PD 117519	96392-15-3	98%
T7509	PD 117519 (CI947) is an agonist of adenosine receptor
T7340	5'-N-Ethylcarboxamidoadenosine	35920-39-9	98%
T7340	5'-N-Ethylcarboxamidoadenosine (NECA) is an agonist of Adenosine receptor, increases cerebral extravasation of fluorescein and low molecular weight dextran indep...
T39039	FSCPX	156547-56-7	98%
T39039	FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency. Additionally, FSCPX can ef...
T2373	Vipadenant	442908-10-3	98%
T2373	Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).
T16136	MRS-1706	264622-53-9	97.95%
T16136	MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B ...
T23535L	Xanthine amine congener trihydrochloride	2459963-12-1	97.85%
T23535L	Xanthine amine congener trihydrochloride is a potent adenosine antagonist that reverses the reduction in urine flow, sodium excretion and heart rate produced by ...