Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T21519	2-Chloro-N6-cyclopentyladenosine	37739-05-2	98%
2-Chloro-N6-cyclopentyladenosine is a potent and selective agonist of adenosine A1 receptor
T22744	DPCPX	102146-07-6	98%
DPCPX is an A1 adenosine receptor antagonist
T12163	N6-(2-Phenylethyl)adenosine	20125-39-7	98%
N6-(2-Phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.
T1681	Aminophylline	317-34-0	98%
Aminophylline is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.
T23336	SCH442416	316173-57-6	98%
SCH-442416 is an selective antagonist of adenosine A2A receptor. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 ...
T2205	Acefylline	652-37-9	98%
Theophylline-7-acetic acid, a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhydramine in the...
T1083	Theophylline	58-55-9	98%
Theophylline is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervous system stimulant act...
T0480	Doxofylline	69975-86-6	98%
Doxofylline is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofylline has shown...
T6745	5-Iodotubercidin	24386-93-4	98%
5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinase, phosphoryl...
T0362	Ticlopidine hydrochloride	53885-35-1	98%
Ticlopidine hydrochloride is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.
T12161	N6-Ethyladenosine	14357-08-5	98%
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).
T8598	CHEMBL241987	109740-09-2	98%
CHEMBL241987 targets the Adenosine receptor A3 (human)
T23203	PSB-603	1092351-10-4	98%
PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.
T37793	A2B receptor antagonist 2	784-90-7	98%
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T23535	Xanthine amine congener	96865-92-8	98%
Adenosine receptor antagonist

Cat. No.

Product name

CAS No.

Purity

Chemical Structure

T21519

2-Chloro-N6-cyclopentyladenosine

37739-05-2

98%

2-Chloro-N6-cyclopentyladenosine is a potent and selective agonist of adenosine A1 receptor

T22744

DPCPX

102146-07-6

98%

DPCPX is an A1 adenosine receptor antagonist

T12163

N6-(2-Phenylethyl)adenosine

20125-39-7

98%

N6-(2-Phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.

T1681

Aminophylline

317-34-0

98%

Aminophylline is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.

T23336

SCH442416

316173-57-6

98%

SCH-442416 is an selective antagonist of adenosine A2A receptor. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 ...

T2205

Acefylline

652-37-9

98%

Theophylline-7-acetic acid, a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhydramine in the...

T1083

Theophylline

58-55-9

98%

Theophylline is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervous system stimulant act...

T0480

Doxofylline

69975-86-6

98%

Doxofylline is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofylline has shown...

T6745

5-Iodotubercidin

24386-93-4

98%

5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinase, phosphoryl...

T0362

Ticlopidine hydrochloride

53885-35-1

98%